Sameer P Kawatkar

Sameer P Kawatkar

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Sameer P Kawatkar

Sameer P Kawatkar

Publications by authors named "Sameer P Kawatkar"

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8Publications

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Rapid Identification of Novel Allosteric PRC2 Inhibitors.

ACS Chem Biol 2019 Oct 23;14(10):2134-2140. Epub 2019 Sep 23.

Mechanistic Biology and Profiling, Discovery Sciences , R&D, AstraZeneca , Cambridge , CB4 0WG U.K.

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http://dx.doi.org/10.1021/acschembio.9b00468DOI Listing
October 2019

Antibacterial inhibitors of Gram-positive thymidylate kinase: structure-activity relationships and chiral preference of a new hydrophobic binding region.

J Med Chem 2014 Jun 3;57(11):4584-97. Epub 2014 Jun 3.

Infection Innovative Medicines and ‡Discovery Sciences, AstraZeneca , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.

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http://dx.doi.org/10.1021/jm500463cDOI Listing
June 2014

Sulfonylpiperidines as novel, antibacterial inhibitors of Gram-positive thymidylate kinase (TMK).

Bioorg Med Chem Lett 2013 Jan 5;23(1):169-73. Epub 2012 Nov 5.

AstraZeneca Infection Innovative Medicines, 35 Gatehouse Drive, Waltham, MA 02451, USA.

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http://dx.doi.org/10.1016/j.bmcl.2012.10.128DOI Listing
January 2013

Structural basis of the inhibition of Golgi alpha-mannosidase II by mannostatin A and the role of the thiomethyl moiety in ligand-protein interactions.

J Am Chem Soc 2006 Jun;128(25):8310-9

Complex Carbohydrate Research Center, University of Georgia, 315 Riverbend Road, Athens, Georgia 30602, USA.

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http://dx.doi.org/10.1021/ja061216pDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2553320PMC
June 2006

Cycloaromatization of 1,4-pentadiynes: a viable possibility?

Org Lett 2002 Oct;4(21):3643-6

Department of Chemistry, University of Georgia, Athens, Georgia 30605-2556, USA.

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http://dx.doi.org/10.1021/ol0266424DOI Listing
October 2002