John A Katzenellenbogen

John A Katzenellenbogen

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John A Katzenellenbogen

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Estrogens and selective estrogen receptor modulators differentially antagonize Runx2 in ST2 mesenchymal progenitor cells.

J Steroid Biochem Mol Biol 2018 10 8;183:10-17. Epub 2018 May 8.

Center of Craniofacial Molecular Biology, Ostrow School of Dentistry, University of Southern California, Los Angeles, CA, USA; Departments of Biochemistry and Molecular Medicine, Los Angeles, CA, USA; Institute for Genetic Medicine, Keck School of Medicine of the University of Southern California, Los Angeles, CA, USA; Departments of Orthopedic Surgery, Los Angeles, CA, USA. Electronic address:

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http://dx.doi.org/10.1016/j.jsbmb.2018.05.002DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6128776PMC
October 2018

Triaryl Pyrazole Toll-Like Receptor Signaling Inhibitors: Structure-Activity Relationships Governing Pan- and Selective Signaling Inhibitors.

ChemMedChem 2018 10 13;13(20):2208-2216. Epub 2018 Sep 13.

Department of Chemistry, University of Illinois, 505 South Mathews Avenue, Urbana, IL, 61801, USA.

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http://dx.doi.org/10.1002/cmdc.201800417DOI Listing
October 2018

Publisher Correction: Structural underpinnings of oestrogen receptor mutations in endocrine therapy resistance.

Nat Rev Cancer 2018 Oct;18(10):662

Human Oncology and Pathogenesis Program, Memorial Sloan Kettering Cancer Center, New York, NY, USA.

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http://dx.doi.org/10.1038/s41568-018-0053-0DOI Listing
October 2018

Identification of Toll-like receptor signaling inhibitors based on selective activation of hierarchically acting signaling proteins.

Sci Signal 2018 08 14;11(543). Epub 2018 Aug 14.

Department of Infectious Diseases, St. Jude Children's Research Hospital, 262 Danny Thomas Place, Memphis, TN 38105, USA.

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http://dx.doi.org/10.1126/scisignal.aaq1077DOI Listing
August 2018

New Class of Selective Estrogen Receptor Degraders (SERDs): Expanding the Toolbox of PROTAC Degrons.

ACS Med Chem Lett 2018 Aug 5;9(8):803-808. Epub 2018 Jul 5.

Department of Chemistry and Chemical Biology, Stevens Institute of Technology, Hoboken, New Jersey 07601 United States.

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http://dx.doi.org/10.1021/acsmedchemlett.8b00106DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6088359PMC
August 2018

Increase in chemokine CXCL1 by ERβ ligand treatment is a key mediator in promoting axon myelination.

Proc Natl Acad Sci U S A 2018 06 29;115(24):6291-6296. Epub 2018 May 29.

Division of Biomedical Sciences, University of California, Riverside School of Medicine, Riverside, CA 92521;

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http://dx.doi.org/10.1073/pnas.1721732115DOI Listing
June 2018

Copper-Mediated Nucleophilic Radiobromination of Aryl Boron Precursors: Convenient Preparation of a Radiobrominated PARP-1 Inhibitor.

Tetrahedron Lett 2018 May 11;59(20):1963-1967. Epub 2018 Apr 11.

Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, IL 61801.

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http://dx.doi.org/10.1016/j.tetlet.2018.04.024DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6195330PMC
May 2018

Estrogens and androgens inhibit association of RANKL with the pre-osteoblast membrane through post-translational mechanisms.

J Cell Physiol 2017 Dec 11;232(12):3798-3807. Epub 2017 May 11.

Department of Biochemistry and Molecular Medicine , Keck School of Medicine, University of Southern California, Los Angeles, California.

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http://dx.doi.org/10.1002/jcp.25862DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5562539PMC
December 2017

Evaluation of aromatic radiobromination by nucleophilic substitution using diaryliodonium salt precursors.

J Labelled Comp Radiopharm 2017 07 14;60(9):450-456. Epub 2017 Jun 14.

Department of Chemistry, University of Illinois at Urbana-Champaign, Champaign, IL, USA.

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http://dx.doi.org/10.1002/jlcr.3519DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5550022PMC
July 2017

Selenophenes: Introducing a New Element into the Core of Non-Steroidal Estrogen Receptor Ligands.

ChemMedChem 2017 02 9;12(3):235-249. Epub 2017 Jan 9.

State Key Laboratory of Virology, Key Laboratory of Combinatorial Biosynthesis and Drug Discovery, Wuhan University, Ministry of Education, Wuhan University School of Pharmaceutical Sciences, 185 East Lake Road, Wuhan, 430071, P.R. China.

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http://dx.doi.org/10.1002/cmdc.201600593DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5405701PMC
February 2017

Exploring the Structural Compliancy versus Specificity of the Estrogen Receptor Using Isomeric Three-Dimensional Ligands.

ACS Chem Biol 2017 02 29;12(2):494-503. Epub 2016 Dec 29.

Department of Chemistry, University of Illinois at Urbana-Champaign , 600 South Mathews Avenue, Urbana, Illinois 61801, United States.

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http://dx.doi.org/10.1021/acschembio.6b00918DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5315646PMC
February 2017

Estrogen receptor-α and aryl hydrocarbon receptor involvement in the actions of botanical estrogens in target cells.

Mol Cell Endocrinol 2016 12 16;437:190-200. Epub 2016 Aug 16.

Department of Molecular and Integrative Physiology, University of Illinois at Urbana-Champaign, Urbana, IL 61801, USA. Electronic address:

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http://dx.doi.org/10.1016/j.mce.2016.08.025DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5873581PMC
December 2016

Nonnuclear Estrogen Receptor Activation Improves Hepatic Steatosis in Female Mice.

Endocrinology 2016 Oct 23;157(10):3731-3741. Epub 2016 Aug 23.

Center for Pulmonary and Vascular Biology (K.L.C., J.B., M.U., J.U., L.H., C.M., P.W.S.), Department of Pediatrics, University of Texas Southwestern Medical Center, Dallas, Texas, 75390; and Departments of Chemistry (S.H.K., J.A.K.), Food Science and Human Nutrition (Z.M.-E.), and Molecular and Integrative Physiology (B.S.K.), University of Illinois at Urbana-Champaign, Urbana, Illinois, 61801.

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http://dx.doi.org/10.1210/en.2015-1629DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5045504PMC
October 2016

Extranuclear Actions of the Androgen Receptor Enhance Glucose-Stimulated Insulin Secretion in the Male.

Cell Metab 2016 May 28;23(5):837-51. Epub 2016 Apr 28.

Diabetes Discovery Research and Gender Medicine Laboratory, Department of Medicine, Section of Endocrinology and Metabolism, Tulane University Health Sciences Center, New Orleans, LA 70112, USA; Department of Medicine, Division of Endocrinology, Metabolism and Molecular Medicine, Northwestern University, Feinberg School of Medicine, Chicago, IL 60611, USA. Electronic address:

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http://www.cell.com/cell-metabolism/pdf/S1550-4131(16)30118-
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http://linkinghub.elsevier.com/retrieve/pii/S155041311630118
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http://dx.doi.org/10.1016/j.cmet.2016.03.015DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4864089PMC
May 2016

Science Signaling podcast for 24 May 2016: Designer estrogens.

Sci Signal 2016 May 24;9(429):pc12. Epub 2016 May 24.

Web Editor, Science Signaling, American Association for the Advancement of Science, 1200 New York Avenue, NW, Washington, DC 20005, USA.

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http://dx.doi.org/10.1126/scisignal.aag1040DOI Listing
May 2016

Multiple Beneficial Roles of Repressor of Estrogen Receptor Activity (REA) in Suppressing the Progression of Endometriosis.

Endocrinology 2016 Feb 14;157(2):900-12. Epub 2015 Dec 14.

Departments of Molecular and Integrative Physiology (Y.Z., Y.C., M.K.B., B.S.K.) and Chemistry (J.A.K.), University of Illinois at Urbana-Champaign, Urbana, Illinois 61801; Department of Gynecology and Obstetrics (Y.K.), The Second Affiliated Hospital of Harbin Medical University, Harbin, Heilongjiang 150086, China; and Department of Obstetrics and Gynecology (R.N.T.), Wake Forest School of Medicine, Winston-Salem, North Carolina 27157.

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http://dx.doi.org/10.1210/en.2015-1324DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4733120PMC
February 2016

Imaging Diagnostic and Therapeutic Targets: Steroid Receptors in Breast Cancer.

J Nucl Med 2016 Feb;57 Suppl 1:75S-80S

Division of Nuclear Medicine, Mallinckrodt Institute of Radiology, Washington University, St. Louis, Missouri.

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http://dx.doi.org/10.2967/jnumed.115.157933DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4795822PMC
February 2016

Estrogen Receptor-Selective Agonists Modulate Learning in Female Rats in a Dose- and Task-Specific Manner.

Endocrinology 2016 Jan 14;157(1):292-303. Epub 2015 Oct 14.

Neuroscience Program (S.L.P., S.L.N., S.L.S., D.L.K.) and Department of Chemistry (J.A.K.), University of Illinois at Urbana-Champaign, Urbana, Illinois 61801; Department of Comparative Biosciences (S.L.N., S.L.S.), University of Illinois at Urbana-Champaign, Urbana, Illinois 61802; Department of Psychology and Neuroscience (S.L.N.), Baldwin Wallace University, Berea, Ohio 44017; and Department of Biology (D.L.K.), Syracuse University, Syracuse, New York 13244.

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http://dx.doi.org/10.1210/en.2015-1616DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4701887PMC
January 2016

Estrogen receptor alpha/co-activator interaction assay: TR-FRET.

Methods Mol Biol 2015 ;1278:545-53

Department of Chemistry, University of Illinois at Urbana-Champaign, 600 S. Mathews Avenue, Urbana, IL, 61801, USA.

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http://dx.doi.org/10.1007/978-1-4939-2425-7_36DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4893311PMC
December 2015

Protective Hematopoietic Effect of Estrogens in a Mouse Model of Thrombosis: Respective Roles of Nuclear Versus Membrane Estrogen Receptor α.

Endocrinology 2015 Nov 17;156(11):4293-301. Epub 2015 Aug 17.

INSERM U1048 and Université Toulouse III I2MC (M.-C.V., C.F., F.L., C.C., M.G., N.S., B.P., J.-F.A.), Toulouse, 31432 France; Faculté de Chirurgie Dentaire (M.-C.V.), Université de Toulouse III, Toulouse, 31432 France; Department of Chemistry (H.H.K., J.A.K.), University of Illinois at Urbana-Champaign, Urbana, IL 61801; Institut de Génétique et de Biologie Moléculaire et Cellulaire (P.C.), Collège de France, Université de Strasbourg, Illkirch, 67400 France; Department of Physiology and Cell Biology (B.S.K.), University of Illinois at Urbana-Champaign, Urbana, IL 61801; and Laboratoire d'Hématologie (B.P.), Centre Hospitalier Universitaire de Toulouse, Toulouse, 31432 France.

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https://academic.oup.com/endo/article-lookup/doi/10.1210/en.
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http://dx.doi.org/10.1210/en.2015-1522DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4606746PMC
November 2015

Fluorescent Nanoconjugate Derivatives with Enhanced Photostability for Single Molecule Imaging.

Anal Chem 2015 Nov 20;87(21):11048-57. Epub 2015 Oct 20.

Department of Chemical and Biomolecular Engineering, University of Illinois at Urbana-Champaign , Urbana, Illinois 61801, United States.

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http://pubs.acs.org/doi/10.1021/acs.analchem.5b03059
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http://dx.doi.org/10.1021/acs.analchem.5b03059DOI Listing
November 2015

Preparation of o-Fluorophenols from Nonaromatic Precursors: Mechanistic Considerations for Adaptation to Fluorine-18 Radiolabeling.

Org Lett 2015 Nov 4;17(22):5540-3. Epub 2015 Nov 4.

Department of Chemistry, University of Illinois at Urbana-Champaign , 600 South Mathews Avenue, Urbana, Illinois 61801, United States.

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http://pubs.acs.org/doi/10.1021/acs.orglett.5b02640
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http://dx.doi.org/10.1021/acs.orglett.5b02640DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4795842PMC
November 2015

The Activation Function-1 of Estrogen Receptor Alpha Prevents Arterial Neointima Development Through a Direct Effect on Smooth Muscle Cells.

Circ Res 2015 Oct 27;117(9):770-8. Epub 2015 Aug 27.

From the Department of Vascular Biology of the Institute of Metabolic and Cardiovascular Diseases (I2MC), Université de Toulouse 3, Institut National de la Santé et de la Recherche Médicale (INSERM) UMR1048, Institut des Maladies Métaboliques et Cardiovasculaires, Toulouse, France (N.F.S., C.F., M.B., A.L., A.V., M.-C.V., M.G., N.M., F.L., P.G., M.L., J.-F.A.); Laboratory of Tumor and Developmental Biology, GIGA-Cancer, Université de Liège, Groupe Interdisciplinaire de Génoprotéomique Appliquée, Liège, Belgique (J.-M.F.); UMR INRA/DGER 1225, Université de Toulouse, INP, ENVT, Toulouse, France (I.R.-L.); Departments of Molecular and Integrative Biology (B.S.K.) and Chemistry, University of Illinois at Urbana-Champaign (J.A.K.).

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http://dx.doi.org/10.1161/CIRCRESAHA.115.306416DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4596486PMC
October 2015

Imidoyl dichlorides as new reagents for the rapid formation of 2-aminobenzimidazoles and related azoles.

Tetrahedron Lett 2015 Oct;56(44):6097-6099

Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, Illinois 61801, United States.

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http://dx.doi.org/10.1016/j.tetlet.2015.09.076DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4620578PMC
October 2015

Neural-Network Scoring Functions Identify Structurally Novel Estrogen-Receptor Ligands.

J Chem Inf Model 2015 Sep 4;55(9):1953-61. Epub 2015 Sep 4.

Department of Chemistry & Biochemistry and the National Biomedical Computation Resource, University of California, San Diego , La Jolla, California 92093, United States.

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http://dx.doi.org/10.1021/acs.jcim.5b00241DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4780411PMC
September 2015

PI3K inhibition results in enhanced estrogen receptor function and dependence in hormone receptor-positive breast cancer.

Sci Transl Med 2015 Apr;7(283):283ra51

Human Oncology and Pathogenesis Program and Memorial Sloan Kettering Cancer Center, 1275 York Avenue, Box 20, New York, NY 10065, USA. Breast Medicine Service, Department of Medicine, Memorial Sloan Kettering Cancer Center, New York, NY 10065, USA. Weill Cornell Medical College, New York, NY 10065, USA.

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http://dx.doi.org/10.1126/scitranslmed.aaa4442DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4433148PMC
April 2015

Facile purification and click labeling with 2-[F]fluoroethyl azide using solid phase extraction cartridges.

Tetrahedron Lett 2015 Feb 4;56(7):952-954. Epub 2014 Nov 4.

Department of Chemistry, University of Illinois, Urbana, IL 61801, USA.

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http://dx.doi.org/10.1016/j.tetlet.2014.10.126DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4792033PMC
February 2015

Multiple functional therapeutic effects of the estrogen receptor β agonist indazole-Cl in a mouse model of multiple sclerosis.

Proc Natl Acad Sci U S A 2014 Dec 1;111(50):18061-6. Epub 2014 Dec 1.

Department of Neurology, Division of Biomedical Sciences at the School of Medicine, University of California, Riverside, CA 92521; Intellectual and Developmental Disabilities Research Center, Semel Institute for Neuroscience at the School of Medicine, University of California, Los Angeles, CA 90095; and Brain Research Institute, and

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http://dx.doi.org/10.1073/pnas.1411294111DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4273334PMC
December 2014

Estrogen receptors alpha (ERα) and beta (ERβ): subtype-selective ligands and clinical potential.

Steroids 2014 Nov 24;90:13-29. Epub 2014 Jun 24.

Dipartimento di Farmacia, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy. Electronic address:

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http://dx.doi.org/10.1016/j.steroids.2014.06.012DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4192010PMC
November 2014

Utilizing electrostatic interactions to facilitate F-18 radiolabeling of poly(amido)amine (PAMAM) dendrimers.

Org Biomol Chem 2014 Nov;12(43):8696-701

Washington University Medical School, Mallinckrodt Institute of Radiology, Saint Louis, MO 63110, USA.

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http://dx.doi.org/10.1039/c4ob01616eDOI Listing
November 2014

Synthesis and receptor binding in trans-CD ring-fused A-CD estrogens: comparison with the cis-fused isomers.

Bioorg Med Chem Lett 2014 Aug 27;24(16):3841-4. Epub 2014 Jun 27.

Department of Chemistry, University of Ottawa, D'Iorio Hall, 10 Marie Curie St., Ottawa K1N 6N5, Canada. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2014.06.066DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4249688PMC
August 2014

Cyclin D1 integrates estrogen-mediated DNA damage repair signaling.

Cancer Res 2014 Jul 15;74(14):3959-70. Epub 2014 May 15.

Authors' Affiliations: Departments of Cancer Biology and Kimmel Cancer Center, Thomas Jefferson University, Philadelphia, Pennsylvania; and

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http://dx.doi.org/10.1158/0008-5472.CAN-13-3137DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4102655PMC
July 2014

π-π interaction energies as determinants of the photodimerization of mono-, di-, and triazastilbenes.

J Org Chem 2014 Jun 28;79(12):5448-62. Epub 2014 May 28.

Department of Chemistry University of Illinois at Urbana-Champaign Urbana, Illinois 61801, United States.

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http://dx.doi.org/10.1021/jo500457nDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4076016PMC
June 2014

Triaryl-substituted Schiff bases are high-affinity subtype-selective ligands for the estrogen receptor.

J Med Chem 2014 Apr 7;57(8):3532-45. Epub 2014 Apr 7.

Key Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, State Key Laboratory of Virology, Wuhan University School of Pharmaceutical Sciences , Wuhan 430071, China.

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http://dx.doi.org/10.1021/jm500268jDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4002130PMC
April 2014

Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens.

FASEB J 2013 Nov 23;27(11):4406-18. Epub 2013 Jul 23.

1Department of Molecular and Integrative Physiology, University of Illinois and College of Medicine at Urbana-Champaign, Urbana, IL 61801, USA.

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http://dx.doi.org/10.1096/fj.13-234617DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3804744PMC
November 2013

Selective Delivery of an Anticancer Drug with Aptamer-Functionalized Liposomes to Breast Cancer Cells and

J Mater Chem B 2013 Oct;1(39):5288-5297

Department of Chemistry, University of Illinois at Urbana-Champaign, Urbana, Illinois 61801, USA. Tel: +1-217-333-2619 ; Beckman Institute for Advanced Science and Technology, University of Illinois at Urbana-Champaign, Urbana, Illinois 61801, USA. Tel: +1-217-244-5023.

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http://xlink.rsc.org/?DOI=c3tb20412j
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http://dx.doi.org/10.1039/C3TB20412JDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3800741PMC
October 2013

Experimental versus predicted affinities for ligand binding to estrogen receptor: iterative selection and rescoring of docked poses systematically improves the correlation.

J Comput Aided Mol Des 2013 Aug 24;27(8):707-21. Epub 2013 Aug 24.

Department of Chemistry, Carleton University, 1125 Colonel By Dr., Ottawa, K1S 5B6, Canada,

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http://link.springer.com/10.1007/s10822-013-9670-6
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http://dx.doi.org/10.1007/s10822-013-9670-6DOI Listing
August 2013

c-Src modulates estrogen-induced stress and apoptosis in estrogen-deprived breast cancer cells.

Cancer Res 2013 Jul 23;73(14):4510-20. Epub 2013 May 23.

Department of Oncology, Lombardi Comprehensive Cancer Center, Georgetown University, Washington, DC 20057, USA.

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http://dx.doi.org/10.1158/0008-5472.CAN-12-4152DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3715569PMC
July 2013

Integrative genomics of gene and metabolic regulation by estrogen receptors α and β, and their coregulators.

Mol Syst Biol 2013 Jun 18;9:676. Epub 2013 Jun 18.

Department of Molecular and Integrative Physiology, and Cell and Developmental Biology, University of Illinois at Urbana-Champaign, Urbana, IL 61801, USA.

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http://dx.doi.org/10.1038/msb.2013.28DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3964312PMC
June 2013

Nonsteroidal bivalent estrogen ligands: an application of the bivalent concept to the estrogen receptor.

ACS Chem Biol 2013 Apr 30;8(4):707-15. Epub 2013 Jan 30.

Institut für Chemie und Biochemie, Freie Universität Berlin, Takustrasse 3, 14195 Berlin, Germany.

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http://pubs.acs.org/doi/10.1021/cb3006243
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http://dx.doi.org/10.1021/cb3006243DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3631453PMC
April 2013

Non-nuclear-initiated actions of the estrogen receptor protect cortical bone mass.

Mol Endocrinol 2013 Apr 26;27(4):649-56. Epub 2013 Feb 26.

Division of Endocrinology and Metabolism, University of Arkansas for Medical Sciences, 4301 West Markham Street, MS 587, Little Rock, Arkansas 72205, USA.

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https://academic.oup.com/mend/article-lookup/doi/10.1210/me.
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http://dx.doi.org/10.1210/me.2012-1368DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3607700PMC
April 2013

Dendrimer probes for enhanced photostability and localization in fluorescence imaging.

Biophys J 2013 Apr;104(7):1566-75

Department of Chemical and Biomolecular Engineering, University of Illinois at Urbana-Champaign, Urbana, Illinois, USA.

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http://dx.doi.org/10.1016/j.bpj.2013.01.052DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3617423PMC
April 2013

Designer antiandrogens join the race against drug resistance.

Elife 2013 Apr 9;2:e00692. Epub 2013 Apr 9.

is at the Department of Chemistry , University of Illinois at Urbana-Champaign , Urbana , United States

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http://dx.doi.org/10.7554/eLife.00692DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3622176PMC
April 2013

Thiophene-core estrogen receptor ligands having superagonist activity.

J Med Chem 2013 Apr 15;56(8):3346-66. Epub 2013 Apr 15.

Key Laboratory of Combinatorial Biosynthesis and Drug Discovery (Wuhan University), Ministry of Education, State Key Laboratory of Virology, Wuhan University School of Pharmaceutical Sciences, Wuhan 430072, China.

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http://link.springer.com/content/pdf/10.1186%2Fs13071-016-16
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http://pubs.acs.org/doi/abs/10.1021/jm400157e
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http://dx.doi.org/10.1021/jm400157eDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3666579PMC
April 2013

Pharmacokinetics of the estrogen receptor subtype-selective ligands, PPT and DPN: quantification using UPLC-ES/MS/MS.

J Pharm Biomed Anal 2012 Dec 24;71:119-26. Epub 2012 Aug 24.

National Center for Toxicological Research, U.S. Food and Drug Administration, Jefferson, AR 72079, USA.

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http://dx.doi.org/10.1016/j.jpba.2012.08.022DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3509942PMC
December 2012

Specific labeling of zinc finger proteins using noncanonical amino acids and copper-free click chemistry.

Bioconjug Chem 2012 Sep 30;23(9):1891-901. Epub 2012 Aug 30.

Department of Chemical and Biomolecular Engineering, University of Illinois at Urbana-Champaign, Urbana, Illinois 61801, USA.

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http://dx.doi.org/10.1021/bc300262hDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3462365PMC
September 2012

BC-spiro-estradiols. Synthesis and estrogen receptor binding affinity of four new estradiol isomers.

Bioorg Med Chem Lett 2012 Jun 11;22(11):3713-7. Epub 2012 Apr 11.

Department of Chemistry, University of Ottawa, Ottawa, Canada.

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http://dx.doi.org/10.1016/j.bmcl.2012.04.022DOI Listing
June 2012

64Cu Core-labeled nanoparticles with high specific activity via metal-free click chemistry.

ACS Nano 2012 Jun 8;6(6):5209-19. Epub 2012 May 8.

Mallinckrodt Institute of Radiology, Washington University School of Medicine, St. Louis, Missouri 63110, USA.

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http://dx.doi.org/10.1021/nn300974sDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3383893PMC
June 2012