Publications by authors named "Mindy I Davis"

32Publications

Identification of Novel Plasmodium falciparum Hexokinase Inhibitors with Antiparasitic Activity.

Antimicrob Agents Chemother 2016 10 23;60(10):6023-33. Epub 2016 Sep 23.

Eukaryotic Pathogens Innovation Center, Department of Genetics and Biochemistry, Clemson University, Clemson, South Carolina, USA

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http://dx.doi.org/10.1128/AAC.00914-16DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5038330PMC
October 2016

Breaking Cryo-EM Resolution Barriers to Facilitate Drug Discovery.

Cell 2016 Jun 26;165(7):1698-1707. Epub 2016 May 26.

Laboratory of Cell Biology, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, USA. Electronic address:

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http://dx.doi.org/10.1016/j.cell.2016.05.040DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4931924PMC
June 2016

Diaphorase Coupling Protocols for Red-Shifting Dehydrogenase Assays.

Assay Drug Dev Technol 2016 Apr;14(3):207-12

NCATS Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health , Rockville, Maryland.

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http://dx.doi.org/10.1089/adt.2016.706DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4840998PMC
April 2016

Avoiding Fluorescence Assay Interference-The Case for Diaphorase.

Assay Drug Dev Technol 2016 Apr;14(3):175-9

NCATS Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health , Rockville, Maryland.

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http://dx.doi.org/10.1089/adt.2016.707DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4840916PMC
April 2016

Ubiquitin-Specific Proteases as Druggable Targets.

Drug Target Rev 2015 ;2(3):60-64

Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20850, USA.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4729384PMC
January 2015

Method for Assaying the Lipid Kinase Phosphatidylinositol-5-phosphate 4-kinase α in Quantitative High-Throughput Screening (qHTS) Bioluminescent Format.

Methods Mol Biol 2016 ;1376:1-9

Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, 20850, USA.

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http://dx.doi.org/10.1007/978-1-4939-3170-5_1DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4696767PMC
August 2016

Bioluminescence Methods for Assaying Kinases in Quantitative High-Throughput Screening (qHTS) Format Applied to Yes1 Tyrosine Kinase, Glucokinase, and PI5P4Kα Lipid Kinase.

Methods Mol Biol 2016 ;1360:47-58

Division of Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA.

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http://dx.doi.org/10.1007/978-1-4939-3073-9_4DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4734380PMC
August 2016

Inheritance of rare functional GCKR variants and their contribution to triglyceride levels in families.

Hum Mol Genet 2014 Oct 30;23(20):5570-8. Epub 2014 May 30.

Oxford Centre for Diabetes, Endocrinology & Metabolism, University of Oxford, Oxford OX3 7LE, UK, NIHR Oxford Biomedical Research Centre, ORH Trust, OCDEM, Churchill Hospital, Oxford OX3 7LE, UK

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https://academic.oup.com/hmg/article-lookup/doi/10.1093/hmg/
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http://dx.doi.org/10.1093/hmg/ddu269DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4168830PMC
October 2014

Biochemical, cellular, and biophysical characterization of a potent inhibitor of mutant isocitrate dehydrogenase IDH1.

J Biol Chem 2014 May 25;289(20):13717-25. Epub 2014 Mar 25.

From the NIH Chemical Genomics Center, National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, Maryland 20892,

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http://dx.doi.org/10.1074/jbc.M113.511030DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4022846PMC
May 2014

Identification of potent Yes1 kinase inhibitors using a library screening approach.

Bioorg Med Chem Lett 2013 Aug 29;23(15):4398-403. Epub 2013 May 29.

Basic Science Program, SAIC-Frederick Inc., Frederick National Laboratory for Cancer Research, Frederick, MD 21702, United States.

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http://dx.doi.org/10.1016/j.bmcl.2013.05.072DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3769177PMC
August 2013

[none].

Assay Drug Dev Technol 2013 Apr;11(3):139-51

1 Novartis Institutes for BioMedical Research , Cambridge, Massachusetts.

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http://dx.doi.org/10.1089/adt.2013.1103.lrDOI Listing
April 2013

Comprehensive analysis of kinase inhibitor selectivity.

Nat Biotechnol 2011 Oct 30;29(11):1046-51. Epub 2011 Oct 30.

Ambit Biosciences, San Diego, California, USA.

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http://dx.doi.org/10.1038/nbt.1990DOI Listing
October 2011

Literature search and review.

Assay Drug Dev Technol 2011 Jun;9(3):198-212

Novartis Institutes for BioMedical Research , Cambridge, Massachusetts.

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http://dx.doi.org/10.1089/adt.2011.0903.lrDOI Listing
June 2011

Spectroscopic and electronic structure studies of 2,3-dihydroxybiphenyl 1,2-dioxygenase: O2 reactivity of the non-heme ferrous site in extradiol dioxygenases.

J Am Chem Soc 2003 Sep;125(37):11214-27

Department of Chemistry and Stanford Synchrotron Radiation Laboratory, Stanford University, Stanford, California 94305-5080, USA.

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http://dx.doi.org/10.1021/ja029746iDOI Listing
September 2003

Crystal structure of prostate-specific membrane antigen, a tumor marker and peptidase.

Proc Natl Acad Sci U S A 2005 Apr 18;102(17):5981-6. Epub 2005 Apr 18.

Division of Biology 114-96 and Howard Hughes Medical Institute, California Institute of Technology, Pasadena, CA 91125, USA.

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http://www.pnas.org/cgi/doi/10.1073/pnas.0502101102
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http://dx.doi.org/10.1073/pnas.0502101102DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC556220PMC
April 2005

Spectroscopic Investigation of Reduced Protocatechuate 3,4-Dioxygenase: Charge-Induced Alterations in the Active Site Iron Coordination Environment.

Inorg Chem 1999 Aug;38(16):3676-3683

Department of Chemistry and Stanford Synchrotron Radiation Laboratory, Stanford University, Stanford, California 94305, and Department of Biochemistry and the Center for Metals in Biocatalysis, University of Minnesota, Minneapolis, Minnesota 55455.

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http://dx.doi.org/10.1021/ic981464pDOI Listing
August 1999