Publications by authors named "Thierry Billard"

58Publications

Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate.

Beilstein J Org Chem 2020 10;16:3032-3037. Epub 2020 Dec 10.

Institute of Chemistry and Biochemistry (ICBMS-UMR CNRS 5246), Univ Lyon, Université Lyon 1, CNRS, CPE, INSA, 43 Bd du 11 novembre 1918, 69622 Villeurbanne, France.

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December 2020

Preclinical validation of [F]2FNQ1P as a specific PET radiotracer of 5-HT receptors in rat, pig, non-human primate and human brain tissue.

Nucl Med Biol 2020 Mar - Apr;82-83:57-63. Epub 2020 Jan 22.

Lyon Neuroscience Research Center, Université de Lyon, CNRS, INSERM, Lyon, France; Hospices Civils de Lyon, Bron, France; CERMEP Imaging Platform, Bron, France.

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January 2020

Difluoro(aryl)(perfluoroalkyl)-λ -sulfanes and Selanes: Missing Links of Trichloroisocyanuric Acid/Potassium Fluoride Chemistry.

Angew Chem Int Ed Engl 2019 12 18;58(52):18937-18941. Epub 2019 Nov 18.

Department of Chemistry and Applied Biosciences, ETH Zürich, Vladimir-Prelog-Weg 2, 8093, Zürich, Switzerland.

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December 2019

Chalcogen OCF Isosteres Modulate Drug Properties without Introducing Inherent Liabilities.

ChemMedChem 2019 09 21;14(17):1586-1589. Epub 2019 Aug 21.

Novartis Institutes for BioMedical Research, 181 Massachusetts Avenue, Cambridge, MA, 02139, USA.

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September 2019

Merging Visible-Light Catalysis for the Direct Late-Stage Group-16-Trifluoromethyl Bond Formation.

Chemistry 2019 May 22;25(26):6482-6495. Epub 2019 Feb 22.

Institute of Chemistry and Biochemistry (ICBMS-UMR, CNRS 5246), Univ Lyon, Université Lyon 1, CNRS, CPE-Lyon, INSA, 43 Bd du 11 Novembre 1918, 69622, Villeurbanne, France.

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May 2019

Evaluation of [ F]2FP3 in pigs and non-human primates.

J Labelled Comp Radiopharm 2019 01 6;62(1):34-42. Epub 2018 Dec 6.

Neurobiology Research Unit and Center for Integrated Molecular Brain Imaging, Copenhagen University Hospital, Rigshospitalet, Copenhagen, Denmark.

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January 2019

Visible-light promoted fluoroalkylselenolation: toward the reactivity of unsaturated compounds.

Chem Commun (Camb) 2018 Sep 14;54(71):9909-9912. Epub 2018 Aug 14.

Institute of Chemistry and Biochemistry (ICBMS - UMR CNRS 5246), Unvi. Lyon, Université Lyon 1, CNRS, 43 Bd du 11 novembre 1918, F-69622 Villeurbanne, France.

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September 2018

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α-Synuclein PET Imaging.

Mol Pharm 2018 08 25;15(8):3153-3166. Epub 2018 Jul 25.

Université de Lyon, Université Claude Bernard Lyon 1, Lyon Neuroscience Research Center, CNRS UMR5292, INSERM U1028 , Lyon 69361 , France.

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August 2018

Visible-Light-Mediated Metal-Free Synthesis of Trifluoromethylselenolated Arenes.

Angew Chem Int Ed Engl 2018 Sep 1;57(36):11781-11785. Epub 2018 Aug 1.

Institute of Chemistry and Biochemistry (ICBMS-UMR, CNRS 5246), Univ Lyon, Université Lyon 1, CNRS, CPE-Lyon, INSA, 43 Bd du 11 Novembre 1918, 69622, Villeurbanne, France.

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September 2018

Amyloid-Beta Radiotracer [F]BF-227 Does Not Bind to Cytoplasmic Glial Inclusions of Postmortem Multiple System Atrophy Brain Tissue.

Contrast Media Mol Imaging 2018 6;2018:9165458. Epub 2018 Feb 6.

Lyon Neuroscience Research Center, CNRS UMR5292, INSERM U1028, Université Claude Bernard Lyon 1, Université de Lyon, Lyon, France.

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July 2019

Electrophilic trifluoromethylselenolation of terminal alkynes with -(trifluoromethyl) 4-methylbenzenesulfonoselenoate.

Beilstein J Org Chem 2017 7;13:2626-2630. Epub 2017 Dec 7.

Institute of Chemistry and Biochemistry, Univ Lyon, Université Lyon 1, CNRS, 43 Bd du 11 novembre 1918, F-69622 Villeurbanne, France.

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December 2017

A Metal-Free Route to Heterocyclic Trifluoromethyl- and Fluoroalkylselenolated Molecules.

Org Lett 2018 01 13;20(1):56-59. Epub 2017 Dec 13.

Institute of Chemistry and Biochemistry (ICBMS UMR CNRS 5246), Univ Lyon, Université Lyon 1 , CNRS, 43 Bd du 11 novembre 1918, 69622 Villeurbanne, France.

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January 2018

Fluorous l-Carbidopa Precursors: Highly Enantioselective Synthesis and Computational Prediction of Bioactivity.

J Org Chem 2018 01 21;83(1):303-313. Epub 2017 Dec 21.

Department of Chemistry, Centro de Innovación en Química Avanzada (ORFEO-CINQA), Universitat Autònoma de Barcelona , Cerdanyola del Vallès, Barcelona 08193, Spain.

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January 2018

Exploring the Reactivity of Trifluoromethyl Tolueneselenosulfonate with Alkynes under Copper Catalysis.

Chemistry 2018 Jan 6;24(1):97-100. Epub 2017 Dec 6.

Institute of Chemistry and Biochemistry, ICBMS-UMR CNRS 5246, Univ Lyon, Université Lyon 1, CNRS, 43 Bd du 11 Novembre 1918, 69622, Villeurbanne, France.

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January 2018

Synthetic Approaches to Trifluoromethylselenolated Compounds.

Chemistry 2018 Mar 12;24(15):3659-3670. Epub 2017 Dec 12.

Institute of Chemistry and Biochemistry (ICBMS-UMR CNRS 5246), Univ Lyon, Université Lyon 1, CNRS, 43 Bd du 11 Novembre 1918, 69622, Villeurbanne, France.

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March 2018