Kentaro Umei

Kentaro Umei

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Kentaro Umei

Kentaro Umei

Publications by authors named "Kentaro Umei"

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4Publications

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Discovery of novel pyrazolo[1,5-a]pyridine-based EP receptor antagonists by scaffold hopping: Design, synthesis, and structure-activity relationships.

Bioorg Med Chem Lett 2017 09 25;27(17):4044-4050. Epub 2017 Jul 25.

Watarase Research Center, Discovery Research Headquarters, Kyorin Pharmaceutical Co., Ltd., 1848, Nogi, Nogi-machi, Shimotsuga-gun, Tochigi 329-0114, Japan. Electronic address:

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September 2017

Identification of novel 1,2,3,6-tetrahydropyridyl-substituted benzo[d]thiazoles: Lead generation and optimization toward potent and orally active EP receptor antagonists.

Bioorg Med Chem 2017 07 26;25(13):3406-3430. Epub 2017 Apr 26.

Watarase Research Center, Discovery Research Headquarters, Kyorin Pharmaceutical Co., Ltd., 1848, Nogi, Nogi-machi, Shimotsuga-gun, Tochigi 329-0114, Japan. Electronic address:

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July 2017

Novel pyrazolo[1,5-a]pyridines as orally active EP receptor antagonists: Synthesis, structure-activity relationship studies, and biological evaluation.

Bioorg Med Chem 2017 05 14;25(9):2635-2642. Epub 2017 Mar 14.

Watarase Research Center, Discovery Research Headquarters, Kyorin Pharmaceutical Co., Ltd., 1848, Nogi, Nogi-machi, Shimotsuga-gun, Tochigi 329-0114, Japan. Electronic address:

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May 2017

Synthesis of Paclitaxel. 1. Synthesis of the ABC Ring of Paclitaxel by SmI2-Mediated Cyclization.

Org Lett 2015 Jun 26;17(11):2570-3. Epub 2015 May 26.

†Department Applied Chemistry, Faculty of Science and Technology, Keio University, 3-14-1 Hiyoshi, Kohoku-ku, Yokohama 223-8522, Japan.

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June 2015