Publications by authors named "Michael S Christodoulou"

45Publications

Biological Properties of New Chiral 2-Methyl-5,6,7,8-tetrahydroquinolin-8-amine-based Compounds.

Molecules 2020 Nov 27;25(23). Epub 2020 Nov 27.

DISFARM, Sezione di Chimica Generale e Organica "A. Marchesini", Università degli Studi di Milano via Venezian, 21, 20133 Milano, Italy.

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November 2020

A small library of chalcones induce liver cancer cell death through Akt phosphorylation inhibition.

Sci Rep 2020 07 16;10(1):11814. Epub 2020 Jul 16.

CanSyL, Graduate School of Informatics, Middle East Technical University, 06800, Ankara, Turkey.

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July 2020

Antiproliferative effects of chalcones on T cell acute lymphoblastic leukemia-derived cells: Role of PKCβ.

Arch Pharm (Weinheim) 2020 Jul 12;353(7):e2000062. Epub 2020 May 12.

DISFARM, Sezione di Chimica Generale e Organica "A. Marchesini", Università degli Studi di Milano, Milano, Italy.

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July 2020

Divergent Conversion of 4-Naphthoquinone-substituted 4-Isoxazolones to Different Benzo-fused Indole Derivatives.

Org Lett 2020 Apr 17;22(7):2735-2739. Epub 2020 Mar 17.

Dipartimento di Scienza e Alta Tecnologia, Università degli Studi dell'Insubria, Via Valleggio 9, 22100 Como, Italy.

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April 2020

Novel 3,3-disubstituted oxindole derivatives. Synthesis and evaluation of the anti-proliferative activity.

Bioorg Med Chem Lett 2020 01 3;30(2):126845. Epub 2019 Dec 3.

DISFARM, Sezione di Chimica Generale e Organica "A. Marchesini" Università degli Studi di Milano, via Venezian 21, 20133 Milano, Italy.

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January 2020

Vancomycin-Iridium (III) Interaction: An Unexplored Route for Enantioselective Imine Reduction.

Molecules 2019 Jul 30;24(15). Epub 2019 Jul 30.

Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Venezian 21, 20133 Milano, Italy.

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July 2019

2-Phenyloxazole-4-carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B.

ChemMedChem 2019 09 7;14(18):1641-1652. Epub 2019 Aug 7.

Dipartimento di Scienze del Farmaco, Università degli Studi di Padova, Via F. Marzolo 5, 35131, Padova, Italy.

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September 2019

Cascade Reaction by Chemo- and Biocatalytic Approaches to Obtain Chiral Hydroxy Ketones and 1,3-Diols.

ChemistryOpen 2018 May 25;7(5):393-400. Epub 2018 May 25.

Dipartimento di Scienze Farmaceutiche Università degli Studi di Milano Via Venezian 21 20133 Milano Italia.

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May 2018

The 1,2,3-triazole ring as a bioisostere in medicinal chemistry.

Drug Discov Today 2017 10 1;22(10):1572-1581. Epub 2017 Jul 1.

Dipartimento di Chimica, Università degli Studi di Milano, Via Golgi 19, 20133 Milano, Italy. Electronic address:

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October 2017