Publications by authors named "Stefania Gagliardi"

20Publications

Chiral resolution and pharmacological characterization of the enantiomers of the Hsp90 inhibitor 2-amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one oxime.

ChemMedChem 2014 Jul 17;9(7):1574-85. Epub 2014 Apr 17.

Genextra Group, Congenia s.r.l., Via Adamello 16, 20139 Milan (Italy); Current address: Drug Discovery Program, Department of Experimental Oncology, IEO-European Institute of Oncology, Via Adamello 16, 20139 Milan (Italy).

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July 2014

Synthesis of (+)-dumetorine and congeners by using flow chemistry technologies.

Chemistry 2011 May 19;17(22):6221-6. Epub 2011 Apr 19.

Dipartimento di Chimica Organica e Industriale, Università degli Studi di Milano, Via Venezian 21, 20133 Milano, Italy.

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May 2011

Inhibition of Plasmodium falciparum pH regulation by small molecule indole derivatives results in rapid parasite death.

Biochem Pharmacol 2010 May 11;79(9):1291-9. Epub 2010 Jan 11.

Research School of Biology, The Australian National University, Canberra, ACT 0200, Australia.

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May 2010

Efficient continuous flow synthesis of hydroxamic acids and suberoylanilide hydroxamic acid preparation.

J Org Chem 2009 May;74(9):3540-3

Dipartimento di Chimica Organica e Industriale, Università degli Studi di Milano, Via Venezian 21, 20133 Milan, Italy.

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May 2009

Identification of small molecule agonists of the motilin receptor.

Bioorg Med Chem Lett 2008 Dec 19;18(24):6423-8. Epub 2008 Oct 19.

Neurology & GI Centre of Excellence for Drug Discovery, GlaxoSmithKline, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, UK.

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December 2008

Antagonists at the neurokinin receptors--recent patent literature.

IDrugs 2003 Aug;6(8):758-72

NiKem Research Srl, Via Zambeletti 25, 20021-Baranzate di Bollate, Milan, Italy.

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August 2003

Morphinan derivatives--A review of the recent patent literature.

IDrugs 2003 Feb;6(2):129-37

NiKem Research Srl, Via Zambeletti 25, 20021 - Baranzate di Bollate, Milan, Italy.

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February 2003

Synthesis of photoactivable inhibitors of osteoclast vacuolar ATPase.

Bioorg Med Chem 2003 May;11(10):2247-54

Dipartimento di Scienze Molecolari Agroalimentari, Università di Milano, Via Celoria 2, 20133 Milan, Italy.

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May 2003

Selective Oxidation of Hydroxy Groups of Bafilomycin A(1).

J Org Chem 1996 Oct;61(20):7185-7188

SmithKline Beecham SpA, via Zambeletti, 20021 Baranzate di Bollate (Milano), Italy.

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October 1996