Publications by authors named "Vincent Bordas"

9Publications

Potent achiral agonists of the ghrelin (growth hormone secretagogue) receptor. Part I: Lead identification.

Bioorg Med Chem Lett 2007 Dec 25;17(23):6584-7. Epub 2007 Sep 25.

Department of Medicinal Chemistry & DMPK, Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

View Article and Find Full Text PDF
December 2007

Pyridone derivatives as potent, orally bioavailable VLA-4 integrin antagonists.

Bioorg Med Chem Lett 2006 Nov 22;16(21):5538-41. Epub 2006 Aug 22.

Department of DMPK and Medicinal Chemistry, Neurology and GI Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

View Article and Find Full Text PDF
November 2006

Pyridone derivatives as potent and selective VLA-4 integrin antagonists.

Bioorg Med Chem Lett 2006 Apr 7;16(8):2256-9. Epub 2006 Feb 7.

Department of Medicinal Chemistry, Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Harlow, Essex, CM19 5AW, UK.

View Article and Find Full Text PDF
April 2006

6-heteroaryl-pyrazolo[3,4-b]pyridines: potent and selective inhibitors of glycogen synthase kinase-3 (GSK-3).

Bioorg Med Chem Lett 2003 Sep;13(18):3059-62

Department of Medicinal Chemistry, Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

View Article and Find Full Text PDF
September 2003

6-aryl-pyrazolo[3,4-b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3).

Bioorg Med Chem Lett 2003 Sep;13(18):3055-7

Department of Medicinal Chemistry, Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

View Article and Find Full Text PDF
September 2003

5-aryl-pyrazolo[3,4-b]pyridazines: potent inhibitors of glycogen synthase kinase-3 (GSK-3).

Bioorg Med Chem Lett 2003 May;13(9):1581-4

Department of Medicinal Chemistry, Neurology Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Essex CM19 5AW, Harlow, UK.

View Article and Find Full Text PDF
May 2003

5-aryl-pyrazolo[3,4-b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3).

Bioorg Med Chem Lett 2003 May;13(9):1577-80

Department of Medicinal Chemistry, Neurology Centre of Excellence for Drug Discovery, GlaxoSmithKline Research Limited, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

View Article and Find Full Text PDF
May 2003