Publications by authors named "Maria Antonietta Stasi"

14Publications

Hedgehog pathway inhibitors of the acylthiourea and acylguanidine class show antitumor activity on colon cancer in vitro and in vivo.

Authors:
Loredana Vesci Ferdinando Maria Milazzo Maria Antonietta Stasi Silvia Pace Francesco Manera Carlo Tallarico Elena Cini Elena Petricci Fabrizio Manetti Rita De Santis Giuseppe Giannini

Eur J Med Chem 2018 Sep 27;157:368-379. Epub 2018 Jul 27.

Research & Development, Alfasigma SpA, via Pontina, Km 30.400, I-00040, Pomezia, Italy. Electronic address:

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September 2018

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands.

Authors:
Silvia Pace Giandomenico Brogin Maria Antonietta Stasi Teresa Riccioni Franco Borsini Francesca Capocasa Francesco Manera Carlo Tallarico Pietro Grossi Federica Vacondio Michele Bassi Francesca Bartoccini Simone Lucarini Giovanni Piersanti Giorgio Tarzia Walter Cabri Patrizia Minetti

ChemMedChem 2015 Jul 7;10(7):1149-52. Epub 2015 May 7.

Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. Via Pontina Km 30, 400, 00040 Pomezia (Italy).

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July 2015

Animal models of Parkinson׳s disease: Effects of two adenosine A2A receptor antagonists ST4206 and ST3932, metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535).

Authors:
Maria Antonietta Stasi Patrizia Minetti Katia Lombardo Teresa Riccioni Antonio Caprioli Mario Vertechy Stefano Di Serio Silvia Pace Franco Borsini

Eur J Pharmacol 2015 Aug 30;761:353-61. Epub 2015 Apr 30.

Research & Development Area, Sigma-tau, Italy.

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August 2015

Propionyl-L-Carnitine is Efficacious in Ulcerative Colitis Through its Action on the Immune Function and Microvasculature.

Authors:
Maria Giovanna Scioli Maria Antonietta Stasi Daniela Passeri Elena Doldo Gaetana Costanza Roberto Camerini Paolo Fociani Gaetano Arcuri Katia Lombardo Silvia Pace Franco Borsini Augusto Orlandi

Clin Transl Gastroenterol 2014 Mar 20;5:e55. Epub 2014 Mar 20.

Anatomic Pathology, Tor Vergata University, Rome, Italy.

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March 2014

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

Authors:
Giovanni Piersanti Francesca Bartoccini Simone Lucarini Walter Cabri Maria Antonietta Stasi Teresa Riccioni Franco Borsini Giorgio Tarzia Patrizia Minetti

J Med Chem 2013 Jul 24;56(13):5456-63. Epub 2013 Jun 24.

Dipartimento di Scienze Biomolecolari, Università degli Studi di Urbino , Piazza Rinascimento 6, I-61029 Urbino (PU), Italy.

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July 2013

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

Authors:
Silvia Rivara Giovanni Piersanti Francesca Bartoccini Giuseppe Diamantini Daniele Pala Teresa Riccioni Maria Antonietta Stasi Walter Cabri Franco Borsini Marco Mor Giorgio Tarzia Patrizia Minetti

J Med Chem 2013 Feb 16;56(3):1247-61. Epub 2013 Jan 16.

Dipartimento di Farmacia, Università degli Studi di Parma, Viale G.P. Usberti 27 A, I-43124 Parma, Italy.

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February 2013

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases.

Authors:
Stefania Butini Margherita Brindisi Sandra Gemma Patrizia Minetti Walter Cabri Grazia Gallo Silvia Vincenti Emanuela Talamonti Franco Borsini Antonio Caprioli Maria Antonietta Stasi Stefano Di Serio Sindu Ros Giuseppe Borrelli Samuele Maramai Filomena Fezza Giuseppe Campiani Mauro Maccarrone

J Med Chem 2012 Aug 26;55(15):6898-915. Epub 2012 Jul 26.

European Research Centre for Drug Discovery and Development (NatSynDrugs), Università degli Studi di Siena , Via Aldo Moro 2, 53100 Siena, Italy.

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August 2012

The effects of clozapine on quinpirole-induced non-regulatory drinking and prepulse inhibition disruption in rats.

Authors:
Lorenza De Carolis Maria Antonietta Stasi Ottaviano Serlupi-Crescenzi Franco Borsini Paolo Nencini

Psychopharmacology (Berl) 2010 Sep 10;212(1):105-15. Epub 2010 Jul 10.

Department of Physiology and Pharmacology "Vittorio Erspamer", Sapienza University of Rome, Italy.

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September 2010

Propionyl-L-carnitine improves postischemic blood flow recovery and arteriogenetic revascularization and reduces endothelial NADPH-oxidase 4-mediated superoxide production.

Authors:
Maria Antonietta Stasi Maria Giovanna Scioli Gaetano Arcuri Giovan Giuseppe Mattera Katia Lombardo Marcella Marcellini Teresa Riccioni Sandro De Falco Claudio Pisano Luigi Giusto Spagnoli Franco Borsini Augusto Orlandi

Arterioscler Thromb Vasc Biol 2010 Mar 7;30(3):426-35. Epub 2010 Jan 7.

Dept. of Biopathology and Image Diagnostics, Tor Vergata University of Rome, Via Montpellier, 00133 Rome, Italy.

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March 2010

Effects of ST2472, a novel antipsychotic, on prepulse inhibition.

Authors:
Katia Lombardo Maria Antonietta Stasi Franco Borsini

Eur J Pharmacol 2009 Oct 6;621(1-3):53-60. Epub 2009 Sep 6.

Central & Peripheral Nervous System and General Pharmacology Department, R&D, Sigma-Tau Industrie Farmaceutiche Riunite SpA, Pomezia Rome, Italy.

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October 2009

Haloperidol both prevents and reverses quinpirole-induced nonregulatory water intake, a putative animal model of psychogenic polydipsia.

Authors:
Davide Amato Maria Antonietta Stasi Franco Borsini Paolo Nencini

Psychopharmacology (Berl) 2008 Oct 3;200(2):157-65. Epub 2008 Jul 3.

Department of Human Physiology and Pharmacology "Vittorio Erspamer", University of Rome "La Sapienza", Piazzale Aldo Moro 5, 00185, Rome, Italy.

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October 2008

ST 1535: a preferential A2A adenosine receptor antagonist.

Authors:
Maria Antonietta Stasi Franco Borsini Katia Varani Fabrizio Vincenzi Maria Assunta Di Cesare Patrizia Minetti Orlando Ghirardi Paolo Carminati

Int J Neuropsychopharmacol 2006 Oct 23;9(5):575-84. Epub 2005 Nov 23.

Sigma-Tau Industrie Farmaceutiche Riunite S.p.A., Pomezia (Rome), Italy.

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October 2006

Ameliorating effects of the immunomodulator 3-(2-ethylphenyl)-5-(3-methoxyphenyl)-1H-1,2,4-triazole in an experimental model of colitis in the rat.

Authors:
Maria Antonietta Stasi Vito Ruggiero Angela Ursillo Roberto Taurelli Margherita Aglianò Elisabetta Weber Paola Lorenzoni Vincenzo Sorrentino Licia Pacifici Paolo Carminati

Eur J Pharmacol 2004 Jun;494(2-3):263-72

Pharmacology Department-R&D, Sigma-tau S.p.A., Via Pontina km 30.400, 00040 Pomezia (RM), Italy.

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June 2004

EEG power spectra changes and forebrain ischemia in rats.

Authors:
Giuseppina Mariucci Maria Antonietta Stasi Roberto Taurelli Paolo Nardò Michela Tantucci Licia Pacifici Paolo Carminati Maria Vittoria Ambrosini

Can J Neurol Sci 2003 Feb;30(1):54-60

Department of Experimental Medicine and Biochemical Sciences, University of Perugia, Perugia, Italy.

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February 2003