Mohamed A Abdelgawad

Mohamed A Abdelgawad

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Mohamed A Abdelgawad

Mohamed A Abdelgawad

Publications by authors named "Mohamed A Abdelgawad"

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Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamidesAQ3 as carbonic anhydrase isoforms I and II inhibitors.

J Enzyme Inhib Med Chem 2019 Dec;34(1):1457-1464

d Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence , Firenze , Italy.

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http://dx.doi.org/10.1080/14756366.2019.1652282DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6713088PMC
December 2019

New pyrimidine-benzoxazole/benzimidazole hybrids: Synthesis, antioxidant, cytotoxic activity, in vitro cyclooxygenase and phospholipase A2-V inhibition.

Bioorg Chem 2019 Nov 26;92:103218. Epub 2019 Aug 26.

Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2019.103218DOI Listing
November 2019

Novel pyrimidine-pyridine hybrids: Synthesis, cyclooxygenase inhibition, anti-inflammatory activity and ulcerogenic liability.

Bioorg Chem 2018 04 31;77:339-348. Epub 2018 Jan 31.

Department of Pharmacology and Toxicology, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2018.01.028DOI Listing
April 2018

Design, synthesis and biological evaluation of some novel benzothiazole/benzoxazole and/or benzimidazole derivatives incorporating a pyrazole scaffold as antiproliferative agents.

Bioorg Chem 2017 10 15;74:82-90. Epub 2017 Jul 15.

Sharjah Institute for Medical Research, College of Medicine, University of Sharjah, Sharjah, United Arab Emirates; Department of Pharmacology, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2017.07.007DOI Listing
October 2017

Pyrazole-hydrazone derivatives as anti-inflammatory agents: Design, synthesis, biological evaluation, COX-1,2/5-LOX inhibition and docking study.

Bioorg Chem 2017 10 30;74:212-220. Epub 2017 Aug 30.

Department of Zoology, Faculty of Science, Beni-Suef University, Beni-Suef 62514, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2017.08.014DOI Listing
October 2017

Discovery of a COX-2 selective inhibitor hit with anti-inflammatory activity and gastric ulcer protective effect.

Future Med Chem 2017 10 27;9(16):1899-1912. Epub 2017 Oct 27.

Department of Pharmaceutical Chemistry, College of Pharmacy, Aljouf University, Sakaka, Aljouf 2014, Kingdom of Saudi Arabia.

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http://dx.doi.org/10.4155/fmc-2017-0115DOI Listing
October 2017

Synthesis and Biological Evaluation of New Diarylpyrazole and Triarylimidazoline Derivatives as Selective COX-2 Inhibitors.

Arch Pharm (Weinheim) 2017 Aug 12;350(8). Epub 2017 Jun 12.

Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt.

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http://dx.doi.org/10.1002/ardp.201600386DOI Listing
August 2017

Design, synthesis and biological screening of some novel celecoxib and etoricoxib analogs with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile.

Bioorg Chem 2017 02 26;70:173-183. Epub 2016 Dec 26.

Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni Suef University, Beni Suef 62514, Egypt; Pharmaceutical Sciences Department, Ibn Sina National College for Medical Studies, Jeddah 21418, Kingdom of Saudi Arabia.

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https://linkinghub.elsevier.com/retrieve/pii/S00452068163023
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http://dx.doi.org/10.1016/j.bioorg.2016.12.008DOI Listing
February 2017

Design, synthesis and antitumor activity of novel pyrazolo[3,4-d]pyrimidine derivatives as EGFR-TK inhibitors.

Bioorg Chem 2016 06 24;66:88-96. Epub 2016 Mar 24.

Department of Pharmacology, Faulty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2016.03.011DOI Listing
June 2016

Design, synthesis and biological screening of new 4-thiazolidinone derivatives with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile.

Bioorg Chem 2016 Feb 6;64:1-12. Epub 2015 Nov 6.

Department of Pharmaceutical Organic Chemistry, Beni Suef University, Beni Suef 62514, Egypt.

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http://dx.doi.org/10.1016/j.bioorg.2015.11.001DOI Listing
February 2016

Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of novel triarylpyrazoline derivatives as selective COX-2 inhibitors.

Bioorg Med Chem Lett 2015 Dec 19;25(24):5787-91. Epub 2015 Oct 19.

Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt.

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http://dx.doi.org/10.1016/j.bmcl.2015.10.047DOI Listing
December 2015

Synthesis and anti-inflammatory evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing an aminosulphonyl pharmacophore.

Arch Pharm Res 2015 Nov 23;38(11):1932-42. Epub 2015 Apr 23.

Department of Pharmacology, Faculty of Veterinary, Cairo University, Cairo, Egypt.

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http://dx.doi.org/10.1007/s12272-015-0606-7DOI Listing
November 2015

Synthesis and anticancer activity of some new pyrazolo[3,4-d]pyrimidin-4-one derivatives.

Molecules 2014 Mar 18;19(3):3297-309. Epub 2014 Mar 18.

Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.

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http://www.mdpi.com/1420-3049/19/3/3297
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http://dx.doi.org/10.3390/molecules19033297DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6270843PMC
March 2014

Synthesis, anti-breast cancer activity, and molecular modeling of some benzothiazole and benzoxazole derivatives.

Arch Pharm (Weinheim) 2013 Jul 5;346(7):534-41. Epub 2013 Jun 5.

Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt.

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http://doi.wiley.com/10.1002/ardp.201300044
Publisher Site
http://dx.doi.org/10.1002/ardp.201300044DOI Listing
July 2013