Myles H Akabas

Myles H Akabas

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Myles H Akabas

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MD-PhD graduates remain underrepresented in orthopaedic surgery: National MD-PhD Program Outcome Survey update.

J Orthop Res 2020 Mar 21. Epub 2020 Mar 21.

Department of Orthopaedic Surgery, Stanford Hospital and Clinics, Redwood City, California.

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http://dx.doi.org/10.1002/jor.24669DOI Listing
March 2020

Identification via a Parallel Hit Progression Strategy of Improved Small Molecule Inhibitors of the Malaria Purine Uptake Transporter that Inhibit Parasite Proliferation.

ACS Infect Dis 2019 10 14;5(10):1738-1753. Epub 2019 Aug 14.

Platform Technology & Science and Discovery Partners in Academia , GlaxoSmithKline , 1250 South Collegeville Road , Collegeville , Pennsylvania 19426 , United States.

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http://dx.doi.org/10.1021/acsinfecdis.9b00168DOI Listing
October 2019

The national MD-PhD program outcomes study: Outcomes variation by sex, race, and ethnicity.

JCI Insight 2019 Oct 3;4(19). Epub 2019 Oct 3.

Department of Medicine and Pharmacology, University of Pennsylvania Perelman School of Medicine, Philadelphia, Pennsylvania, USA.

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http://dx.doi.org/10.1172/jci.insight.133010DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6795407PMC
October 2019

The national MD-PhD program outcomes study: Relationships between medical specialty, training duration, research effort, and career paths.

JCI Insight 2019 Oct 3;4(19). Epub 2019 Oct 3.

Department of Physiology & Biophysics, Neuroscience, and Medicine, Albert Einstein College of Medicine, Bronx, New York, USA.

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http://dx.doi.org/10.1172/jci.insight.133009DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6795497PMC
October 2019

In Reply to Sun et al.

Acad Med 2018 02;93(2):150-151

Joseph R. Kahn Professor, chair of pathology, and director, Medical Scientist Training Program, Case Western Reserve University and University Hospitals Cleveland Medical Center, Cleveland, Ohio; e-mail: ORCID: http://orcid.org/0000-0002-6333-162X. Professor of physiology and biophysics and director, Medical Scientist Training Program, Albert Einstein College of Medicine, Bronx, New York; ORCID: http://orcid.org/0000-0001-8781-7846. Professor of physiology and biophysics, Weill Cornell Medical College, and director, Weill Cornell/Rockefeller/Sloan Kettering Tri-Institutional MD-PhD Program, New York, New York; ORCID: http://orcid.org/0000-0002-3026-6710.

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http://dx.doi.org/10.1097/ACM.0000000000002036DOI Listing
February 2018

History and Outcomes of 50 Years of Physician-Scientist Training in Medical Scientist Training Programs.

Acad Med 2017 10;92(10):1390-1398

C.V. Harding is Joseph R. Kahn Professor, chair of pathology, and director, Medical Scientist Training Program, Case Western Reserve University and University Hospitals Cleveland Medical Center, Cleveland, Ohio. M.H. Akabas is professor of physiology and biophysics, and director, Medical Scientist Training Program, Albert Einstein College of Medicine, Bronx, New York. O.S. Andersen is professor of physiology and biophysics, Weill Cornell Medical College, and director, Weill Cornell/Rockefeller/Sloan Kettering Tri-institutional MD-PhD Program, New York, New York.

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http://dx.doi.org/10.1097/ACM.0000000000001779DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5617793PMC
October 2017

Implementing competency based admissions at the Albert Einstein College of Medicine.

Med Educ Online 2016 3;21:30000. Epub 2016 Feb 3.

Department of Obstetrics & Gynecology and Women's Health, Montefiore Medical Center, Albert Einstein College of Medicine, Bronx, NY, USA;

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4742465PMC
http://dx.doi.org/10.3402/meo.v21.30000DOI Listing
October 2016

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond.

Authors:
Wesley C Van Voorhis John H Adams Roberto Adelfio Vida Ahyong Myles H Akabas Pietro Alano Aintzane Alday Yesmalie Alemán Resto Aishah Alsibaee Ainhoa Alzualde Katherine T Andrews Simon V Avery Vicky M Avery Lawrence Ayong Mark Baker Stephen Baker Choukri Ben Mamoun Sangeeta Bhatia Quentin Bickle Lotfi Bounaadja Tana Bowling Jürgen Bosch Lauren E Boucher Fabrice F Boyom Jose Brea Marian Brennan Audrey Burton Conor R Caffrey Grazia Camarda Manuela Carrasquilla Dee Carter Maria Belen Cassera Ken Chih-Chien Cheng Worathad Chindaudomsate Anthony Chubb Beatrice L Colon Daisy D Colón-López Yolanda Corbett Gregory J Crowther Noemi Cowan Sarah D'Alessandro Na Le Dang Michael Delves Joseph L DeRisi Alan Y Du Sandra Duffy Shimaa Abd El-Salam El-Sayed Michael T Ferdig José A Fernández Robledo David A Fidock Isabelle Florent Patrick V T Fokou Ani Galstian Francisco Javier Gamo Suzanne Gokool Ben Gold Todd Golub Gregory M Goldgof Rajarshi Guha W Armand Guiguemde Nil Gural R Kiplin Guy Michael A E Hansen Kirsten K Hanson Andrew Hemphill Rob Hooft van Huijsduijnen Takaaki Horii Paul Horrocks Tyler B Hughes Christopher Huston Ikuo Igarashi Katrin Ingram-Sieber Maurice A Itoe Ajit Jadhav Amornrat Naranuntarat Jensen Laran T Jensen Rays H Y Jiang Annette Kaiser Jennifer Keiser Thomas Ketas Sebastien Kicka Sunyoung Kim Kiaran Kirk Vidya P Kumar Dennis E Kyle Maria Jose Lafuente Scott Landfear Nathan Lee Sukjun Lee Adele M Lehane Fengwu Li David Little Liqiong Liu Manuel Llinás Maria I Loza Aristea Lubar Leonardo Lucantoni Isabelle Lucet Louis Maes Dalu Mancama Nuha R Mansour Sandra March Sheena McGowan Iset Medina Vera Stephan Meister Luke Mercer Jordi Mestres Alvine N Mfopa Raj N Misra Seunghyun Moon John P Moore Francielly Morais Rodrigues da Costa Joachim Müller Arantza Muriana Stephen Nakazawa Hewitt Bakela Nare Carl Nathan Nathalie Narraidoo Sujeevi Nawaratna Kayode K Ojo Diana Ortiz Gordana Panic George Papadatos Silvia Parapini Kailash Patra Ngoc Pham Sarah Prats David M Plouffe Sally-Ann Poulsen Anupam Pradhan Celia Quevedo Ronald J Quinn Christopher A Rice Mohamed Abdo Rizk Andrea Ruecker Robert St Onge Rafaela Salgado Ferreira Jasmeet Samra Natalie G Robinett Ulrich Schlecht Marjorie Schmitt Filipe Silva Villela Francesco Silvestrini Robert Sinden Dennis A Smith Thierry Soldati Andreas Spitzmüller Serge Maximilian Stamm David J Sullivan William Sullivan Sundari Suresh Brian M Suzuki Yo Suzuki S Joshua Swamidass Donatella Taramelli Lauve R Y Tchokouaha Anjo Theron David Thomas Kathryn F Tonissen Simon Townson Abhai K Tripathi Valentin Trofimov Kenneth O Udenze Imran Ullah Cindy Vallieres Edgar Vigil Joseph M Vinetz Phat Voong Vinh Hoan Vu Nao-Aki Watanabe Kate Weatherby Pamela M White Andrew F Wilks Elizabeth A Winzeler Edward Wojcik Melanie Wree Wesley Wu Naoaki Yokoyama Paul H A Zollo Nada Abla Benjamin Blasco Jeremy Burrows Benoît Laleu Didier Leroy Thomas Spangenberg Timothy Wells Paul A Willis

PLoS Pathog 2016 07 28;12(7):e1005763. Epub 2016 Jul 28.

Medicines for Malaria Venture, Geneva, Switzerland.

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http://dx.doi.org/10.1371/journal.ppat.1005763DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4965013PMC
July 2016

Substrate and Inhibitor Specificity of the Plasmodium berghei Equilibrative Nucleoside Transporter Type 1.

Mol Pharmacol 2016 06 5;89(6):678-85. Epub 2016 Apr 5.

Departments of Physiology and Biophysics (A.A., R.D., Y.S., S.N.N., M.H.A.) and Neuroscience and Medicine (M.H.A.), Albert Einstein College of Medicine, Bronx, New York; and Departments Microbiology and Immunology (P.P.H., T.R.S.K., D.A.F.) and Medicine (D.A.F.), Columbia University Medical Center, New York, New York

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http://dx.doi.org/10.1124/mol.115.101386DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4885503PMC
June 2016

Targeting the Plasmodium vivax equilibrative nucleoside transporter 1 (PvENT1) for antimalarial drug development.

Int J Parasitol Drugs Drug Resist 2016 Apr 28;6(1):1-11. Epub 2015 Nov 28.

Department of Physiology & Biophysics, Albert Einstein College of Medicine, Bronx, New York, USA; Department of Neuroscience, Albert Einstein College of Medicine, Bronx, New York, USA; Department of Medicine, Albert Einstein College of Medicine, Bronx, New York, USA. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S22113207153002
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http://dx.doi.org/10.1016/j.ijpddr.2015.11.003DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4706624PMC
April 2016

Cysteine Modification: Probing Channel Structure, Function and Conformational Change.

Authors:
Myles H Akabas

Adv Exp Med Biol 2015 ;869:25-54

Departments of Physiology & Biophysics, Neuroscience and Medicine, Albert Einstein College of Medicine, 1300 Morris Park Avenue, 10461, Bronx, NY, USA.

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http://dx.doi.org/10.1007/978-1-4939-2845-3_3DOI Listing
March 2016

Purine import into malaria parasites as a target for antimalarial drug development.

Ann N Y Acad Sci 2015 Apr 25;1342:19-28. Epub 2014 Nov 25.

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Bronx, New York.

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http://dx.doi.org/10.1111/nyas.12568DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4405406PMC
April 2015

A closer look at attrition in MD-PhD programs.

Acad Med 2014 Jul;89(7):958

Professor of physiology and biophysics and director, Medical Scientist Training Program, Albert Einstein College of Medicine, Bronx, New York; Professor of medicine and director, Medical Scientist Training Program, University of Pennsylvania School of Medicine, Philadelphia, Pennsylvania;

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http://dx.doi.org/10.1097/ACM.0000000000000299DOI Listing
July 2014

Using molecular dynamics to elucidate the structural basis for function in pLGICs.

Authors:
Myles H Akabas

Proc Natl Acad Sci U S A 2013 Oct 4;110(42):16700-1. Epub 2013 Oct 4.

Departments of Physiology and Biophysics, Neuroscience, and Medicine, Albert Einstein College of Medicine, Bronx, NY 10461.

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http://dx.doi.org/10.1073/pnas.1316157110DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3801075PMC
October 2013

Channels: Rotamers affect ion conductance.

Authors:
Myles H Akabas

Nat Chem Biol 2012 Dec;8(12):953-4

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http://dx.doi.org/10.1038/nchembio.1115DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4758366PMC
December 2012

Length and amino acid sequence of peptides substituted for the 5-HT3A receptor M3M4 loop may affect channel expression and desensitization.

PLoS One 2012 23;7(4):e35563. Epub 2012 Apr 23.

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York, United States of America.

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http://journals.plos.org/plosone/article?id=10.1371/journal.pone.0035563PLOS
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3335078PMC
September 2012

Malaria parasite type 4 equilibrative nucleoside transporters (ENT4) are purine transporters with distinct substrate specificity.

Biochem J 2012 Sep;446(2):179-90

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, NY 10461, USA.

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http://biochemj.org/lookup/doi/10.1042/BJ20112220
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http://dx.doi.org/10.1042/BJ20112220DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3756485PMC
September 2012

Gating-induced conformational rearrangement of the γ-aminobutyric acid type A receptor β-α subunit interface in the membrane-spanning domain.

J Biol Chem 2012 Aug 22;287(33):27762-70. Epub 2012 Jun 22.

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M112.363341DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3431678PMC
August 2012

5-HT3 receptor ion size selectivity is a property of the transmembrane channel, not the cytoplasmic vestibule portals.

J Gen Physiol 2011 Oct;138(4):453-66

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, NY 10461, USA.

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http://dx.doi.org/10.1085/jgp.201110686DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3182448PMC
October 2011

Ion channels: Manipulating the munchies in mice.

Authors:
Myles H Akabas

Nat Chem Biol 2011 Oct 18;7(11):759-60. Epub 2011 Oct 18.

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http://dx.doi.org/10.1038/nchembio.697DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4646841PMC
October 2011

Taking Charge: Feeding Malaria via Anion Channels.

Cell 2011 May;145(5):645-7

Department of Microbiology & Immunology, Columbia University College of Physicians and Surgeons, New York, NY 10032, USA.

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https://linkinghub.elsevier.com/retrieve/pii/S00928674110053
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http://dx.doi.org/10.1016/j.cell.2011.05.012DOI Listing
May 2011

Structure of the M2 transmembrane segment of GLIC, a prokaryotic Cys loop receptor homologue from Gloeobacter violaceus, probed by substituted cysteine accessibility.

J Biol Chem 2011 Apr 1;286(16):14098-109. Epub 2011 Mar 1.

Department of Physiology & Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M111.221895DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3077611PMC
April 2011

Drosophila pacemaker neurons require g protein signaling and GABAergic inputs to generate twenty-four hour behavioral rhythms.

Neuron 2010 Dec;68(5):964-77

Department of Biology, New York University, 100 Washington Square East, New York, NY 10003, USA.

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http://dx.doi.org/10.1016/j.neuron.2010.11.017DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3030199PMC
December 2010

Transmembrane segment 11 appears to line the purine permeation pathway of the Plasmodium falciparum equilibrative nucleoside transporter 1 (PfENT1).

J Biol Chem 2010 May 24;285(22):17001-10. Epub 2010 Mar 24.

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M110.115758DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2878030PMC
May 2010

Are MD-PhD programs meeting their goals? An analysis of career choices made by graduates of 24 MD-PhD programs.

Acad Med 2010 Apr;85(4):692-701

Department of Medicine, University of Pennsylvania School of Medicine, Philadelphia, Pennsylvania 19104, USA.

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http://dx.doi.org/10.1097/ACM.0b013e3181d3ca17DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4441397PMC
April 2010

Erythrocytic adenosine monophosphate as an alternative purine source in Plasmodium falciparum.

J Biol Chem 2008 Nov 17;283(47):32889-99. Epub 2008 Sep 17.

Department of Biochemistry, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M804497200DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2583302PMC
November 2008

Modular design of Cys-loop ligand-gated ion channels: functional 5-HT3 and GABA rho1 receptors lacking the large cytoplasmic M3M4 loop.

J Gen Physiol 2008 Feb;131(2):137-46

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, NY 10461, USA.

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http://dx.doi.org/10.1085/jgp.200709896DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2213565PMC
February 2008

Rodent intestinal folate transporters (SLC46A1): secondary structure, functional properties, and response to dietary folate restriction.

Am J Physiol Cell Physiol 2007 Nov 26;293(5):C1669-78. Epub 2007 Sep 26.

Department of Medicine, Albert Einstein College of Medicine, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1152/ajpcell.00202.2007DOI Listing
November 2007

Channel opening by anesthetics and GABA induces similar changes in the GABAA receptor M2 segment.

Biophys J 2007 May 9;92(9):3130-9. Epub 2007 Feb 9.

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1529/biophysj.106.094490DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1852347PMC
May 2007

The location of a closed channel gate in the GABAA receptor channel.

J Gen Physiol 2007 Feb 16;129(2):145-59. Epub 2007 Jan 16.

Department of Physiology, Albert Einstein College of Medicine of Yeshiva University, Bronx, NY 10461, USA.

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http://dx.doi.org/10.1085/jgp.200609639DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2154354PMC
February 2007

Chloroquine-resistant isoforms of the Plasmodium falciparum chloroquine resistance transporter acidify lysosomal pH in HEK293 cells more than chloroquine-sensitive isoforms.

Mol Biochem Parasitol 2006 Dec 25;150(2):288-99. Epub 2006 Sep 25.

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, 1300 Morris Park Avenue, Bronx, NY 10461, USA.

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http://dx.doi.org/10.1016/j.molbiopara.2006.09.001DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1687154PMC
December 2006

State-dependent cross-linking of the M2 and M3 segments: functional basis for the alignment of GABAA and acetylcholine receptor M3 segments.

J Neurosci 2006 Apr;26(17):4492-9

Department of Physiology, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1523/JNEUROSCI.0224-06.2006DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6674078PMC
April 2006

Watching single protons bind.

Authors:
Myles H Akabas

Nat Chem Biol 2006 Mar;2(3):128-30

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http://dx.doi.org/10.1038/nchembio0306-128DOI Listing
March 2006

Spontaneous thermal motion of the GABA(A) receptor M2 channel-lining segments.

J Biol Chem 2005 Oct 9;280(42):35506-12. Epub 2005 Aug 9.

Department of Physiology and Biophysics, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York 10461, USA.

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http://www.jbc.org/lookup/doi/10.1074/jbc.M504645200
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http://dx.doi.org/10.1074/jbc.M504645200DOI Listing
October 2005

Emerging molecular mechanisms of general anesthetic action.

Trends Pharmacol Sci 2005 Oct;26(10):503-10

Departments of Anesthesiology and Pharmacology, Weill Cornell Medical College, 1300 York Avenue, Box 50, New York, NY 10021, USA.

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http://linkinghub.elsevier.com/retrieve/pii/S016561470500204
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http://dx.doi.org/10.1016/j.tips.2005.08.006DOI Listing
October 2005

A role for the beta 1-beta 2 loop in the gating of 5-HT3 receptors.

J Neurosci 2005 Oct;25(41):9358-66

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1523/JNEUROSCI.1045-05.2005DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6725699PMC
October 2005

Differential protein mobility of the gamma-aminobutyric acid, type A, receptor alpha and beta subunit channel-lining segments.

J Biol Chem 2005 Jan 2;280(2):1573-81. Epub 2004 Nov 2.

Departments of Physiology and Biophysics and of Neuroscience, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M410881200DOI Listing
January 2005

Functional and structural analysis of the GABAA receptor alpha 1 subunit during channel gating and alcohol modulation.

J Biol Chem 2005 Jan 2;280(1):308-16. Epub 2004 Nov 2.

Cell and Molecular Biology Program and Waggoner Center for Alcohol and Addiction Research, University of Texas at Austin, Austin, Texas 78712, USA.

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http://dx.doi.org/10.1074/jbc.M409871200DOI Listing
January 2005

GABAA receptor structure-function studies: a reexamination in light of new acetylcholine receptor structures.

Authors:
Myles H Akabas

Int Rev Neurobiol 2004 ;62:1-43

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1016/S0074-7742(04)62001-0DOI Listing
December 2004

Na+/Ca2+ exchange inhibitors: potential drugs to mitigate the severity of ischemic injury.

Authors:
Myles H Akabas

Mol Pharmacol 2004 Jul;66(1):8-10

Department of Physiology and Biophysics, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, NY 10461, USA.

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http://dx.doi.org/10.1124/mol.104.000232.DOI Listing
July 2004

Loose protein packing around the extracellular half of the GABA(A) receptor beta1 subunit M2 channel-lining segment.

J Biol Chem 2004 Mar 8;279(12):11198-205. Epub 2004 Jan 8.

Departments of Physiology and Biophysics and of Neuroscience, Albert Einstein College of Medicine of Yeshiva University, Bronx, New York 10461, USA.

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http://dx.doi.org/10.1074/jbc.M314050200DOI Listing
March 2004

Defining the propofol binding site location on the GABAA receptor.

Mol Pharmacol 2004 Jan;65(1):68-76

Department of Physiology, Albert Einstein College of Medicine, Yeshiva University, Bronx, NY 10461, USA.

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http://molpharm.aspetjournals.org/lookup/doi/10.1124/mol.65.
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http://dx.doi.org/10.1124/mol.65.1.68DOI Listing
January 2004

GABA(A) receptor M2-M3 loop secondary structure and changes in accessibility during channel gating.

J Biol Chem 2002 Nov 10;277(45):43002-10. Epub 2002 Sep 10.

Department of Physiology & Biophysics, Albert Einstein College of Medicine, Bronx, New York 10461, USA.

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http://www.jbc.org/lookup/doi/10.1074/jbc.M206321200
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http://dx.doi.org/10.1074/jbc.M206321200DOI Listing
November 2002

Probing CFTR channel structure and function using the substituted-cysteine-accessibility method.

Authors:
Myles H Akabas

Methods Mol Med 2002 ;70:159-74

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Bronx, NY, USA.

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http://dx.doi.org/10.1385/1-59259-187-6:159DOI Listing
September 2002

Structural evidence that propofol stabilizes different GABA(A) receptor states at potentiating and activating concentrations.

J Neurosci 2002 Sep;22(17):7417-24

Department of Physiology and Biophysics, Albert Einstein College of Medicine, Bronx, New York 10461, USA.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6757991PMC
September 2002