Michael Delves

Michael Delves

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Michael Delves

Michael Delves

Publications by authors named "Michael Delves"

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Structure-Activity Relationship Studies of a Novel Class of Transmission Blocking Antimalarials Targeting Male Gametes.

J Med Chem 2020 Mar 20;63(5):2240-2262. Epub 2019 Sep 20.

Department of Chemistry, Imperial College London, Molecular Sciences Research Hub, White City Campus, Wood Lane, London W12 0BZ, United Kingdom.

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http://dx.doi.org/10.1021/acs.jmedchem.9b00898DOI Listing
March 2020

The antimalarial screening landscape-looking beyond the asexual blood stage.

Curr Opin Chem Biol 2019 06 12;50:1-9. Epub 2019 Mar 12.

Department of Life Sciences, Imperial College London, Sir Alexander Fleming Building, Exhibition Road, South Kensington, London SW7 2AZ, UK. Electronic address:

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http://dx.doi.org/10.1016/j.cbpa.2019.01.029DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6591700PMC
June 2019

Lysyl-tRNA synthetase as a drug target in malaria and cryptosporidiosis.

Proc Natl Acad Sci U S A 2019 04 20;116(14):7015-7020. Epub 2019 Mar 20.

Wellcome Centre for Anti-Infectives Research, Drug Discovery Unit, Division of Biological Chemistry and Drug Discovery, University of Dundee, DD1 5EH Dundee, United Kingdom;

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http://www.pnas.org/lookup/doi/10.1073/pnas.1814685116
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http://dx.doi.org/10.1073/pnas.1814685116DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6452685PMC
April 2019

8-Aminoquinolines with an Aminoxyalkyl Side Chain Exert in vitro Dual-Stage Antiplasmodial Activity.

ChemMedChem 2019 02 14;14(4):501-511. Epub 2019 Jan 14.

Institut für Pharmazeutische und Medizinische Chemie, Heinrich-Heine-Universität Düsseldorf, Universitätsstrasse 1, 40225, Düsseldorf, Germany.

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http://dx.doi.org/10.1002/cmdc.201800691DOI Listing
February 2019

Allele-Specific Isothermal Amplification Method Using Unmodified Self-Stabilizing Competitive Primers.

Anal Chem 2018 10 2;90(20):11972-11980. Epub 2018 Oct 2.

Centre for Bio-Inspired Technology, Department of Electrical and Electronic Engineering , Imperial College London , London , SW7 2AZ , United Kingdom.

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http://dx.doi.org/10.1021/acs.analchem.8b02416DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6195307PMC
October 2018

Adaptation of targeted nanocarriers to changing requirements in antimalarial drug delivery.

Nanomedicine 2017 02 5;13(2):515-525. Epub 2016 Oct 5.

Nanomalaria Group, Institute for Bioengineering of Catalonia (IBEC), Barcelona, Spain; Barcelona Institute for Global Health (ISGlobal), Barcelona Center for International Health Research (CRESIB, Hospital Clínic-Universitat de Barcelona), Barcelona, Spain; Nanoscience and Nanotechnology Institute (IN2UB), University of Barcelona, Barcelona, Spain. Electronic address:

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http://dx.doi.org/10.1016/j.nano.2016.09.010DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5332526PMC
February 2017

A Malaria Transmission-Blocking (+)-Usnic Acid Derivative Prevents Plasmodium Zygote-to-Ookinete Maturation in the Mosquito Midgut.

ACS Chem Biol 2016 12 17;11(12):3461-3472. Epub 2016 Nov 17.

W. Harry Feinstone Department of Molecular Microbiology and Immunology, Malaria Research Institute, Johns Hopkins Bloomberg School of Public Health , Baltimore, Maryland, United States.

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http://dx.doi.org/10.1021/acschembio.6b00902DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6503959PMC
December 2016

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond.

Authors:
Wesley C Van Voorhis John H Adams Roberto Adelfio Vida Ahyong Myles H Akabas Pietro Alano Aintzane Alday Yesmalie Alemán Resto Aishah Alsibaee Ainhoa Alzualde Katherine T Andrews Simon V Avery Vicky M Avery Lawrence Ayong Mark Baker Stephen Baker Choukri Ben Mamoun Sangeeta Bhatia Quentin Bickle Lotfi Bounaadja Tana Bowling Jürgen Bosch Lauren E Boucher Fabrice F Boyom Jose Brea Marian Brennan Audrey Burton Conor R Caffrey Grazia Camarda Manuela Carrasquilla Dee Carter Maria Belen Cassera Ken Chih-Chien Cheng Worathad Chindaudomsate Anthony Chubb Beatrice L Colon Daisy D Colón-López Yolanda Corbett Gregory J Crowther Noemi Cowan Sarah D'Alessandro Na Le Dang Michael Delves Joseph L DeRisi Alan Y Du Sandra Duffy Shimaa Abd El-Salam El-Sayed Michael T Ferdig José A Fernández Robledo David A Fidock Isabelle Florent Patrick V T Fokou Ani Galstian Francisco Javier Gamo Suzanne Gokool Ben Gold Todd Golub Gregory M Goldgof Rajarshi Guha W Armand Guiguemde Nil Gural R Kiplin Guy Michael A E Hansen Kirsten K Hanson Andrew Hemphill Rob Hooft van Huijsduijnen Takaaki Horii Paul Horrocks Tyler B Hughes Christopher Huston Ikuo Igarashi Katrin Ingram-Sieber Maurice A Itoe Ajit Jadhav Amornrat Naranuntarat Jensen Laran T Jensen Rays H Y Jiang Annette Kaiser Jennifer Keiser Thomas Ketas Sebastien Kicka Sunyoung Kim Kiaran Kirk Vidya P Kumar Dennis E Kyle Maria Jose Lafuente Scott Landfear Nathan Lee Sukjun Lee Adele M Lehane Fengwu Li David Little Liqiong Liu Manuel Llinás Maria I Loza Aristea Lubar Leonardo Lucantoni Isabelle Lucet Louis Maes Dalu Mancama Nuha R Mansour Sandra March Sheena McGowan Iset Medina Vera Stephan Meister Luke Mercer Jordi Mestres Alvine N Mfopa Raj N Misra Seunghyun Moon John P Moore Francielly Morais Rodrigues da Costa Joachim Müller Arantza Muriana Stephen Nakazawa Hewitt Bakela Nare Carl Nathan Nathalie Narraidoo Sujeevi Nawaratna Kayode K Ojo Diana Ortiz Gordana Panic George Papadatos Silvia Parapini Kailash Patra Ngoc Pham Sarah Prats David M Plouffe Sally-Ann Poulsen Anupam Pradhan Celia Quevedo Ronald J Quinn Christopher A Rice Mohamed Abdo Rizk Andrea Ruecker Robert St Onge Rafaela Salgado Ferreira Jasmeet Samra Natalie G Robinett Ulrich Schlecht Marjorie Schmitt Filipe Silva Villela Francesco Silvestrini Robert Sinden Dennis A Smith Thierry Soldati Andreas Spitzmüller Serge Maximilian Stamm David J Sullivan William Sullivan Sundari Suresh Brian M Suzuki Yo Suzuki S Joshua Swamidass Donatella Taramelli Lauve R Y Tchokouaha Anjo Theron David Thomas Kathryn F Tonissen Simon Townson Abhai K Tripathi Valentin Trofimov Kenneth O Udenze Imran Ullah Cindy Vallieres Edgar Vigil Joseph M Vinetz Phat Voong Vinh Hoan Vu Nao-Aki Watanabe Kate Weatherby Pamela M White Andrew F Wilks Elizabeth A Winzeler Edward Wojcik Melanie Wree Wesley Wu Naoaki Yokoyama Paul H A Zollo Nada Abla Benjamin Blasco Jeremy Burrows Benoît Laleu Didier Leroy Thomas Spangenberg Timothy Wells Paul A Willis

PLoS Pathog 2016 07 28;12(7):e1005763. Epub 2016 Jul 28.

Medicines for Malaria Venture, Geneva, Switzerland.

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http://dx.doi.org/10.1371/journal.ppat.1005763DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4965013PMC
July 2016

Changes in metabolic phenotypes of Plasmodium falciparum in vitro cultures during gametocyte development.

Malar J 2014 Dec 1;13:468. Epub 2014 Dec 1.

Department of Life Sciences, Imperial College London, London SW7 2AZ, UK.

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http://dx.doi.org/10.1186/1475-2875-13-468DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4289216PMC
December 2014

Laboratory maintenance of rodent malaria parasites.

Methods Mol Biol 2013 ;923:51-72

The Malaria Centre, Department of Life Sciences, Imperial College, London, UK.

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http://dx.doi.org/10.1007/978-1-62703-026-7_5DOI Listing
January 2013

Assessing transmission blockade in Plasmodium spp.

Methods Mol Biol 2013 ;923:577-600

The Malaria Centre, Department of Life Sciences, Imperial College, London, UK.

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http://link.springer.com/10.1007/978-1-62703-026-7_40
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http://dx.doi.org/10.1007/978-1-62703-026-7_40DOI Listing
January 2013

Plasmodium cell biology should inform strategies used in the development of antimalarial transmission-blocking drugs.

Authors:
Michael J Delves

Future Med Chem 2012 Dec;4(18):2251-63

Cell & Molecular Biology, Imperial College, South Kensington, London, SW7 2AZ, UK.

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http://dx.doi.org/10.4155/fmc.12.182DOI Listing
December 2012

The design and interpretation of laboratory assays measuring mosquito transmission of Plasmodium.

Trends Parasitol 2012 Nov 11;28(11):457-65. Epub 2012 Sep 11.

The Malaria Centre, Imperial College London, South Kensington, London SW7 2AZ, UK.

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http://dx.doi.org/10.1016/j.pt.2012.07.005DOI Listing
November 2012

A GFP-actin reporter line to explore microfilament dynamics across the malaria parasite lifecycle.

Mol Biochem Parasitol 2012 Mar-Apr;182(1-2):93-6. Epub 2011 Nov 25.

Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, 3052, Australia.

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http://dx.doi.org/10.1016/j.molbiopara.2011.11.008DOI Listing
May 2012

Plasmodium male development gene-1 (mdv-1) is important for female sexual development and identifies a polarised plasma membrane during zygote development.

Int J Parasitol 2009 Jun 24;39(7):755-61. Epub 2008 Dec 24.

The Division of Cell and Molecular Biology, Imperial College London, London, UK.

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http://dx.doi.org/10.1016/j.ijpara.2008.11.008DOI Listing
June 2009