Publications by authors named "Paola Gallinari"

26Publications

Octreotide Conjugates for Tumor Targeting and Imaging.

Pharmaceutics 2019 May 7;11(5). Epub 2019 May 7.

Department of Chemistry, Organic and Bioorganic Chemistry, Bielefeld University, Universitätsstraße 25, DE-33615 Bielefeld, Germany.

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http://dx.doi.org/10.3390/pharmaceutics11050220DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6571972PMC
May 2019

Blocking the association of HDAC4 with MAP1S accelerates autophagy clearance of mutant Huntingtin.

Aging (Albany NY) 2015 Oct;7(10):839-53

Institute of Biosciences and Technology, Texas A&M Health Science Center, Houston, TX 77030, USA.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4637209PMC
http://dx.doi.org/10.18632/aging.100818DOI Listing
October 2015

Benzodeazaoxaflavins as sirtuin inhibitors with antiproliferative properties in cancer stem cells.

J Med Chem 2012 Sep 7;55(18):8193-7. Epub 2012 Sep 7.

Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, Piazzale Aldo Moro 5, 00185 Roma, Italy.

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http://dx.doi.org/10.1021/jm301115rDOI Listing
September 2012

Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222.

Bioorg Med Chem 2010 May 15;18(9):3252-60. Epub 2010 Mar 15.

Dipartimento di Scienze Farmaceutiche, Università degli Studi di Salerno, Via Ponte Don Melillo, 84084 Fisciano (SA), Italy.

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http://linkinghub.elsevier.com/retrieve/pii/S096808961000226
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http://dx.doi.org/10.1016/j.bmc.2010.03.022DOI Listing
May 2010

Smoothened antagonists: a promising new class of antitumor agents.

Expert Opin Drug Discov 2009 May;4(5):525-44

Istituto di Ricerche di Biologia Molecolare P. Angeletti, Department of Oncology, IRBM- Merck Research Laboratories Rome, Via Pontina Km 30,600, 00040 Pomezia, Italy +39 06 91093232 ; +39 06 91093549 ;

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http://dx.doi.org/10.1517/17460440902852686DOI Listing
May 2009

Probing the elusive catalytic activity of vertebrate class IIa histone deacetylases.

Bioorg Med Chem Lett 2008 Mar 14;18(6):1814-9. Epub 2008 Feb 14.

IRBM/Merck Research Laboratories, Via Pontina km 30,600, 00040 Pomezia, Italy.

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X080020
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http://dx.doi.org/10.1016/j.bmcl.2008.02.025DOI Listing
March 2008

PP2A regulates HDAC4 nuclear import.

Mol Biol Cell 2008 Feb 28;19(2):655-67. Epub 2007 Nov 28.

Dipartimento di Scienze e Tecnologie Biomediche, Sezione di Biologia and MATI Center of Excellence, Universita' di Udine, 33100 Udine, Italy.

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http://www.molbiolcell.org/doi/10.1091/mbc.e07-06-0623
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http://dx.doi.org/10.1091/mbc.e07-06-0623DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2230598PMC
February 2008

Substrate binding to histone deacetylases as shown by the crystal structure of the HDAC8-substrate complex.

EMBO Rep 2007 Sep 10;8(9):879-84. Epub 2007 Aug 10.

Istituto di Ricerche di Biologia Molecolare P. Angeletti, Via Pontina Km 30.600, 00040 Pomezia, Rome, Italy.

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http://dx.doi.org/10.1038/sj.embor.7401047DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1973954PMC
September 2007

HDACs, histone deacetylation and gene transcription: from molecular biology to cancer therapeutics.

Cell Res 2007 Mar;17(3):195-211

Istituto di Ricerche di Biologia Molecolare P. Angeletti-IRBM-Merck Research Laboratories Rome, Pomezia, Italy.

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http://dx.doi.org/10.1038/sj.cr.7310149DOI Listing
March 2007

Molecular insights into azumamide e histone deacetylases inhibitory activity.

J Am Chem Soc 2007 Mar 21;129(10):3007-12. Epub 2007 Feb 21.

Department of Chemistry, University of Salerno, Via Ponte Don Melillo, 84084 Fisciano, Salerno, Italy.

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http://dx.doi.org/10.1021/ja0686256DOI Listing
March 2007

Characterization of prejunctional serotonin receptors modulating [3H]acetylcholine release in the human detrusor.

J Pharmacol Exp Ther 2006 Jan 15;316(1):129-35. Epub 2005 Sep 15.

Department of Experimental and Applied Pharmacology, School of Pharmacy, University of Pavia, Viale Taramelli 14, I-27100 Pavia, Italy.

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http://dx.doi.org/10.1124/jpet.105.092551DOI Listing
January 2006