Publications by authors named "Thierry Cresteil"

68Publications

Targeting prohibitin with small molecules to promote melanogenesis and apoptosis in melanoma cells.

Eur J Med Chem 2018 Jul 23;155:880-888. Epub 2018 Jun 23.

Laboratory of Therapeutic Innovation (UMR 7200), CNRS/University of Strasbourg, Faculty of Pharmacy, Illkirch, France; Laboratory of Biomolecules (UMR7203), Sorbonne University-CNRS, 4 Place Jussieu, 75005, Paris, France; Sino-French Joint Lab of Food Nutrition/Safety and Medicinal Chemistry, College of Biotechnology, Tianjin University of Science and Technology, Tianjin, China. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2018.06.052DOI Listing
July 2018

First-in-Class Combination Therapy of a Copper(II) Metallo-Phosphorus Dendrimer with Cytotoxic Agents.

Oncology 2018 13;94(5):324-328. Epub 2018 Mar 13.

Laboratoire de Chimie de Coordination CNRS, Toulouse, France.

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http://dx.doi.org/10.1159/000486680DOI Listing
May 2018

Anticancer copper(II) phosphorus dendrimers are potent proapoptotic Bax activators.

Eur J Med Chem 2017 May 21;132:142-156. Epub 2017 Mar 21.

ICSN-CNRS UPR 2301, Avenue de la Terrasse, 91198 Gif sur Yvette, France; IPSIT, Faculté de Pharmacie, Université Paris Sud, 92290 Chatenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2017.03.035DOI Listing
May 2017

A novel class of ethacrynic acid derivatives as promising drug-like potent generation of anticancer agents with established mechanism of action.

Eur J Med Chem 2016 Oct 11;122:656-673. Epub 2016 Jun 11.

Laboratoire de Chimie de Coordination CNRS, 205 route de Narbonne, BP 44099, 31077, Toulouse Cedex 4, France; Université de Toulouse, UPS, INPT, F-31077, Toulouse Cedex4, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2016.05.063DOI Listing
October 2016

Novel benzylidenephenylpyrrolizinones with pleiotropic activities potentially useful in Alzheimer's disease treatment.

Eur J Med Chem 2016 May 12;114:365-79. Epub 2016 Mar 12.

Normandie Université, UNICAEN, CERMN (Centre d'Etudes et de Recherche sur le Médicament de Normandie), F-14032 Caen, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2016.03.023DOI Listing
May 2016

Antidiabetic potential of two medicinal plants used in Gabonese folk medicine.

BMC Complement Altern Med 2016 Feb 22;16:71. Epub 2016 Feb 22.

Institut des Biomolécules Max Mousseron (IBMM) UMR 5247 CNRS-Université Montpellier-ENSCM, Bâtiment E, Faculté de Pharmacie, 15, avenue Charles Flahault BP14491, 34093, Montpellier, cedex 5, France.

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http://dx.doi.org/10.1186/s12906-016-1052-xDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4763413PMC
February 2016

Boronic species as promising inhibitors of the Staphylococcus aureus NorA efflux pump: study of 6-substituted pyridine-3-boronic acid derivatives.

Eur J Med Chem 2015 May 2;95:185-98. Epub 2015 Mar 2.

Normandie Univ, France; UNICAEN, CERMN (Centre d'Etudes et de Recherche sur le Médicament de Normandie) - FR CNRS INC3M, Boulevard Becquerel, 14032 Caen, France.

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https://linkinghub.elsevier.com/retrieve/pii/S02235234150015
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http://dx.doi.org/10.1016/j.ejmech.2015.02.056DOI Listing
May 2015

Synthesis of 2,3-di- and 2,2,3-trisubstituted-3-methoxycarbonyl-γ-butyrolactones as potent antitumor agents.

Eur J Med Chem 2015 Jan 28;89:654-70. Epub 2014 Oct 28.

Ciblothèque cellulaire, Institut de Chimie des Substances Naturelles, CNRS-UPR 2301, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1016/j.ejmech.2014.10.074DOI Listing
January 2015

α-Glucosidase inhibitory activity of marine sponges collected in Mauritius waters.

Nat Prod Res 2015 13;29(4):383-7. Epub 2014 Aug 13.

a Mauritius Oceanography Institute (MOI) , France Centre, Victoria Avenue, Quatre-Bornes , Mauritius.

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http://www.tandfonline.com/doi/abs/10.1080/14786419.2014.945
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http://dx.doi.org/10.1080/14786419.2014.945173DOI Listing
April 2015

Design, synthesis and biological evaluation of Pontin ATPase inhibitors through a molecular docking approach.

Bioorg Med Chem Lett 2014 Jun 13;24(11):2512-6. Epub 2014 Apr 13.

Université de Bordeaux, CNRS UMR 5248, CBMN, IECB, 2 rue Robert Escarpit, 33607 Pessac, France. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2014.04.003DOI Listing
June 2014

A concise formation of N-substituted 3,4-diarylpyrroles--synthesis and cytotoxic activity.

Org Biomol Chem 2014 Mar;12(9):1518-24

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1039/c3ob42309cDOI Listing
March 2014

Synthesis and evaluation of cytotoxic activities of new guanidines derived from carbazoles.

Bioorg Med Chem Lett 2014 Jan 17;24(2):467-72. Epub 2013 Dec 17.

Université de Caen Basse-Normandie, Centre d'Etudes et de Recherche sur le Médicament de Normandie UPRES EA 4258 - FR CNRS 3038 INC3M, Bd Becquerel, 14032 Caen Cedex, France.

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http://dx.doi.org/10.1016/j.bmcl.2013.12.047DOI Listing
January 2014

Synthesis and evaluation of 3-deoxy and 3-deoxy-3-fluoro derivatives of gluco- and manno-configured tetrahydropyridoimidazole glycosidase inhibitors.

Carbohydr Res 2013 Aug 21;377:35-43. Epub 2013 May 21.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette, France.

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http://dx.doi.org/10.1016/j.carres.2013.05.011DOI Listing
August 2013

The cytosolic chaperonin CCT/TRiC and cancer cell proliferation.

PLoS One 2013 16;8(4):e60895. Epub 2013 Apr 16.

Laboratoire d'Enzymologie et Biochimie Structurales, CNRS, Gif-sur-Yvette, France.

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http://journals.plos.org/plosone/article?id=10.1371/journal.pone.0060895PLOS
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3628893PMC
November 2013

Ethyl acetate extract of the Mauritian sponge Jaspis sp. induces cell arrest in human promyelocytic leukemia cells.

Environ Toxicol Pharmacol 2013 Jul 15;36(1):58-65. Epub 2013 Mar 15.

Mauritius Oceanography Institute, Quatre-Bornes, Mauritius.

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http://dx.doi.org/10.1016/j.etap.2013.03.002DOI Listing
July 2013

Original multivalent copper(II)-conjugated phosphorus dendrimers and corresponding mononuclear copper(II) complexes with antitumoral activities.

Mol Pharm 2013 Apr 7;10(4):1459-64. Epub 2013 Mar 7.

Institute of Nanomaterials & Nanotechnology, Moroccan Advanced Science, Innovation and Research Foundation, Avenue de l'Armée Royale, Madinat El Irfane, 10100, Rabat, Morocco.

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http://dx.doi.org/10.1021/mp4000184DOI Listing
April 2013

MR22388, a novel anti-cancer agent with a strong FLT-3 ITD kinase affinity.

Cancer Lett 2013 Apr 23;331(1):92-8. Epub 2012 Dec 23.

CERMN, UFR des Sciences Pharmaceutiques, UPRES EA 4258 - FR CNRS 3038 INC3M - SF 4206 ICORE, Université de Caen Basse-Normandie, Bd Becquerel, 14032 Caen cedex, France.

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https://linkinghub.elsevier.com/retrieve/pii/S03043835120073
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http://dx.doi.org/10.1016/j.canlet.2012.12.017DOI Listing
April 2013

N-O bond as a glycosidic-bond surrogate: synthetic studies toward polyhydroxylated N-alkoxypiperidines.

Chemistry 2013 Feb 19;19(6):2168-79. Epub 2012 Dec 19.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette, France.

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http://dx.doi.org/10.1002/chem.201202374DOI Listing
February 2013

Flavaglines as potent anticancer and cytoprotective agents.

J Med Chem 2012 Nov 23;55(22):10064-73. Epub 2012 Oct 23.

Therapeutic Innovation Laboratory, UMR7200, CNRS/Université de Strasbourg, Illkirch, France.

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http://dx.doi.org/10.1021/jm301201zDOI Listing
November 2012

Cytotoxic activities of hexane, ethyl acetate and butanol extracts of marine sponges from Mauritian Waters on human cancer cell lines.

Environ Toxicol Pharmacol 2012 Sep 9;34(2):397-408. Epub 2012 Jun 9.

Mauritius Oceanography Institute, France Centre, Quatre-Bornes, Mauritius. Electronic address:

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http://dx.doi.org/10.1016/j.etap.2012.05.013DOI Listing
September 2012

Synthesis of novel 7-oxo and 7-hydroxy trifluoroallocolchicinoids with cytotoxic effect.

Bioorg Med Chem 2012 Apr 3;20(8):2614-23. Epub 2012 Mar 3.

Université de Caen Basse Normandie, Centre d'Etudes et de Recherche sur le Médicament de Normandie UPRES EA 4258 - FR CNRS 3038 INC3M, UFR des Sciences Pharmaceutiques, Bd Becquerel, 14032 Caen cedex, France.

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http://dx.doi.org/10.1016/j.bmc.2012.02.043DOI Listing
April 2012

Pipestelides A-C: cyclodepsipeptides from the Pacific marine sponge Pipestela candelabra.

J Nat Prod 2012 Apr 24;75(4):759-63. Epub 2012 Feb 24.

Centre de Recherche de Gif-sur-Yvette, Institut de Chimie des Substances Naturelles, UPR 2301, ICSN-CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette, France.

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http://dx.doi.org/10.1021/np200714mDOI Listing
April 2012

Synthesis and biological investigation of the β-thiolactone and β-lactam analogs of tetrahydrolipstatin.

Org Biomol Chem 2012 Apr 21;10(13):2629-32. Epub 2012 Feb 21.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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http://dx.doi.org/10.1039/c2ob06976hDOI Listing
April 2012

Synthesis and biological evaluation of acridine derivatives as antimalarial agents.

ChemMedChem 2012 Apr 13;7(4):587-605. Epub 2012 Feb 13.

Université Paris-Sud 11, Institut de Chimie Moléculaire et des Matériaux d'Orsay, Equipe de Chimie Bioorganique et Bioinorganique, Orsay 91405 CEDEX, France.

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http://dx.doi.org/10.1002/cmdc.201100554DOI Listing
April 2012

Influence of the skeleton on the cytotoxicity of flavonoids.

Bioorg Med Chem 2012 Feb 30;20(3):1231-9. Epub 2011 Dec 30.

Laboratoire de Pharmacognosie, (Univ. Paris-Sud 11, BIOCIS, UMR-8076 CNRS), Faculté de Pharmacie, av. J.B. Clément, 92296 Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1016/j.bmc.2011.12.038DOI Listing
February 2012

Synthesis and cytotoxic evaluation of novel paraconic acid analogs.

Bioorg Med Chem Lett 2011 Dec 29;21(23):7054-8. Epub 2011 Sep 29.

Électrochimie et Synthèse Organique, Institut de Chimie et des Matériaux Paris-Est, UMR 7182 CNRS-Université Paris-Est Créteil, Thiais, France.

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http://dx.doi.org/10.1016/j.bmcl.2011.09.092DOI Listing
December 2011

Exploring the potential of the β-thiolactones in bioorganic chemistry.

Org Biomol Chem 2011 Oct 2;9(20):7134-43. Epub 2011 Sep 2.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190, Gif-sur-Yvette, France.

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http://dx.doi.org/10.1039/c1ob05967jDOI Listing
October 2011

Swinholide J, a potent cytotoxin from the marine sponge Theonella swinhoei.

Mar Drugs 2011 22;9(6):1133-41. Epub 2011 Jun 22.

Department of Chemistry of Natural Compounds, University of Naples, Federico II, via D. Montesano 49, 80131 Napoli, Italy.

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http://dx.doi.org/10.3390/md9061133DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3131564PMC
January 2012

Bioactive indole derivatives from the South Pacific marine sponges Rhopaloeides odorabile and Hyrtios sp.

Mar Drugs 2011 24;9(5):879-88. Epub 2011 May 24.

Laboratoire Molécules de Communication et Adaptation des Micro-organismes, UMR 7245 MNHN-CNRS, Muséum National d'Histoire Naturelle, 57 Rue Cuvier (C.P. 54), 75005 Paris, France.

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http://dx.doi.org/10.3390/md9050879DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3111189PMC
November 2011

Design, synthesis and antiproliferative activities of biarylolefins based on polyhydroxylated and carbohydrate scaffolds.

Eur J Med Chem 2011 Sep 13;46(9):3570-80. Epub 2011 May 13.

UMR 7565 SRSMC, Nancy Université-CNRS, Groupe SUCRES, BP 239, F-54506 Nancy Vandœuvre, France.

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http://dx.doi.org/10.1016/j.ejmech.2011.05.021DOI Listing
September 2011

Investigation of a series of silver-N-heterocyclic carbenes as antibacterial agents: activity, synergistic effects, and cytotoxicity.

Chemistry 2011 Feb 5;17(5):1442-6. Epub 2011 Jan 5.

Institut Parisien de Chimie Moléculaire, UMR CNRS 7201, Université Pierre et Marie Curie, Paris 6, 4, place Jussieu, 75252 Paris CEDEX 05, France.

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http://dx.doi.org/10.1002/chem.201002812DOI Listing
February 2011

Synthesis of antiproliferative flavones from calycopterin, major flavonoid of Calycopteris floribunda Lamk.

Bioorg Med Chem 2011 Jan 20;19(1):186-96. Epub 2010 Nov 20.

Laboratoire de Pharmacognosie, (Univ. Paris-Sud 11, BIOCIS, UMR-8076 CNRS), Faculté de Pharmacie, Av. J.B. Clément, 92296 Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1016/j.bmc.2010.11.035DOI Listing
January 2011

Novel flavaglines displaying improved cytotoxicity.

J Med Chem 2011 Jan 13;54(1):411-5. Epub 2010 Dec 13.

Therapeutic Innovation Laboratory (UMR 7200), Department of Medicinal Chemistry, Faculté de Pharmacie, CNRS-Université de Strasbourg, Illkirch, France.

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http://dx.doi.org/10.1021/jm101318bDOI Listing
January 2011

Semisynthesis of natural flavones inhibiting tubulin polymerization, from hesperidin.

J Nat Prod 2010 Apr;73(4):702-6

Laboratoire de Pharmacognosie, Faculte de Pharmacie, Universite Paris-Sud 11 BIOCIS UMR-8076 CNRS, Avenue J.B. Clement, 92296 Chatenay-Malabry Cedex, France.

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http://dx.doi.org/10.1021/np100065vDOI Listing
April 2010

Hydrogenative desulphurization of thienopyrrolizinones: an easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity.

Eur J Med Chem 2010 Mar 21;45(3):1146-50. Epub 2009 Dec 21.

Centre d'Etudes et de Recherche sur le Médicament de Normandie, UPRES EA 4258, FR CNRS 3038 INC3M UFR des Sciences Pharmaceutiques, Université de Caen Basse Normandie, Bd Becquerel, 14032 Caen cedex France.

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http://dx.doi.org/10.1016/j.ejmech.2009.12.021DOI Listing
March 2010

Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin.

Bioorg Med Chem 2009 Dec 9;17(23):8032-9. Epub 2009 Oct 9.

Equipe de Chimie Bioorganique et Bioinorganique, Institut de Chimie Moléculaire et des Matériaux d'Orsay, Bât. 420, CNRS UMR 8182, Univ Paris-Sud, 91405 Orsay Cedex, France.

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http://dx.doi.org/10.1016/j.bmc.2009.10.005DOI Listing
December 2009

Synthesis, reactivity and biological evaluation of novel halogenated tripentones.

Bioorg Med Chem 2009 Nov 19;17(22):7783-8. Epub 2009 Sep 19.

Centre d'Etudes et de Recherche sur le Médicament de Normandie (UPRES EA 4258-FR CNRS 3038 INC3M), UFR des Sciences Pharmaceutiques, Université de Caen Basse-Normandie, Boulevard Becquerel, 14032 Caen cedex, France.

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http://dx.doi.org/10.1016/j.bmc.2009.09.027DOI Listing
November 2009

Metabolism of sanguinarine in human and in rat: characterization of oxidative metabolites produced by human CYP1A1 and CYP1A2 and rat liver microsomes using liquid chromatography-tandem mass spectrometry.

J Pharm Biomed Anal 2010 Jul 16;52(3):391-7. Epub 2009 Sep 16.

Institut de cancérologie Gustave Roussy, Research Department IFR54, Mass Spectrometry Facility, 39 rue Camille Desmoulins, 94805 Villejuif Cedex, France.

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http://dx.doi.org/10.1016/j.jpba.2009.09.014DOI Listing
July 2010

Homophymines B-E and A1-E1, a family of bioactive cyclodepsipeptides from the sponge Homophymia sp.

Org Biomol Chem 2009 Oct 22;7(19):4037-44. Epub 2009 Jul 22.

Dipartimento di Chimica delle Sostanze Naturali, Università di Napoli Federico II, via D. Montesano 49, 80131, Napoli, Italy.

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http://dx.doi.org/10.1039/b910015fDOI Listing
October 2009

Semisynthesis and antiproliferative evaluation of a series of 3'-aminoflavones.

Bioorg Med Chem Lett 2009 Jul 7;19(13):3502-6. Epub 2009 May 7.

Laboratoire de Pharmacognosie, (Univ. Paris-Sud 11, BIOCIS, UMR-8076 CNRS), Faculté de Pharmacie, av. J.B. Clément, 92296 Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1016/j.bmcl.2009.05.008DOI Listing
July 2009

Synthesis and biological evaluation of a series of tangeretin-derived chalcones.

Bioorg Med Chem Lett 2009 Jan 5;19(1):167-9. Epub 2008 Nov 5.

Faculté de Pharmacie, Laboratoire de Pharmacognosie, Univ Paris-Sud 11, BIOCIS, UMR-8076 CNRS, Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1016/j.bmcl.2008.10.126DOI Listing
January 2009

Discovery and refinement of a new structural class of potent peptide deformylase inhibitors.

J Med Chem 2007 Jan;50(1):10-20

UPR2355, Centre National de la Recherche Scientifique, Bâtiment 23, 1 Avenue de la Terrasse, F-91198 Gif-Sur-Yvette Cedex, France.

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http://dx.doi.org/10.1021/jm060910cDOI Listing
January 2007

In vitro oxidative metabolism study of (-)-rhazinilam.

Bioorg Med Chem 2006 Mar 27;14(5):1558-64. Epub 2005 Oct 27.

Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette, France.

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http://dx.doi.org/10.1016/j.bmc.2005.10.015DOI Listing
March 2006

CYP3A5 mRNA degradation by nonsense-mediated mRNA decay.

Mol Pharmacol 2005 Sep 13;68(3):808-15. Epub 2005 Jun 13.

ICSN, CNRS UPR2301, Avenue de la Terrasse, 91198 Gif-sur-Yvette, France.

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http://dx.doi.org/10.1124/mol.105.014225DOI Listing
September 2005

Phenotyping-genotyping of alternatively spliced genes in one step: study of CYP3A5*3 polymorphism.

Pharmacogenet Genomics 2005 Jun;15(6):433-9

ICSN--CNRS UPR2301, 91198 Gif-sur-Yvette, France.

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http://dx.doi.org/10.1097/01213011-200506000-00010DOI Listing
June 2005

In vitro metabolism study of buprenorphine: evidence for new metabolic pathways.

Drug Metab Dispos 2005 May 2;33(5):689-95. Epub 2005 Mar 2.

Department of Medical Pharmacology, University of Limoges, France.

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http://dx.doi.org/10.1124/dmd.105.003681DOI Listing
May 2005

Characterization of a phase 1 metabolite of mycophenolic acid produced by CYP3A4/5.

Ther Drug Monit 2004 Dec;26(6):600-8

Department of Pharmacology and Toxicology, University Hospital, 87042 Limoges, France.

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http://dx.doi.org/10.1097/00007691-200412000-00004DOI Listing
December 2004

Dexamethasone as a probe for docetaxel clearance.

Cancer Chemother Pharmacol 2004 Sep 5;54(3):265-72. Epub 2004 May 5.

Institut Claudius-Regaud, Université Paul-Sabatier, 31052 Toulouse, France.

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http://dx.doi.org/10.1007/s00280-004-0823-0DOI Listing
September 2004

Quantitative liquid chromatographic determination of sanguinarine in cell culture medium and in rat urine and plasma.

J Chromatogr B Analyt Technol Biomed Life Sci 2004 Jan;799(2):195-200

CNRS UPR 2301, Institut de Chimie des Substances Naturelles, Avenue de la Terrasse, 91198 Cedex, Gif sur Yvette, France.

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http://dx.doi.org/10.1016/j.jchromb.2003.10.023DOI Listing
January 2004

Downregulation of cytochromes P450 in growth-stimulated rat hepatocytes: role of c-Myc induction and impaired C/EBP binding to DNA.

J Hepatol 2003 Aug;39(2):171-8

Institut National de la Santé et de la Recherche Médicale (INSERM) Unité 481, Faculté de Médecine Xavier Bichat, 16 rue Henri Huchard, 75018, Paris, France.

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http://dx.doi.org/10.1016/s0168-8278(03)00238-1DOI Listing
August 2003

Regioselective metabolism of taxoids by human CYP3A4 and 2C8: structure-activity relationship.

Drug Metab Dispos 2002 Apr;30(4):438-45

Centre National de la Recherche Scientifique Unité Mixte Recherche 8532, Villejuif, France.

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http://dx.doi.org/10.1124/dmd.30.4.438DOI Listing
April 2002