Louis Maes

Louis Maes

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HPLC-DAD-SPE-NMR isolation of tetracyclic spiro-alkaloids with antiplasmodial activity from the seeds of .

Nat Prod Res 2020 Apr 3;34(7):1037-1040. Epub 2019 Jan 3.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Antwerp, Belgium.

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http://dx.doi.org/10.1080/14786419.2018.1539976DOI Listing
April 2020

C6-O-alkylated 7-deazainosine nucleoside analogues: Discovery of potent and selective anti-sleeping sickness agents.

Eur J Med Chem 2020 Feb 3;188:112018. Epub 2020 Jan 3.

Laboratory for Medicinal Chemistry (Campus Heymans), Ghent University, Ottergemsesteenweg 460, B-9000, Gent, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2019.112018DOI Listing
February 2020

Phenotypic adaptations of Leishmania donovani to recurrent miltefosine exposure and impact on sand fly infection.

Parasit Vectors 2020 Feb 22;13(1):96. Epub 2020 Feb 22.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Antwerp, Belgium.

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http://dx.doi.org/10.1186/s13071-020-3972-zDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7036194PMC
February 2020

Bioactive Metabolites of Marine Origin Have Unusual Effects on Model Membrane Systems.

Mar Drugs 2020 Feb 19;18(2). Epub 2020 Feb 19.

Department of Biological Sciences, University of Bergen, Thormøhlensgate 55, NO-5006 Bergen, Norway.

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http://dx.doi.org/10.3390/md18020125DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7073740PMC
February 2020

Structure-activity relationship of 4-azaindole-2-piperidine derivatives as agents against Trypanosoma cruzi.

Bioorg Med Chem Lett 2020 Jan 31;30(1):126779. Epub 2019 Oct 31.

Institute of Chemistry, University of Campinas (UNICAMP), Rua Josué de Castro, S/N, Cidade Universitária, Campinas, SP 13083-861, Brazil. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2019.126779DOI Listing
January 2020

Identification of Phenylphthalazinones as a New Class of Leishmania infantum Inhibitors.

ChemMedChem 2020 Jan 9;15(2):219-227. Epub 2019 Dec 9.

Division of Medicinal Chemistry, Faculty of Sciences, Amsterdam Institute for Molecules, Medicines and Systems (AIMMS), Vrije Universiteit Amsterdam, De Boelelaan 1108, 1081 HZ, Amsterdam, The Netherlands.

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http://dx.doi.org/10.1002/cmdc.201900538DOI Listing
January 2020

In Vitro Growth Inhibition Assays of Leishmania spp.

Methods Mol Biol 2020 ;2116:791-800

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Wilrijk-Antwerp, Belgium.

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http://dx.doi.org/10.1007/978-1-0716-0294-2_47DOI Listing
January 2020

Impaired development of a miltefosine-resistant Leishmania infantum strain in the sand fly vectors Phlebotomus perniciosus and Lutzomyia longipalpis.

Int J Parasitol Drugs Drug Resist 2019 12 10;11:1-7. Epub 2019 Sep 10.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, B-2610, Wilrijk, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.ijpddr.2019.09.003DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6804374PMC
December 2019

In-depth comparison of cell-based methodological approaches to determine drug susceptibility of visceral Leishmania isolates.

PLoS Negl Trop Dis 2019 12 2;13(12):e0007885. Epub 2019 Dec 2.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Antwerp, Belgium.

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http://dx.doi.org/10.1371/journal.pntd.0007885DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6907865PMC
December 2019

The synthesis and in vitro biological evaluation of novel fluorinated tetrahydrobenzo[j]phenanthridine-7,12-diones against Mycobacterium tuberculosis.

Eur J Med Chem 2019 Nov 19;181:111549. Epub 2019 Jul 19.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Universiteitsplein 1, B-2610, Wilrijk, Belgium.

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http://dx.doi.org/10.1016/j.ejmech.2019.07.052DOI Listing
November 2019

Isolation and Characterization of Clinical RSV Isolates in Belgium during the Winters of 2016-2018.

Viruses 2019 Nov 6;11(11). Epub 2019 Nov 6.

Laboratory of Microbiology, Parasitology and Hygiene, and Infla-Med Centre of Excellence, University of Antwerp (UA), Universiteitsplein 1 S.7, 2610 Antwerp, Belgium.

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http://dx.doi.org/10.3390/v11111031DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6893609PMC
November 2019

In vitro and in vivo antiplasmodial activity of extracts and isolated constituents of Alstonia congensis root bark.

J Ethnopharmacol 2019 Oct 11;242:111736. Epub 2019 Feb 11.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Universiteitsplein 1, B-2610 Antwerp, Belgium.

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http://dx.doi.org/10.1016/j.jep.2019.02.019DOI Listing
October 2019

Discovery of Pyrrolo[2,3-]pyridine (1,7-Dideazapurine) Nucleoside Analogues as Anti- Agents.

J Med Chem 2019 Oct 20;62(19):8847-8865. Epub 2019 Sep 20.

Laboratory for Medicinal Chemistry (Campus Heymans) , Ghent University , Ottergemsesteenweg 460 , B-9000 Gent , Belgium.

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http://dx.doi.org/10.1021/acs.jmedchem.9b01275DOI Listing
October 2019

Identification of Phenylpyrazolone Dimers as a New Class of Anti-Trypanosoma cruzi Agents.

ChemMedChem 2019 Sep 23;14(18):1662-1668. Epub 2019 Aug 23.

Division of Medicinal Chemistry, Faculty of Sciences, Amsterdam Institute for Molecules, Medicines and Systems (AIMMS), Vrije Universiteit Amsterdam, De Boelelaan 1108, 1081 HZ, Amsterdam, The Netherlands.

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http://dx.doi.org/10.1002/cmdc.201900370DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6771560PMC
September 2019

Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors.

Bioorg Med Chem 2019 Sep 18;27(18):3998-4012. Epub 2019 Jun 18.

Division of Medicinal Chemistry, Amsterdam Institute for Molecules, Medicines and Systems, Vrije Universiteit Amsterdam, De Boelelaan 1108, 1081 HZ Amsterdam, The Netherlands. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2019.06.027DOI Listing
September 2019

Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2).

Bioorg Med Chem 2019 Sep 5;27(18):4013-4029. Epub 2019 Jul 5.

Division of Medicinal Chemistry, Amsterdam Institute for Molecules, Medicines and Systems, Vrije Universiteit Amsterdam, 1081 HZ Amsterdam, The Netherlands. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2019.06.026DOI Listing
September 2019

Double prodrugs of a fosmidomycin surrogate as antimalarial and antitubercular agents.

Bioorg Med Chem Lett 2019 05 7;29(10):1232-1235. Epub 2019 Mar 7.

Laboratory for Medicinal Chemistry, Ghent University, Ottergemsesteenweg 460, B-9000 Ghent, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2019.03.009DOI Listing
May 2019

Amino acid based prodrugs of a fosmidomycin surrogate as antimalarial and antitubercular agents.

Bioorg Med Chem 2019 03 17;27(5):729-747. Epub 2019 Jan 17.

Laboratory for Medicinal Chemistry, Ghent University, Ottergemsesteenweg 460, B-9000 Ghent, Belgium. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S09680896183195
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http://dx.doi.org/10.1016/j.bmc.2019.01.016DOI Listing
March 2019

Miltefosine enhances the fitness of a non-virulent drug-resistant Leishmania infantum strain.

J Antimicrob Chemother 2019 02;74(2):395-406

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Wilrijk, Belgium.

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http://fdslive.oup.com/www.oup.com/pdf/production_in_progres
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http://dx.doi.org/10.1093/jac/dky450DOI Listing
February 2019

Synthesis and antimicrobial activities of N-hydroxyagelasine analogs and revision of the structure of ageloximes.

Bioorg Med Chem 2019 02 4;27(4):620-629. Epub 2019 Jan 4.

Department of Chemistry, University of Oslo, P.O.Box 1033, Blindern, 0315 Oslo, Norway. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2019.01.002DOI Listing
February 2019

Revisiting tubercidin against kinetoplastid parasites: Aromatic substitutions at position 7 improve activity and reduce toxicity.

Eur J Med Chem 2019 Feb 21;164:689-705. Epub 2018 Dec 21.

Laboratory for Medicinal Chemistry (Campus Heymans), Ghent University, Ottergemsesteenweg 460, B-9000, Gent, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2018.12.050DOI Listing
February 2019

Optimization and Characterization of a Larval Infection Model for Virulence Studies and the Evaluation of Therapeutics Against .

Front Microbiol 2019 21;10:311. Epub 2019 Feb 21.

Laboratory of Microbiology, Parasitology and Hygiene, Department of Pharmaceutical Sciences, University of Antwerp, Wilrijk, Belgium.

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http://dx.doi.org/10.3389/fmicb.2019.00311DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6394149PMC
February 2019

Discovery of Novel, Drug-Like Ferroptosis Inhibitors with in Vivo Efficacy.

J Med Chem 2018 11 6;61(22):10126-10140. Epub 2018 Nov 6.

Laboratory of Medicinal Chemistry , University of Antwerp , Universiteitsplein 1 , 2610 Antwerp , Belgium.

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http://pubs.acs.org/doi/10.1021/acs.jmedchem.8b01299
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http://dx.doi.org/10.1021/acs.jmedchem.8b01299DOI Listing
November 2018

Discovery of Novel 7-Aryl 7-Deazapurine 3'-Deoxy-ribofuranosyl Nucleosides with Potent Activity against Trypanosoma cruzi.

J Med Chem 2018 10 3;61(20):9287-9300. Epub 2018 Oct 3.

Laboratory for Medicinal Chemistry (Campus Heymans) , Ghent University , Ottergemsesteenweg 460 , Gent B-9000 , Belgium.

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http://dx.doi.org/10.1021/acs.jmedchem.8b00999DOI Listing
October 2018

Discovery of benzimidazole-based Leishmania mexicana cysteine protease CPB2.8ΔCTE inhibitors as potential therapeutics for leishmaniasis.

Chem Biol Drug Des 2018 09 31;92(3):1585-1596. Epub 2018 May 31.

Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, Messina, Italy.

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http://doi.wiley.com/10.1111/cbdd.13326
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http://dx.doi.org/10.1111/cbdd.13326DOI Listing
September 2018

Optimization of the pharmacokinetic properties of potent anti-trypanosomal triazine derivatives.

Eur J Med Chem 2018 May 23;151:18-26. Epub 2018 Mar 23.

Laboratory of Medicinal Chemistry, University of Antwerp, Universiteitsplein 1, B-2610, Antwerp, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2018.03.048DOI Listing
May 2018

Synthesis and in vitro investigation of halogenated 1,3-bis(4-nitrophenyl)triazenide salts as antitubercular compounds.

Chem Biol Drug Des 2018 02 14;91(2):631-640. Epub 2017 Sep 14.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), S7, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Wilrijk, Belgium.

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http://dx.doi.org/10.1111/cbdd.13087DOI Listing
February 2018

Ensemble-based ADME-Tox profiling and virtual screening for the discovery of new inhibitors of the Leishmania mexicana cysteine protease CPB2.8ΔCTE.

Chem Biol Drug Des 2018 02 10;91(2):597-604. Epub 2017 Nov 10.

Dipartimento di Scienze Chimiche, Biologiche, Farmaceutiche ed Ambientali, Università di Messina, Messina, Italy.

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http://dx.doi.org/10.1111/cbdd.13124DOI Listing
February 2018

Miltefosine-resistant Leishmania infantum strains with an impaired MT/ROS3 transporter complex retain amphotericin B susceptibility.

J Antimicrob Chemother 2018 02;73(2):392-394

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, B-2610 Wilrijk, Belgium.

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http://dx.doi.org/10.1093/jac/dkx407DOI Listing
February 2018

UPLC/MS MS data of testosterone metabolites in human and zebrafish liver microsomes and whole zebrafish larval microsomes.

Data Brief 2018 Feb 6;16:644-648. Epub 2017 Dec 6.

Applied Veterinary Morphology, Department of Veterinary Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Universiteitsplein 1, B-2610 Wilrijk, Belgium.

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http://dx.doi.org/10.1016/j.dib.2017.11.079DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5847491PMC
February 2018

Novel triazine dimers with potent antitrypanosomal activity.

Eur J Med Chem 2018 Jan 27;143:306-319. Epub 2017 Nov 27.

Laboratory of Medicinal Chemistry, University of Antwerp, Universiteitsplein 1, B-2610 Antwerp, Belgium. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S02235234173097
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http://dx.doi.org/10.1016/j.ejmech.2017.11.075DOI Listing
January 2018

In vitro CYP-mediated drug metabolism in the zebrafish (embryo) using human reference compounds.

Toxicol In Vitro 2017 Aug 12;42:329-336. Epub 2017 May 12.

Applied Veterinary Morphology, Department of Veterinary Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Universiteitsplein 1, B-2610 Wilrijk, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.tiv.2017.05.009DOI Listing
August 2017

Optimization and characterization of a murine lung infection model for the evaluation of novel therapeutics against Burkholderia cenocepacia.

J Microbiol Methods 2017 08 3;139:181-188. Epub 2017 Jun 3.

Laboratory for Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, 2610 Wilrijk, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.mimet.2017.06.003DOI Listing
August 2017

Comparative analysis of the internalization of the macrophage receptor sialoadhesin in human and mouse primary macrophages and cell lines.

Immunobiology 2017 06 21;222(6):797-806. Epub 2016 Nov 21.

Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp (UA), Antwerp 2610, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.imbio.2016.11.013DOI Listing
June 2017

6-Nitro-2,3-dihydroimidazo[2,1-b][1,3]thiazoles: Facile synthesis and comparative appraisal against tuberculosis and neglected tropical diseases.

Bioorg Med Chem Lett 2017 06 27;27(11):2583-2589. Epub 2017 Mar 27.

Auckland Cancer Society Research Centre, School of Medical Sciences, The University of Auckland, Private Bag 92019, Auckland 1142, New Zealand.

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http://dx.doi.org/10.1016/j.bmcl.2017.03.069DOI Listing
June 2017

Combined treatment of miltefosine and paromomycin delays the onset of experimental drug resistance in Leishmania infantum.

PLoS Negl Trop Dis 2017 May 15;11(5):e0005620. Epub 2017 May 15.

Laboratory for Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Antwerp, Belgium.

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http://dx.doi.org/10.1371/journal.pntd.0005620DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5444850PMC
May 2017

and Antidiabetic and Antimicrobial Evaluation of Constituents from ().

Front Pharmacol 2017 1;8:232. Epub 2017 May 1.

Laboratory of Natural Products and Food Research and Analysis, Department of Pharmaceutical Sciences, University of AntwerpAntwerp, Belgium.

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http://dx.doi.org/10.3389/fphar.2017.00232DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5410595PMC
May 2017

Gold compounds as cysteine protease inhibitors: perspectives for pharmaceutical application as antiparasitic agents.

Biometals 2017 04 10;30(2):313-320. Epub 2017 Mar 10.

Department of Chemistry and Industrial Chemistry, University of Pisa, via Moruzzi, 13, 56124, Pisa, Italy.

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http://dx.doi.org/10.1007/s10534-017-0007-0DOI Listing
April 2017

Antiprotozoal activity of major constituents from the bioactive fraction of Verbesina encelioides.

Nat Prod Res 2017 Mar 6;31(6):676-680. Epub 2016 May 6.

a Faculty of Pharmacy, Department of Pharmacognosy , Cairo University , Cairo , Egypt.

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http://dx.doi.org/10.1080/14786419.2016.1180604DOI Listing
March 2017

Monoclonal antibody binding to the macrophage-specific receptor sialoadhesin alters the phagocytic properties of human and mouse macrophages.

Cell Immunol 2017 02 9;312:51-60. Epub 2016 Dec 9.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp (UA), Antwerp 2610, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.cellimm.2016.11.009DOI Listing
February 2017

Antiplasmodial Activity, Cytotoxicity and Structure-Activity Relationship Study of Cyclopeptide Alkaloids.

Molecules 2017 Feb 2;22(2). Epub 2017 Feb 2.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Universiteitsplein 1, 2610 Antwerp, Belgium.

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http://dx.doi.org/10.3390/molecules22020224DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6155665PMC
February 2017

In-vivo evaluation of apocynin for prevention of Helicobacter pylori-induced gastric carcinogenesis.

Eur J Cancer Prev 2017 01;26(1):10-16

aLaboratory of Microbiology, Parasitology and Hygiene (LMPH), Faculty of Pharmaceutical, Biomedical and Veterinary Sciences bLaboratory for Cell Biology and Histology, University of Antwerp, Antwerp cLaboratory of Pharmaceutical Technology, Department of Pharmaceutics, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.

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http://dx.doi.org/10.1097/CEJ.0000000000000233DOI Listing
January 2017

Pharmacomodulation of the Antimalarial Plasmodione: Synthesis of Biaryl- and N-Arylalkylamine Analogues, Antimalarial Activities and Physicochemical Properties.

Molecules 2017 Jan 19;22(1). Epub 2017 Jan 19.

UMR 7509 CNRS-Université de Strasbourg, Bioorganic and Medicinal Chemistry Team, European School of Chemistry, Polymers and Materials (ECPM), 25, rue Becquerel, F-67087 Strasbourg, France.

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http://dx.doi.org/10.3390/molecules22010161DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6155649PMC
January 2017

Triterpenoid Saponins from Maesa argentea Leaves.

Planta Med 2016 Dec 13;82(18):1568-1575. Epub 2016 Oct 13.

Natural Products & Food Research and Analysis, Department of Pharmaceutical Sciences, University of Antwerp, Antwerp, Belgium.

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http://dx.doi.org/10.1055/s-0042-118189DOI Listing
December 2016

Isolation and Structure Elucidation by LC-DAD-MS and LC-DAD-SPE-NMR of Cyclopeptide Alkaloids from the Roots of Ziziphus oxyphylla and Evaluation of Their Antiplasmodial Activity.

J Nat Prod 2016 11 10;79(11):2865-2872. Epub 2016 Nov 10.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, and ‡Laboratory of Microbiology, Parasitology and Hygiene (LMPH), Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp , Universiteitsplein 1, 2610 Antwerp, Belgium.

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http://dx.doi.org/10.1021/acs.jnatprod.6b00633DOI Listing
November 2016

Phytochemical and Pharmacological Investigations on Nymphoides indica Leaf Extracts.

Phytother Res 2016 Oct 10;30(10):1624-1633. Epub 2016 Jun 10.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Universiteitsplein 1, 2610, Antwerp, Belgium.

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http://dx.doi.org/10.1002/ptr.5663DOI Listing
October 2016

Molecular detection of infection homogeneity and impact of miltefosine treatment in a Syrian golden hamster model of Leishmania donovani and L. infantum visceral leishmaniasis.

Parasitol Res 2016 Oct 13;115(10):4061-70. Epub 2016 Jul 13.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Room S7.24, Campus Drie Eiken, Universiteitsplein 1, B-2610, Wilrijk, Belgium.

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http://dx.doi.org/10.1007/s00436-016-5179-yDOI Listing
October 2016

In vitro CYP1A activity in the zebrafish: temporal but low metabolite levels during organogenesis and lack of gender differences in the adult stage.

Reprod Toxicol 2016 09 1;64:50-6. Epub 2016 Apr 1.

Applied Veterinary Morphology, Department of Veterinary Sciences, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp, Universiteitsplein 1, B-2610 Wilrijk, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.reprotox.2016.03.049DOI Listing
September 2016

Targeting an Aromatic Hotspot in Plasmodium falciparum 1-Deoxy-d-xylulose-5-phosphate Reductoisomerase with β-Arylpropyl Analogues of Fosmidomycin.

ChemMedChem 2016 09 3;11(18):2024-36. Epub 2016 Aug 3.

Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Biomedical Center, Box 596, 751 24, Uppsala, Sweden.

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http://dx.doi.org/10.1002/cmdc.201600249DOI Listing
September 2016

Antiprotozoal and Antiglycation Activities of Sesquiterpene Coumarins from Ferula narthex Exudate.

Molecules 2016 Sep 26;21(10). Epub 2016 Sep 26.

Natural Products & Food Research and Analysis (NatuRA), Department of Pharmaceutical Sciences, University of Antwerp, Universiteitsplein 1, 2610 Antwerp, Belgium.

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http://dx.doi.org/10.3390/molecules21101287DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6274357PMC
September 2016

Characterizing the in vitro biofilm phenotype of Staphylococcus epidermidis isolates from central venous catheters.

J Microbiol Methods 2016 08 16;127:95-101. Epub 2016 May 16.

Laboratory of Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, 2610 Wilrijk, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.mimet.2016.05.009DOI Listing
August 2016

antileishmanial and antimalarial activity of selected plants of Nepal.

J Intercult Ethnopharmacol 2016 Sep-Dec;5(4):383-389. Epub 2016 Aug 14.

Department of Biomedical Sciences, Laboratory for Microbiology, Parasitology and Hygiene, University of Antwerp, Belgium.

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http://dx.doi.org/10.5455/jice.20160728031236DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5061481PMC
August 2016

The role of the globin-coupled sensor YddV in a mature E. coli biofilm population.

Biochim Biophys Acta 2016 Jul 12;1864(7):835-9. Epub 2016 Apr 12.

Protein Chemistry, Proteomics and Epigenetic Signalling (PPES), Department of Biomedical Sciences, University of Antwerp, Antwerp, Belgium. Electronic address:

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http://dx.doi.org/10.1016/j.bbapap.2016.04.005DOI Listing
July 2016

Pharmacokinetics and pharmacodynamics of oleylphosphocholine in a hamster model of visceral leishmaniasis.

J Antimicrob Chemother 2016 07 15;71(7):1892-8. Epub 2016 Apr 15.

Laboratory for Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, Universiteitsplein 1, Wilrijk-Antwerp, Belgium.

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http://dx.doi.org/10.1093/jac/dkw089DOI Listing
July 2016

Cyclopeptide Alkaloids from Hymenocardia acida.

J Nat Prod 2016 07 28;79(7):1746-51. Epub 2016 Jun 28.

Research and Valorization Center on Medicinal Plants , Dubréka, Guinea-Conakry.

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http://dx.doi.org/10.1021/acs.jnatprod.6b00131DOI Listing
July 2016

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond.

Authors:
Wesley C Van Voorhis John H Adams Roberto Adelfio Vida Ahyong Myles H Akabas Pietro Alano Aintzane Alday Yesmalie Alemán Resto Aishah Alsibaee Ainhoa Alzualde Katherine T Andrews Simon V Avery Vicky M Avery Lawrence Ayong Mark Baker Stephen Baker Choukri Ben Mamoun Sangeeta Bhatia Quentin Bickle Lotfi Bounaadja Tana Bowling Jürgen Bosch Lauren E Boucher Fabrice F Boyom Jose Brea Marian Brennan Audrey Burton Conor R Caffrey Grazia Camarda Manuela Carrasquilla Dee Carter Maria Belen Cassera Ken Chih-Chien Cheng Worathad Chindaudomsate Anthony Chubb Beatrice L Colon Daisy D Colón-López Yolanda Corbett Gregory J Crowther Noemi Cowan Sarah D'Alessandro Na Le Dang Michael Delves Joseph L DeRisi Alan Y Du Sandra Duffy Shimaa Abd El-Salam El-Sayed Michael T Ferdig José A Fernández Robledo David A Fidock Isabelle Florent Patrick V T Fokou Ani Galstian Francisco Javier Gamo Suzanne Gokool Ben Gold Todd Golub Gregory M Goldgof Rajarshi Guha W Armand Guiguemde Nil Gural R Kiplin Guy Michael A E Hansen Kirsten K Hanson Andrew Hemphill Rob Hooft van Huijsduijnen Takaaki Horii Paul Horrocks Tyler B Hughes Christopher Huston Ikuo Igarashi Katrin Ingram-Sieber Maurice A Itoe Ajit Jadhav Amornrat Naranuntarat Jensen Laran T Jensen Rays H Y Jiang Annette Kaiser Jennifer Keiser Thomas Ketas Sebastien Kicka Sunyoung Kim Kiaran Kirk Vidya P Kumar Dennis E Kyle Maria Jose Lafuente Scott Landfear Nathan Lee Sukjun Lee Adele M Lehane Fengwu Li David Little Liqiong Liu Manuel Llinás Maria I Loza Aristea Lubar Leonardo Lucantoni Isabelle Lucet Louis Maes Dalu Mancama Nuha R Mansour Sandra March Sheena McGowan Iset Medina Vera Stephan Meister Luke Mercer Jordi Mestres Alvine N Mfopa Raj N Misra Seunghyun Moon John P Moore Francielly Morais Rodrigues da Costa Joachim Müller Arantza Muriana Stephen Nakazawa Hewitt Bakela Nare Carl Nathan Nathalie Narraidoo Sujeevi Nawaratna Kayode K Ojo Diana Ortiz Gordana Panic George Papadatos Silvia Parapini Kailash Patra Ngoc Pham Sarah Prats David M Plouffe Sally-Ann Poulsen Anupam Pradhan Celia Quevedo Ronald J Quinn Christopher A Rice Mohamed Abdo Rizk Andrea Ruecker Robert St Onge Rafaela Salgado Ferreira Jasmeet Samra Natalie G Robinett Ulrich Schlecht Marjorie Schmitt Filipe Silva Villela Francesco Silvestrini Robert Sinden Dennis A Smith Thierry Soldati Andreas Spitzmüller Serge Maximilian Stamm David J Sullivan William Sullivan Sundari Suresh Brian M Suzuki Yo Suzuki S Joshua Swamidass Donatella Taramelli Lauve R Y Tchokouaha Anjo Theron David Thomas Kathryn F Tonissen Simon Townson Abhai K Tripathi Valentin Trofimov Kenneth O Udenze Imran Ullah Cindy Vallieres Edgar Vigil Joseph M Vinetz Phat Voong Vinh Hoan Vu Nao-Aki Watanabe Kate Weatherby Pamela M White Andrew F Wilks Elizabeth A Winzeler Edward Wojcik Melanie Wree Wesley Wu Naoaki Yokoyama Paul H A Zollo Nada Abla Benjamin Blasco Jeremy Burrows Benoît Laleu Didier Leroy Thomas Spangenberg Timothy Wells Paul A Willis

PLoS Pathog 2016 07 28;12(7):e1005763. Epub 2016 Jul 28.

Medicines for Malaria Venture, Geneva, Switzerland.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4965013PMC
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