Publications by authors named "Michael Kassiou"

176Publications

Reversing binding sensitivity to A147T translocator protein.

RSC Med Chem 2020 Apr 12;11(4):511-517. Epub 2020 Mar 12.

School of Chemistry , The University of Sydney , Sydney , New South Wales 2006 , Australia . Email:

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April 2020

The discovery of a potent and selective pyrazolo-[2,3-e]-[1,2,4]-triazine cannabinoid type 2 receptor agonist.

Eur J Med Chem 2021 Jan 5;210:113087. Epub 2020 Dec 5.

School of Chemistry, The University of Sydney, NSW, 2006, Australia. Electronic address:

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January 2021

Tricyclic heterocycles display diverse sensitivity to the A147T TSPO polymorphism.

Eur J Med Chem 2020 Dec 15;207:112725. Epub 2020 Aug 15.

School of Chemistry, Faculty of Science and the University of Sydney, NSW, 2006, Australia. Electronic address:

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December 2020

Rapid Antibacterial Activity of Cannabichromenic Acid against Methicillin-Resistant .

Antibiotics (Basel) 2020 Aug 16;9(8). Epub 2020 Aug 16.

Discipline of Infectious Diseases and Immunology, School of Medical Sciences, University of Sydney, Sydney, NSW 2006, Australia.

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August 2020

Novel Furan-2-yl-1-pyrazoles Possess Inhibitory Activity against α-Synuclein Aggregation.

ACS Chem Neurosci 2020 08 8;11(15):2303-2315. Epub 2020 Jul 8.

School of Pharmacy and Pharmacology, Griffith University, Gold Coast, Queensland 4222, Australia.

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August 2020

Anaesthetic-dependent changes in gene expression following acute and chronic exposure in the rodent brain.

Sci Rep 2020 06 9;10(1):9366. Epub 2020 Jun 9.

School of Chemistry, The University of Sydney, Sydney, NSW, Australia.

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June 2020

Differential activation of G protein-mediated signaling by synthetic cannabinoid receptor agonists.

Pharmacol Res Perspect 2020 04;8(2):e00566

Department of Biomedical Sciences, Macquarie University, Sydney, NSW, Australia.

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April 2020

Insight into the Structural Features of TSPO: Implications for Drug Development.

Trends Pharmacol Sci 2020 02 18;41(2):110-122. Epub 2019 Dec 18.

Department of Pharmacology and Pharmaceutical Sciences, School of Pharmacy, University of Southern California, Los Angeles, CA 90089, USA.

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February 2020

O-GlcNAcylation of truncated NAC segment alters peptide-dependent effects on α-synuclein aggregation.

Bioorg Chem 2020 01 9;94:103389. Epub 2019 Nov 9.

School of Pharmacy and Pharmacology, Griffith University, Gold Coast, QLD 4222, Australia; Menzies Health Institute Queensland, Griffith University, Gold Coast, QLD 4222, Australia; Quality Use of Medicines Network, Griffith University, Gold Coast, QLD 4222, Australia. Electronic address:

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January 2020

First Nondiscriminating Translocator Protein Ligands Produced from a Carbazole Scaffold.

J Med Chem 2019 09 28;62(17):8235-8248. Epub 2019 Aug 28.

Department of Biomedical Sciences, Faculty of Medicine and Health Sciences , Macquarie University , 2 Technology Place , North Ryde , New South Wales 2109 , Australia.

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September 2019

In vitro determination of the efficacy of illicit synthetic cannabinoids at CB receptors.

Br J Pharmacol 2019 12 10;176(24):4653-4665. Epub 2019 Dec 10.

Department of Biomedical Sciences, Macquarie University, Sydney, NSW, Australia.

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December 2019