Publications by authors named "Giancarlo Fabrizi"

55Publications

Synthesis of pyrano[2,3-f]chromen-2-ones vs. pyrano[3,2-g]chromen-2-ones through site controlled gold-catalyzed annulations.

Org Biomol Chem 2019 12;17(47):10065-10072

Dipartimento di Scienze Fisiche e Chimiche Università degli Studi di L'Aquila, Via Vetoio, 67100 Coppito (AQ), Italy.

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December 2019

Stereo- and regioselective gold(i)-catalyzed hydroamination of 2-(arylethynyl)pyridines with anilines.

Org Biomol Chem 2019 01;17(3):527-532

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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January 2019

Identification of novel quinazoline derivatives as potent antiplasmodial agents.

Eur J Med Chem 2019 Jan 17;161:277-291. Epub 2018 Oct 17.

CIIL U1019-CNRS UMR 8204, Université de Lille, Institut Pasteur de Lille, 1 rue du Professeur Calmette, 59019, Lille, France. Electronic address:

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January 2019

Total Synthesis of (±)-Kuwanol E.

J Nat Prod 2016 10 22;79(10):2495-2503. Epub 2016 Sep 22.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma , p.le Aldo Moro 5, 00185 Roma, Italy.

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October 2016

Construction of the 1,5-Benzodiazepine Skeleton from o-Phenylendiamine and Propargylic Alcohols via a Domino Gold-Catalyzed Hydroamination/Cyclization Process.

Org Lett 2016 08 28;18(15):3511-3. Epub 2016 Jul 28.

Dipartimento di Chimica e Tecnologie del Farmaco, La Sapienza, Università di Roma , P.le A. Moro 5, 00185 Rome, Italy.

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August 2016

Pd- and Rh-Catalyzed Hydroarylation of γ-(2-Methoxycarbonylphenyl)propargylic Alcohols: Approaches to 4- or 5-Substituted Seven-Membered Benzolactones and 3,3-Disubstituted Phthalides.

J Org Chem 2015 Jul 6;80(14):6986-95. Epub 2015 Jul 6.

†Dipartimento di Scienze Fisiche e Chimiche, Università di L'Aquila, Via Vetoio - 67010 Coppito (AQ), Italy.

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July 2015

Palladium-catalyzed synthesis of 2-(aminomethyl)indoles from 3-(o-trifluoroacetamidoaryl)-1-propargylic alcohols and amines.

J Org Chem 2014 Jan 18;79(1):401-7. Epub 2013 Dec 18.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma , P.le A. Moro 5, 00185 Rome, Italy.

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January 2014

New entry to polycyclic fused indoles via gold(I)-catalyzed cascade reaction.

Chem Asian J 2013 Aug 14;8(8):1776-9. Epub 2013 Mar 14.

Department of Chemistry G. Ciamician, Alma Mater Studiorum-University of Bologna, via Selmi 2, 40138 Bologna, Italy.

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August 2013

Palladium-catalyzed cascade reactions of 1-(3-arylprop-2-ynyloxy)-2-bromo benzene derivatives with organoboron compounds.

J Org Chem 2013 May 22;78(9):4490-8. Epub 2013 Apr 22.

Dipartimento di Scienze Fisiche e Chimiche, Università di L'Aquila, Via Vetoio, 67010, Coppito (AQ), Italy.

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May 2013

2-Substituted 3-arylindoles through palladium-catalyzed arylative cyclization of 2-alkynyltrifluoroacetanilides with arylboronic acids under oxidative conditions.

Org Biomol Chem 2013 Jan 6;11(4):545-8. Epub 2012 Dec 6.

Dipartimento di Scienze Fisiche e Chimiche, Università degli Studi di L'Aquila, Via Vetoio, 67010 Coppito, L'Aquila, Italy.

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January 2013

Gold versus silver catalyzed intramolecular hydroarylation reactions of [(3-arylprop-2-ynyl)oxy]benzene derivatives.

Org Biomol Chem 2012 Dec 13;10(48):9700-8. Epub 2012 Nov 13.

Dipartimento di Scienze Fisiche e Chimiche, Università degli Studi di L'Aquila, Via Vetoio, 67010 Coppito, L'Aquila, Italy.

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December 2012

Dibenzo[a,c]carbazoles from 2-(2-bromoaryl)-3-arylindoles via a palladium-catalyzed intramolecular C-H functionalization/C-C bond formation process.

Org Biomol Chem 2012 Dec 29;10(46):9142-7. Epub 2012 Oct 29.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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December 2012

One-pot gold-catalyzed synthesis of azepino[1,2-a]indoles.

Angew Chem Int Ed Engl 2012 Sep 3;51(39):9891-5. Epub 2012 Sep 3.

Dipartimento di Chimica G. Ciamician, Alma Mater Studiorum-Università di Bologna, Bologna, Italy.

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September 2012

Palladium-catalyzed synthesis of 2-amino ketones from propargylic carbonates and secondary amines.

Org Biomol Chem 2012 Jun 18;10(24):4699-703. Epub 2012 May 18.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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June 2012