Publications by authors named "Maria Concepcion Garcia Alvarez"

14Publications

N,N-bis-heteroaryl methylamines: Potent anti-mitotic and highly cytotoxic agents.

Eur J Med Chem 2019 Apr 16;168:176-188. Epub 2019 Feb 16.

BioCIS, Univ. Paris-Sud, CNRS, Université Paris-Saclay, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2019.02.038DOI Listing
April 2019

N-myristoyltransferases inhibitory activity of ellagitannins from Terminalia bentzoë (L.) L. f. subsp. bentzoë.

Fitoterapia 2018 Nov 17;131:91-95. Epub 2018 Oct 17.

Institut de Chimie des Substances Naturelles, CNRS-ICSN, UPR 2301, Université Paris-Saclay, 91198 cedex, Gif-sur-Yvette, France. Electronic address:

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http://dx.doi.org/10.1016/j.fitote.2018.10.014DOI Listing
November 2018

Inhibition of p53-Murine Double Minute 2 (MDM2) Interactions with 3,3'-Spirocyclopentene Oxindole Derivatives.

J Med Chem 2018 10 8;61(20):9386-9392. Epub 2018 Oct 8.

Institut de Chimie des Substances Naturelles, CNRS UPR 2301, Université Paris-Sud, Université Paris-Saclay , 1, Avenue de la Terrasse , 91198 Gif-sur-Yvette , France.

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http://dx.doi.org/10.1021/acs.jmedchem.8b01137DOI Listing
October 2018

Original Vinca Derivatives: From P-Glycoprotein Substrates to P-Glycoprotein Inhibitors.

J Med Chem 2016 12 23;59(23):10774-10780. Epub 2016 Nov 23.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, UPR 2301 du CNRS, Université Paris-Saclay , 1 Avenue de la Terrasse, 91198, Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1021/acs.jmedchem.6b00525DOI Listing
December 2016

Synthesis and biological evaluation of C-13' substituted 7'-homo-anhydrovinblastine derivatives.

Bioorg Med Chem Lett 2015 Apr 7;25(8):1771-1773. Epub 2015 Mar 7.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, UPR 2301 du CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2015.02.045DOI Listing
April 2015

One-pot synthesis of vinca alkaloids-phomopsin hybrids.

J Med Chem 2014 Jun 10;57(12):5470-6. Epub 2014 Jun 10.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, UPR 2301 du CNRS, Avenue de la Terrasse, 91198, Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1021/jm500530vDOI Listing
June 2014

A concise formation of N-substituted 3,4-diarylpyrroles--synthesis and cytotoxic activity.

Org Biomol Chem 2014 Mar;12(9):1518-24

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1039/c3ob42309cDOI Listing
March 2014

Synthesis and biological evaluation of a new series of highly functionalized 7'-homo-anhydrovinblastine derivatives.

J Med Chem 2013 Aug 18;56(15):6088-100. Epub 2013 Jul 18.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, UPR 2301 du CNRS, LabEx Lermit, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1021/jm4004347DOI Listing
August 2013

UPLC-ESI-MS analysis of thymosins β4 and β10 in cell lysates: a simple, rapid and sensitive quantification method.

Anal Methods 2011 Mar;3(3):678-682

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198, Gif-sur-Yvette Cedex, France.

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http://dx.doi.org/10.1039/c0ay00576bDOI Listing
March 2011

Overexpression of the natural tetrapeptide acetyl-N-ser-asp-lys-pro derived from thymosin beta4 in neoplastic diseases.

Ann N Y Acad Sci 2010 Apr;1194:53-9

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette, France.

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http://dx.doi.org/10.1111/j.1749-6632.2010.05488.xDOI Listing
April 2010

In vitro and in vivo properties of ellagic acid in malaria treatment.

Antimicrob Agents Chemother 2009 Mar 17;53(3):1100-6. Epub 2008 Nov 17.

Service de Parasitologie, Toulouse Hospital University, TSA50032, Toulouse Cedex 9, France.

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http://dx.doi.org/10.1128/AAC.01175-08DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2650562PMC
March 2009