Publications by authors named "Mark Rau"

6Publications

Synthesis and Biological Evaluation of Endocannabinoid Uptake Inhibitors Derived from WOBE437.

ChemMedChem 2020 May 5. Epub 2020 May 5.

Department of Chemistry and Applied Biosciences, ETH Zürich HCI H405, Vladimir-Prelog-Weg 4, 8093, Zürich, Switzerland.

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http://dx.doi.org/10.1002/cmdc.202000153DOI Listing
May 2020

Total Synthesis of the Endocannabinoid Uptake Inhibitor Guineensine and SAR Studies.

ChemMedChem 2019 09 23;14(17):1590-1596. Epub 2019 Aug 23.

Department of Chemistry and Applied Biosciences, ETH Zürich, HCI H405, Vladimir-Prelog-Weg 4, 8093, Zürich, Switzerland.

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http://dx.doi.org/10.1002/cmdc.201900390DOI Listing
September 2019

Assay of Endocannabinoid Uptake.

Methods Mol Biol 2016 ;1412:191-203

Institute of Biochemistry and Molecular Medicine, NCCR TransCure, University of Bern, Bern, Switzerland.

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http://dx.doi.org/10.1007/978-1-4939-3539-0_20DOI Listing
December 2017

Correlating FAAH and anandamide cellular uptake inhibition using N-alkylcarbamate inhibitors: from ultrapotent to hyperpotent.

Biochem Pharmacol 2014 Dec 4;92(4):669-89. Epub 2014 Nov 4.

Institute of Biochemistry and Molecular Medicine, NCCR TransCure, University of Bern, Bühlstrasse 28, CH-3012 Bern, Switzerland. Electronic address:

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http://dx.doi.org/10.1016/j.bcp.2014.09.020DOI Listing
December 2014

Identification of endocannabinoid system-modulating N-alkylamides from Heliopsis helianthoides var. scabra and Lepidium meyenii.

J Nat Prod 2014 Jul 27;77(7):1663-9. Epub 2014 Jun 27.

Department of Pharmacognosy, University of Szeged , H-6720 Szeged, Hungary.

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http://pubs.acs.org/doi/10.1021/np500292g
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http://dx.doi.org/10.1021/np500292gDOI Listing
July 2014

Guineensine is a novel inhibitor of endocannabinoid uptake showing cannabimimetic behavioral effects in BALB/c mice.

Pharmacol Res 2014 Feb 8;80:52-65. Epub 2014 Jan 8.

Institute of Biochemistry and Molecular Medicine, NCCR TransCure, University of Bern, CH-3012 Bern, Switzerland. Electronic address:

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http://dx.doi.org/10.1016/j.phrs.2013.12.010DOI Listing
February 2014