Paolo Grieco

Paolo Grieco

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Paolo Grieco

Publications by authors named "Paolo Grieco"

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Natural and synthetic peptides in the cardiovascular diseases: An update on diagnostic and therapeutic potentials.

Arch Biochem Biophys 2019 Feb 24;662:15-32. Epub 2018 Nov 24.

Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131, Naples, Italy. Electronic address:

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http://dx.doi.org/10.1016/j.abb.2018.11.021DOI Listing
February 2019

Short PlGF-derived peptides bind VEGFR-1 and VEGFR-2 in vitro and on the surface of endothelial cells.

J Pept Sci 2019 Jan 16:e3146. Epub 2019 Jan 16.

Istituto di Biostrutture e Bioimmagini-CNR and CIRPEB, Naples, Italy.

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http://dx.doi.org/10.1002/psc.3146DOI Listing
January 2019

Rationally Designed α-Conotoxin Analogues Maintained Analgesia Activity and Weakened Side Effects.

Molecules 2019 Jan 18;24(2). Epub 2019 Jan 18.

State Key Laboratory of Natural Medicines, Ministry of Education, The Engineering Research Center of Synthetic Polypeptide Drug Discovery and Evaluation of Jiangsu Province, Department of Marine Pharmacy, China Pharmaceutical University, Nanjing 211198, China.

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http://dx.doi.org/10.3390/molecules24020337DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6358911PMC
January 2019

Investigation on side-product formation during the synthesis of a lactoferrin-derived lactam-bridged cyclic peptide.

Amino Acids 2018 Oct 4;50(10):1367-1375. Epub 2018 Jul 4.

Dipartimento di Farmacia, Università degli Studi di Salerno, 84084, Fisciano, SA, Italy.

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http://dx.doi.org/10.1007/s00726-018-2612-9DOI Listing
October 2018

Urokinase receptor derived peptides as potent inhibitors of the formyl peptide receptor type 1-triggered cell migration.

Eur J Med Chem 2018 Jan 1;143:348-360. Epub 2017 Dec 1.

Department of Pharmacy, University of Naples 'Federico II', Naples 80131, Italy; Centro Interuniversitario di Ricerca sui Peptidi Bioattivi (CIRPEB) University of Naples "Federico II" and DFM-Scarl, Institute of Biostructures and Bioimaging - CNR Via Mezzocannone 16, 80134 Naples, Italy.

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http://dx.doi.org/10.1016/j.ejmech.2017.11.030DOI Listing
January 2018

Urotensin-II Receptor: A Double Identity Receptor Involved in Vasoconstriction and in the Development of Digestive Tract Cancers and other Tumors.

Curr Cancer Drug Targets 2017 ;17(2):109-121

Department of Clinical and Experimental Medicine, Second University of Naples, Via Pansini 5 80131 Naples, Italy. Select country.

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http://dx.doi.org/10.2174/1568009616666160621101248DOI Listing
October 2017

Multiple beneficial effects of melanocortin MC receptor agonists in experimental neurodegenerative disorders: Therapeutic perspectives.

Prog Neurobiol 2017 Jan 1;148:40-56. Epub 2016 Dec 1.

Department of Biomedical, Metabolic and Neural Sciences, Section of Pharmacology and Molecular Medicine, University of Modena and Reggio Emilia, Modena, Italy. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S03010082153001
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http://dx.doi.org/10.1016/j.pneurobio.2016.11.004DOI Listing
January 2017

Nanocarriers Conjugated with Cell Penetrating Peptides: New Trojan Horses by Modern Ulysses.

Curr Pharm Biotechnol 2016;17(8):700-22

Department of Biochemistry, Biophysics and General Pathology, Second University of Naples, Italy. Via L. De Crecchio, 7. 80138, Naples, Italy.

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December 2016

Targeting "Undruggable" Proteins: Design of Synthetic Cyclopeptides.

Curr Med Chem 2016 ;23(8):748-62

Department of Pharmacy, University "Federico II", Via Mezzocannone, 16, 80134, Naples, Italy.

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November 2016

Treatment with a Urokinase Receptor-derived Cyclized Peptide Improves Experimental Colitis by Preventing Monocyte Recruitment and Macrophage Polarization.

Inflamm Bowel Dis 2016 10;22(10):2390-401

*IBD Center, Humanitas Research Institute, Rozzano, Italy; †Department of Translational Medicine, Università degli Studi di Milano, Milan, Italy; ‡Neoplastic Progression Unit, Department of Experimental Oncology, IRCCS Istituto Nazionale Tumori "Fondazione G. Pascale," Naples, Italy; §SUN, Second University of Naples, Naples, Italy; ‖Department of Pharmacy, University Federico II, Naples, Italy; and ¶Hunimed-Humanitas University, Milan, Italy.

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http://dx.doi.org/10.1097/MIB.0000000000000896DOI Listing
October 2016

Antimicrobial peptides as an opportunity against bacterial diseases.

Curr Med Chem 2015 ;22(14):1665-77

Dipartimento di Farmacia and DFM and Cirpeb- Universita di Napoli "Federico II", Via Mezzocannone 16, 80134, Naples, Italy.

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June 2016

Urotensin II((4-11)) Azasulfuryl Peptides: Synthesis and Biological Activity.

J Med Chem 2016 05 17;59(10):4740-52. Epub 2016 May 17.

Département de Chimie, Université de Montréal , C.P. 6128, Station Centre-ville, Montréal, Québec H3C 3J7, Canada.

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http://dx.doi.org/10.1021/acs.jmedchem.6b00108DOI Listing
May 2016

Chemical modifications in the seed region of miRNAs 221/222 increase the silencing performances in gastrointestinal stromal tumor cells.

Eur J Med Chem 2016 Mar 27;111:15-25. Epub 2016 Jan 27.

Institute of Genetic and Biophysics "Adriano Buzzati Traverso", CNR, Via Pietro Castellino 111, 80131 Naples, Italy. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2016.01.047DOI Listing
March 2016

Discovery of Novel Potent and Selective Agonists at the Melanocortin-3 Receptor.

J Med Chem 2015 Dec 16;58(24):9773-8. Epub 2015 Dec 16.

Dipartimento di Farmacia, Università di Napoli Federico II , Via D. Montesano, 49, 80131, Naples, Italy.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5070805PMC
http://dx.doi.org/10.1021/acs.jmedchem.5b01285DOI Listing
December 2015

The renaissance era of peptides in drug discovery at the 14th Naples workshop on bioactive peptides.

J Pept Sci 2015 May 10;21(5):321-2. Epub 2015 Apr 10.

CIRPeB - Research Centre on Bioactive Peptides, University of Naples "Federico II" Napoli, Naples, Italy.

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http://dx.doi.org/10.1002/psc.2783DOI Listing
May 2015

Melanocortin peptides protect chondrocytes from mechanically induced cartilage injury.

Biochem Pharmacol 2014 Nov 28;92(2):336-47. Epub 2014 Aug 28.

Faculty of Science and Technology, University of Westminster, 115 New Cavendish Street, London W1W 6UW, United Kingdom.

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http://dx.doi.org/10.1016/j.bcp.2014.08.019DOI Listing
November 2014

Urotensin-II receptor is over-expressed in colon cancer cell lines and in colon carcinoma in humans.

Eur J Clin Invest 2014 22;44(3):285-94. Epub 2014 Jan 22.

Gastroenterology Unit, Department of Clinical and Experimental Medicine and Surgery, Second University of Naples, Naples, Italy.

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http://dx.doi.org/10.1111/eci.12231DOI Listing
October 2014

Development of a liposome-based formulation for vitamin K1 nebulization on the skin.

Int J Nanomedicine 2014 10;9:1823-32. Epub 2014 Apr 10.

Department of Pharmacy, Università degli Studi di Napoli Federico II, Naples, Italy.

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http://dx.doi.org/10.2147/IJN.S58365DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3986299PMC
August 2014

Exploitation of viral properties for intracellular delivery.

J Pept Sci 2014 Jul 30;20(7):468-78. Epub 2014 May 30.

Department of Pharmacy, University of Naples "Federico II", Via Mezzocannone 16, and Via Domenico Montesano 49, 80100, Napoli, Italy; Centro Interuniversitario di Ricerca sui Peptidi Bioattivi, University of Naples "Federico II", Via Mezzocannone 16, 80134, Napoli, Italy; Istituto di Biostrutture e Bioimmagini - CNR, Via Mezzocannone 16, 80134, Napoli, Italy; DFM Scarl, Via Mezzocannone 16, 80134, Napoli, Italy.

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http://dx.doi.org/10.1002/psc.2649DOI Listing
July 2014

Urantide conformation and interaction with the urotensin-II receptor.

Arch Pharm (Weinheim) 2014 Mar 4;347(3):185-92. Epub 2013 Dec 4.

Department of Pharmacy, University of Naples "Federico II", Naples, Italy.

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http://dx.doi.org/10.1002/ardp.201300269DOI Listing
March 2014

Modulation of the JAK/ERK/STAT signaling in melanocortin-induced inhibition of local and systemic responses to myocardial ischemia/reperfusion.

Pharmacol Res 2013 Jun 25;72:1-8. Epub 2013 Mar 25.

Department of Biomedical, Metabolic and Neural Sciences, Section of Pharmacology and Molecular Medicine, University of Modena and Reggio Emilia, Modena, Italy.

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http://dx.doi.org/10.1016/j.phrs.2013.03.005DOI Listing
June 2013

Opposite modulation of cell migration by distinct subregions of urokinase connecting peptide.

Chembiochem 2013 May 20;14(7):882-9. Epub 2013 Mar 20.

Institute of Genetics and Biophysics Adriano Buzzati-Traverso, National Research Council, Via Castellino 111, Naples, Italy.

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http://dx.doi.org/10.1002/cbic.201200774DOI Listing
May 2013

NDP-MSH inhibits neutrophil migration through nicotinic and adrenergic receptors in experimental peritonitis.

Naunyn Schmiedebergs Arch Pharmacol 2013 Apr 22;386(4):311-8. Epub 2013 Jan 22.

Department of Pharmacology, Faculty of Medicine of Ribeirão Preto, University of São Paulo, Av. Bandeirantes 3900, Ribeirão Preto, São Paulo, Brazil.

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http://link.springer.com/10.1007/s00210-013-0834-7
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http://dx.doi.org/10.1007/s00210-013-0834-7DOI Listing
April 2013

Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors.

J Amino Acids 2013 26;2013:606282. Epub 2013 Feb 26.

Dipartimento di Scienze Farmaceutiche e Biomediche, Università degli Studi di Salerno, Via Ponte don Melillo, 84084 Fisciano, Italy.

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http://dx.doi.org/10.1155/2013/606282DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3600326PMC
March 2013

Urotensin-II Ligands: An Overview from Peptide to Nonpeptide Structures.

J Amino Acids 2013 25;2013:979016. Epub 2013 Feb 25.

Department of Pharmacy, University of Naples Federico II, 80131 Naples, Italy.

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http://dx.doi.org/10.1155/2013/979016DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3596952PMC
March 2013

The effect of d-amino acid substitution on the selectivity of temporin L towards target cells: identification of a potent anti-Candida peptide.

Biochim Biophys Acta 2013 Feb 10;1828(2):652-60. Epub 2012 Sep 10.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples 'Federico II', I-80131 Naples, Italy.

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http://dx.doi.org/10.1016/j.bbamem.2012.08.027DOI Listing
February 2013

Molecular changes induced in rat liver by hemorrhage and effects of melanocortin treatment.

Anesthesiology 2012 Mar;116(3):692-700

Center for Surgical Research, Fondazione IRCCS Ca' Granda - Ospedale Maggiore Policlinico, Milano, Italy.

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http://dx.doi.org/10.1097/ALN.0b013e318246ea68DOI Listing
March 2012

Conformational study on cyclic melanocortin ligands and new insight into their binding mode at the MC4 receptor.

Eur J Med Chem 2011 Sep 23;46(9):3721-33. Epub 2011 May 23.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, I-80131 Naples, Italy.

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https://linkinghub.elsevier.com/retrieve/pii/S02235234110041
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http://dx.doi.org/10.1016/j.ejmech.2011.05.038DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5102844PMC
September 2011

Discovery of small peptide antagonists of PED/PEA15-D4α interaction from simplified combinatorial libraries.

Chem Biol Drug Des 2011 May 1;77(5):319-27. Epub 2011 Mar 1.

Department of Biological Sciences, School of Biotechnological Sciences, University of Naples Federico II, Via Mezzocannone, 16, 80134, Naples, Italy.

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http://dx.doi.org/10.1111/j.1747-0285.2011.01094.xDOI Listing
May 2011

Alanine scanning analysis and structure-function relationships of the frog-skin antimicrobial peptide temporin-1Ta.

J Pept Sci 2011 May 18;17(5):358-65. Epub 2011 Feb 18.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, I-80131 Naples, Italy.

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http://dx.doi.org/10.1002/psc.1350DOI Listing
May 2011

Structure-activity relationship, conformational and biological studies of temporin L analogues.

J Med Chem 2011 Mar 14;54(5):1298-307. Epub 2011 Feb 14.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, Via D Montesano 49, I-80131 Naples, Italy.

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http://dx.doi.org/10.1021/jm1012853DOI Listing
March 2011

Anti-inflammatory and antiosteoclastogenesis properties of endogenous melanocortin receptor type 3 in experimental arthritis.

FASEB J 2010 Dec 11;24(12):4835-43. Epub 2010 Aug 11.

William Harvey Research Institute, Barts and London School of Medicine, Queen Mary University of London, London, UK.

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http://dx.doi.org/10.1096/fj.10-167759DOI Listing
December 2010

Synthesis and pharmacological evaluation of some 4-oxo-quinoline-2-carboxylic acid derivatives as anti-inflammatory and analgesic agents.

Arch Pharm (Weinheim) 2010 Oct;343(10):561-9

Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Napoli, Italia.

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http://dx.doi.org/10.1002/ardp.201000016DOI Listing
October 2010

Melanocortins counteract inflammatory and apoptotic responses to prolonged myocardial ischemia/reperfusion through a vagus nerve-mediated mechanism.

Eur J Pharmacol 2010 Jul 10;637(1-3):124-30. Epub 2010 Apr 10.

Department of Biomedical Sciences, University of Modena and Reggio Emilia, Modena, Italy.

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http://dx.doi.org/10.1016/j.ejphar.2010.03.052DOI Listing
July 2010

Design and synthesis of spirotryprostatin-inspired diketopiperazine systems from prolyl spirooxoindolethiazolidine derivatives.

Bioorg Med Chem 2010 Jun 29;18(12):4328-37. Epub 2010 Apr 29.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, Via D. Montesano 49, I-80131 Naples, Italy.

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http://dx.doi.org/10.1016/j.bmc.2010.04.079DOI Listing
June 2010

Urotensin II: a novel target in human corpus cavernosum.

J Sex Med 2010 May 25;7(5):1778-86. Epub 2009 Sep 25.

University of Naples, Federico II-Interdepartmental Research Centre for Sexual Medicine (CIRMS), Naples, Italy.

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http://dx.doi.org/10.1111/j.1743-6109.2009.01450.xDOI Listing
May 2010

New insight into the mechanism of action of the temporin antimicrobial peptides.

Biochemistry 2010 Feb;49(7):1477-85

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, I-80131 Naples, Italy.

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http://dx.doi.org/10.1021/bi902166dDOI Listing
February 2010

Synthesis and pharmacological evaluation of analogs of indole-based cannabimimetic agents.

Chem Biol Drug Des 2010 Jan 4;75(1):106-14. Epub 2009 Nov 4.

Dipartimento di Chimica Farmaceutica e Tossicologica, Via D. Montesano 49 Università di Napoli Federico II, Naples, Italy.

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http://dx.doi.org/10.1111/j.1747-0285.2009.00910.xDOI Listing
January 2010

Inflamed phenotype of the mesenteric microcirculation of melanocortin type 3 receptor-null mice after ischemia-reperfusion.

FASEB J 2008 Dec 29;22(12):4228-38. Epub 2008 Aug 29.

William Harvey Research Institute, Barts and The London School of Medicine, Charterhouse Square, London, EC1M 6BQ, UK.

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http://dx.doi.org/10.1096/fj.08-113886DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2700033PMC
December 2008

A role for MC3R in modulating lung inflammation.

Pulm Pharmacol Ther 2008 Dec 17;21(6):866-73. Epub 2008 Oct 17.

Department of Human and Health Sciences, School of Biosciences, University of Westminster, 115 New Cavendish Street, London W1W 6UW, UK.

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http://dx.doi.org/10.1016/j.pupt.2008.09.004DOI Listing
December 2008

Binding site of loperamide: automated docking of loperamide in human mu- and delta-opioid receptors.

Chem Biol Drug Des 2008 Apr 12;71(4):328-35. Epub 2008 Feb 12.

Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, Via D. Montesano, 49-80131 Napoli, Italy.

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http://dx.doi.org/10.1111/j.1747-0285.2008.00637.xDOI Listing
April 2008

A different molecular mechanism underlying antimicrobial and hemolytic actions of temporins A and L.

J Med Chem 2008 Apr 28;51(8):2354-62. Epub 2008 Mar 28.

Department of Pharmaceutical and Toxicological Chemistry, University of Naples "Federico II", I-80131 Naples, Italy.

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http://dx.doi.org/10.1021/jm701604tDOI Listing
April 2008

Conformational stability of Abeta-(25-35) in the presence of thiazolidine derivatives.

Chem Biol Drug Des 2007 Feb;69(2):111-8

Dipartimento di Scienze Farmaceutiche, University of Salerno, 84084 Fisciano, Italy.

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http://dx.doi.org/10.1111/j.1747-0285.2007.00482.xDOI Listing
February 2007

Structure-function relationships and conformational properties of alpha-MSH(6-13) analogues with candidacidal activity.

Chem Biol Drug Des 2007 Jan;69(1):68-74

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, Via D. Montesano 49, I-80131 Naples, Italy.

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http://dx.doi.org/10.1111/j.1747-0285.2007.00473.xDOI Listing
January 2007

[D-Trp8]-gamma-melanocyte-stimulating hormone exhibits anti-inflammatory efficacy in mice bearing a nonfunctional MC1R (recessive yellow e/e mouse).

Mol Pharmacol 2006 Dec 7;70(6):1850-5. Epub 2006 Sep 7.

The William Harvey Research Institute, Charterhouse Square, London, United Kingdom.

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http://dx.doi.org/10.1124/mol.106.028878DOI Listing
December 2006

Melanocortin 3 receptors control crystal-induced inflammation.

FASEB J 2006 Nov;20(13):2234-41

The William Harvey Research Institute, Queen Mary School of Medicine and Dentistry, Charterhouse Sq., London EC1M 6BQ, UK.

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http://dx.doi.org/10.1096/fj.06-6339comDOI Listing
November 2006

Activation of urokinase receptor by a novel interaction between the connecting peptide region of urokinase and alpha v beta 5 integrin.

J Cell Sci 2006 Aug 1;119(Pt 16):3424-34. Epub 2006 Aug 1.

Institute of Genetics and Biophysics Adriano Buzzati-Traverso, National Research Council, Via P. Castellino 111, 80131 Naples, Italy.

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http://dx.doi.org/10.1242/jcs.03067DOI Listing
August 2006

Novel and selective alpha(v)beta3 receptor peptide antagonist: design, synthesis, and biological behavior.

J Med Chem 2006 Jun;49(11):3416-20

Institute of Biostructures and Bioimaging, CNR, Department of Biological Sciences, University of Naples Federico II, and C. I. R. Pe. B., via Mezzocannone 16, 80134 Naples, Italy.

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http://dx.doi.org/10.1021/jm060233mDOI Listing
June 2006

Synthesis and pharmacological activity of 2-(substituted)-3-{2-[(4-phenyl-4-cyano)piperidino]ethyl}-1,3-thiazolidin-4-ones.

Chem Biol Drug Des 2006 Jun;67(6):432-6

Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli Federico II, via D. Montesano 49, 80131 Napoli, Italia.

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http://dx.doi.org/10.1111/j.1747-0285.2006.00399.xDOI Listing
June 2006

Structure-activity studies of new melanocortin peptides containing an aromatic amino acid at the N-terminal position.

Peptides 2006 Feb 21;27(2):472-81. Epub 2005 Nov 21.

Department of Chemistry and Toxicology, University of Arizona, Tuscon, AZ 85721, USA.

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http://dx.doi.org/10.1016/j.peptides.2005.01.032DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1483901PMC
February 2006

Urotensin-II receptor ligands. From agonist to antagonist activity.

J Med Chem 2005 Nov;48(23):7290-7

Department of Pharmaceutical and Toxicological Chemistry, University of Naples Federico II, I-80131 Naples, Italy.

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http://dx.doi.org/10.1021/jm058043jDOI Listing
November 2005

Cross-talk between fMLP and vitronectin receptors triggered by urokinase receptor-derived SRSRY peptide.

J Biol Chem 2005 Jul 2;280(26):25225-32. Epub 2005 May 2.

Department of Experimental Oncology, National Cancer Institute, 80131 Naples, Italy.

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http://dx.doi.org/10.1074/jbc.M412605200DOI Listing
July 2005

A new efficient synthetic methodology for tetrahydroisoquinoline and tetrahydro-beta-carboline derivatives using the Pictet-Spengler reaction.

Mol Divers 2004 ;8(4):427-30

Dipartimento di Chimica Farmaceutica e Tossicologica, University of Naples "Federico II", Naples, Italy.

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May 2005

Morphiceptin analogues containing a dipeptide mimetic structure: an investigation on the bioactive topology at the mu-receptor.

J Med Chem 2005 May;48(9):3153-63

Dipartimento di Chimica Farmaceutica e Tossicologica, Università degli Studi di Napoli "Federico II", I-80131 Napoli, Italy.

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http://dx.doi.org/10.1021/jm040867yDOI Listing
May 2005

Design and synthesis of melanocortin peptides with candidacidal and anti-TNF-alpha properties.

J Med Chem 2005 Mar;48(5):1384-8

Department of Pharmaceutical Chemistry and Toxicology, Università di Napoli, 80131 Naples, Italy.

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http://dx.doi.org/10.1021/jm040890jDOI Listing
March 2005

Urotensin-II receptor peptide agonists.

Med Res Rev 2004 Sep;24(5):577-88

Department of Pharmaceutical Sciences, University of Salerno, I-84084 Fisciano, Italy.

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http://dx.doi.org/10.1002/med.20001DOI Listing
September 2004

Unraveling the active conformation of urotensin II.

J Med Chem 2004 Mar;47(7):1652-61

Department of Pharmaceutical Sciences, University of Salerno, Via Ponte Don Melillo 11C, I-84084 Fisciano, Italy.

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http://dx.doi.org/10.1021/jm0309912DOI Listing
March 2004

Urantide: an ultrapotent urotensin II antagonist peptide in the rat aorta.

Br J Pharmacol 2003 Dec;140(7):1155-8

Department of Pharmacology, Menarini Ricerche SpA, Via Rismondo 12/A, Florence 50131, Italy.

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http://dx.doi.org/10.1038/sj.bjp.0705555DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1574141PMC
December 2003