Publications by authors named "Wael Zeinyeh"

17Publications

Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies.

Bioorg Med Chem 2019 05 4;27(10):2083-2089. Epub 2019 Apr 4.

Université Clermont Auvergne, CNRS, SIGMA Clermont, ICCF, F-63000 Clermont-Ferrand, France. Electronic address:

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May 2019

6-Chloropurine Ribonucleosides from Chloropyrimidines: One-Pot Synthesis.

Curr Protoc Nucleic Acid Chem 2018 09 13;74(1):e57. Epub 2018 Aug 13.

Université Grenoble Alpes, CNRS, DPM, Grenoble, France.

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September 2018

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α-Synuclein PET Imaging.

Mol Pharm 2018 08 25;15(8):3153-3166. Epub 2018 Jul 25.

Université de Lyon, Université Claude Bernard Lyon 1, Lyon Neuroscience Research Center, CNRS UMR5292, INSERM U1028 , Lyon 69361 , France.

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August 2018

Amyloid-Beta Radiotracer [F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue.

Contrast Media Mol Imaging 2018 6;2018:9165458. Epub 2018 Feb 6.

Lyon Neuroscience Research Center, CNRS UMR5292, INSERM U1028, Université Claude Bernard Lyon 1, Université de Lyon, Lyon, France.

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July 2019

A One-Pot Synthesis of Highly Functionalized Purines.

Org Lett 2017 12 10;19(23):6360-6363. Epub 2017 Nov 10.

Univ. Grenoble Alpes , CNRS, DPM, 38000 Grenoble, France.

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December 2017

Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives.

Bioorg Med Chem Lett 2016 09 16;26(17):4327-9. Epub 2016 Jul 16.

Université Clermont Auvergne, Université Blaise Pascal, Institut de Chimie de Clermont-Ferrand, BP 10448, F-63000 Clermont-Ferrand, France; CNRS, UMR 6296, ICCF, F-63178 Aubière, France. Electronic address:

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September 2016

Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.

Eur J Med Chem 2016 Aug 5;118:170-7. Epub 2016 Apr 5.

Université Clermont Auvergne, Université Blaise Pascal, Institut de Chimie de Clermont-Ferrand, BP 10448, F-63000 Clermont-Ferrand, France; CNRS, UMR 6296, ICCF, F-63178 Aubière, France. Electronic address:

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August 2016

Inverse relationship between hSHBG affinity for testosterone and hSHBG concentration revealed by surface plasmon resonance.

Mol Cell Endocrinol 2015 Jan 13;399:201-7. Epub 2014 Oct 13.

Université de Lyon, Lyon F-69000, France; ISPB Faculté de Pharmacie, MATEIS CNRS UMR5510, Université Claude Bernard Lyon-1, 8 Avenue Rockefeller, cedex 08, Lyon F-69373, France; Hôpital Edouard Herriot, Laboratoire de Biochimie et de Biologie Moléculaire, Hospices Civils de Lyon, cedex 03, Lyon 69437, France.

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January 2015

Preparation and characterization of CK2 inhibitor-loaded cyclodextrin nanoparticles for drug delivery.

Int J Pharm 2013 Jan 13;441(1-2):491-8. Epub 2012 Nov 13.

Université de Lyon, Université Lyon 1, CSAp, Institut de Chimie et Biochimie Moléculaires et Supramoléculaires, Bâtiment Raulin, 43 Bd du 11 novembre 1918, 69622 Villeurbanne Cedex, France.

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January 2013

Progesterone-adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: design, synthesis, characterization and biological evaluation.

Steroids 2012 Oct 31;77(12):1177-91. Epub 2012 Jul 31.

Université de Lyon, Université Lyon 1, EA 4446 Biomolécules Cancer Chimiorésistances (B2C), ISPB-Faculté de Pharmacie, UMS 3453 Santé Lyon-Est, 8 Avenue Rockefeller, F-69373 Lyon Cedex 08, France.

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October 2012

Design, synthesis and evaluation of progesterone-adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux.

Bioorg Med Chem Lett 2010 May 28;20(10):3165-8. Epub 2010 Mar 28.

Université de Lyon, Université Lyon 1, ISPB-Faculté de Pharmacie, INSERM U863, F-69373 Lyon cedex 08, France.

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May 2010

Synthesis and modulation properties of imidazo[4,5-b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter.

Eur J Med Chem 2010 Jun 18;45(6):2480-8. Epub 2010 Feb 18.

Université de Lyon, Université Lyon 1, ISPB-Faculté de Pharmacie, EA 4443 (B2C) Biomolécules, Cancer et Chimiorésistances, 8, av. Rockefeller, F-69373, Lyon Cedex 08, France.

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June 2010