Jingrong Cui

Jingrong Cui

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Jingrong Cui

Publications by authors named "Jingrong Cui"

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Synthesis and biological evaluation of curcumin derivatives modified with α-amino boronic acid as proteasome inhibitors.

Bioorg Med Chem Lett 2018 08 2;28(14):2459-2464. Epub 2018 Jun 2.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, PR China. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X183048
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http://dx.doi.org/10.1016/j.bmcl.2018.06.004DOI Listing
August 2018

Cytotoxic oleanane triterpenoid saponins from Albizia julibrissin.

Fitoterapia 2017 Sep 29;121:183-193. Epub 2017 Jul 29.

State Key Laboratory of Natural and Biomimetic Drugs, Department of Natural Medicines, School of Pharmaceutical Sciences, Peking University Health Science Center, Beijing 100191, People's Republic of China. Electronic address:

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http://dx.doi.org/10.1016/j.fitote.2017.07.015DOI Listing
September 2017

Synthesis and biological activity of peptide proline-boronic acids as proteasome inhibitors.

Bioorg Med Chem 2017 08 9;25(15):4031-4044. Epub 2017 Jun 9.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, PR China. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2017.05.049DOI Listing
August 2017

Proteasome Inhibitor YSY01A Abrogates Constitutive STAT3 Signaling via Down-regulation of Gp130 and JAK2 in Human A549 Lung Cancer Cells.

Front Pharmacol 2017 24;8:476. Epub 2017 Aug 24.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking UniversityBeijing, China.

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http://dx.doi.org/10.3389/fphar.2017.00476DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5574410PMC
August 2017

Diasteltoxins A-C, Asteltoxin-Based Dimers from a Mutant of the Sponge-Associated Emericella variecolor Fungus.

Org Lett 2016 09 29;18(18):4678-81. Epub 2016 Aug 29.

State Key Laboratory of Natural and Biomimetic Drugs, Peking University , Beijing 100191, P. R. China.

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http://dx.doi.org/10.1021/acs.orglett.6b02313DOI Listing
September 2016

YSY01A, a Novel Proteasome Inhibitor, Induces Cell Cycle Arrest on G2 Phase in MCF-7 Cells via ERα and PI3K/Akt Pathways.

J Cancer 2015 6;6(4):319-26. Epub 2015 Feb 6.

1. State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, 100083, Beijing, China;

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http://dx.doi.org/10.7150/jca.10733DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4349871PMC
March 2015

Evaluation of the effect of TM208 on the activity of five cytochrome P450 enzymes using on-line solid-phase extraction HPLC-DAD: a cocktail approach.

J Chromatogr B Analyt Technol Biomed Life Sci 2013 Apr 10;923-924:29-36. Epub 2013 Feb 10.

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Beijing, China.

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https://linkinghub.elsevier.com/retrieve/pii/S15700232130008
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http://dx.doi.org/10.1016/j.jchromb.2013.01.031DOI Listing
April 2013

A specific peptide ligand-modified lipid nanoparticle carrier for the inhibition of tumor metastasis growth.

Biomaterials 2013 Jan 30;34(3):756-64. Epub 2012 Oct 30.

State Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing, China; Department of Pharmaceutics, Peking University, Beijing, China.

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http://dx.doi.org/10.1016/j.biomaterials.2012.10.018DOI Listing
January 2013

Furanodiene, a natural product, inhibits breast cancer growth both in vitro and in vivo.

Cell Physiol Biochem 2012 2;30(3):778-90. Epub 2012 Aug 2.

State Key Laboratory of Quality Research in Chinese Medicine, University of Macau, Macau, China.

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https://www.karger.com/Article/FullText/341457
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http://dx.doi.org/10.1159/000341457DOI Listing
December 2012

The use of a tumor metastasis targeting peptide to deliver doxorubicin-containing liposomes to highly metastatic cancer.

Biomaterials 2012 Nov 31;33(33):8451-60. Epub 2012 Aug 31.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, China.

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http://dx.doi.org/10.1016/j.biomaterials.2012.08.031DOI Listing
November 2012

Angiogenesis inhibition and cell cycle arrest induced by treatment with Pseudolarix acid B alone or combined with 5-fluorouracil.

Acta Biochim Biophys Sin (Shanghai) 2012 Jun 2;44(6):490-502. Epub 2012 May 2.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

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http://dx.doi.org/10.1093/abbs/gms029DOI Listing
June 2012

Determination of 4-methylpiperaine-1-carbodithioc acid 3-cyano-3,3-diphenylpropyl ester hydrochloride in rats' plasma by online-SPE-HPLC-DAD: application to a pharmacokinetic study.

J Sep Sci 2012 Mar;35(5-6):721-5

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Beijing, China.

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http://dx.doi.org/10.1002/jssc.201100876DOI Listing
March 2012

Effects of CS-1 on A431 cell proliferation, cell cycle, and epidermal growth factor receptor signal transduction.

Acta Biochim Biophys Sin (Shanghai) 2012 Feb 21;44(2):136-46. Epub 2011 Dec 21.

State Key Laboratory of Natural and Biomimetic Drugs, Peking University, Beijing, China.

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http://dx.doi.org/10.1093/abbs/gmr111DOI Listing
February 2012

Molecular design, synthesis and bioactivity of glycosyl hydrazine and hydrazone derivatives: notable effects of the sugar moiety.

Bioorg Med Chem Lett 2011 Dec 22;21(23):7193-6. Epub 2011 Sep 22.

Department of Applied Chemistry, College of Science, China Agricultural University, Beijing, People's Republic of China.

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X110131
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http://dx.doi.org/10.1016/j.bmcl.2011.09.068DOI Listing
December 2011

Synthesis and SAR study of novel peptide aldehydes as inhibitors of 20S proteasome.

Molecules 2011 Sep 5;16(9):7551-64. Epub 2011 Sep 5.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

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http://dx.doi.org/10.3390/molecules16097551DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6264673PMC
September 2011

Synthesis and structure-activity relationships of a novel class of dithiocarbamic acid esters as anticancer agent.

Arch Pharm (Weinheim) 2011 May 17;344(5):320-32. Epub 2011 Jan 17.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, PR China.

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http://dx.doi.org/10.1002/ardp.201000259DOI Listing
May 2011

New class of potent antitumor acylhydrazone derivatives containing furan.

Eur J Med Chem 2010 Dec 17;45(12):5576-84. Epub 2010 Sep 17.

Key Laboratory of Pesticide Chemistry and Application, Ministry of Agriculture, Department of Applied Chemistry, College of Science, China Agricultural University, Beijing 100193, People's Republic of China.

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http://dx.doi.org/10.1016/j.ejmech.2010.09.007DOI Listing
December 2010

Synthesis and bioactivity of N-benzoyl-N'-[5-(2'-substituted phenyl)-2-furoyl] semicarbazide derivatives.

Molecules 2010 Jun 11;15(6):4267-82. Epub 2010 Jun 11.

Key Laboratory of Pesticide Chemistry and Application, Ministry of Agriculture, Department of Applied Chemistry, College of Science, China Agricultural University, Beijing 100193, China.

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http://dx.doi.org/10.3390/molecules15064267DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6257640PMC
June 2010

Simultaneous determination of 4-methyl-piperazine-1-carbodithioc acid 3-cyano-3,3-diphenylpropyl ester hydrochloride and its major metabolite in rats by HPLC.

J Chromatogr Sci 2010 Feb;48(2):125-9

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Beijing 100083, China.

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http://dx.doi.org/10.1093/chromsci/48.2.125DOI Listing
February 2010

Synthesis, cytotoxicity and DNA-binding levels of new type binuclear platinum(II) complexes.

Eur J Med Chem 2009 Nov 21;44(11):4772-7. Epub 2009 Jun 21.

College of Chemistry and Environmental Science, Hebei University, Baoding 071002, China.

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http://dx.doi.org/10.1016/j.ejmech.2009.06.017DOI Listing
November 2009

Capillary electrophoresis for screening of 20S proteasome inhibitors.

Anal Biochem 2009 Nov 16;394(1):62-7. Epub 2009 Jul 16.

Department of Pharmaceutical Analysis, School of Pharmaceutical Science, Peking University, Beijing 100191, People's Republic of China.

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http://dx.doi.org/10.1016/j.ab.2009.07.020DOI Listing
November 2009

Design, synthesis and biological evaluation of tripeptide boronic acid proteasome inhibitors.

Bioorg Med Chem 2009 Oct 20;17(19):6851-61. Epub 2009 Aug 20.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, PR China.

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https://linkinghub.elsevier.com/retrieve/pii/S09680896090079
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http://dx.doi.org/10.1016/j.bmc.2009.08.023DOI Listing
October 2009

Synthesis of 3-N-sugar-substituted-2, 4(1H,3H)-quinazolinedionesas anti-angiogenesis agents.

Molecules 2009 Jul 8;14(7):2447-57. Epub 2009 Jul 8.

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

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http://dx.doi.org/10.3390/molecules14072447DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6254791PMC
July 2009

Synthesis, characterization and antitumor activity of new type binuclear platinum(II) complexes.

Eur J Med Chem 2009 May 27;44(5):2322-7. Epub 2008 Apr 27.

College of Chemistry and Environmental Science, Hebei University, Baoding 071002, China.

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http://dx.doi.org/10.1016/j.ejmech.2008.04.005DOI Listing
May 2009

Novel 8-deaza-5,6,7,8-tetrahydroaminopterin derivatives as dihydrofolate inhibitor: design, synthesis and antifolate activity.

Eur J Med Chem 2009 Feb 4;44(2):764-71. Epub 2008 May 4.

Department of Chemical Biology, School of Pharmaceutical Sciences, Peking University, Beijing 100083, China.

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http://dx.doi.org/10.1016/j.ejmech.2008.04.017DOI Listing
February 2009

Two newly synthesized 5-methyltetrahydrofolate-like compounds inhibit methionine synthase activity accompanied by cell cycle arrest in G1/S phase and apoptosis in vitro.

Anticancer Drugs 2008 Aug;19(7):697-704

State Key Laboratory of Natural and Biomimetic Drugs, Peking University Health Science Center, Beijing, PR China.

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http://dx.doi.org/10.1097/CAD.0b013e32830317f2DOI Listing
August 2008

Polynuclear diorganotin(IV) complexes with arylhydroxamates: Syntheses, structures and in vitro cytotoxic activities.

J Inorg Biochem 2008 Apr 23;102(4):901-9. Epub 2007 Dec 23.

School of Pharmaceutical Science, Shanxi Medical University, Taiyuan 030001, PR China.

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http://linkinghub.elsevier.com/retrieve/pii/S016201340700354
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http://dx.doi.org/10.1016/j.jinorgbio.2007.12.010DOI Listing
April 2008

Synthesis, cytotoxicity and DNA binding levels of tri-functional mononuclear platinum(II) complexes.

Eur J Med Chem 2008 Feb 18;43(2):441-7. Epub 2007 May 18.

College of Chemistry and Environmental Science, Hebei University, Baoding 071002, PR China.

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http://dx.doi.org/10.1016/j.ejmech.2007.04.015DOI Listing
February 2008

Anticancer activity and mechanisms of norcantharidin-Nd3II on hepatoma.

Anticancer Drugs 2007 Nov;18(10):1133-7

State Key Laboratory of Natural and Biomimetic Drugs, Peking University Health Science Center, Beijing, PRC.

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http://dx.doi.org/10.1097/CAD.0b013e3282eeb1c5DOI Listing
November 2007

Studies on the metabolism of 4-methyl-piperazine-1-carbodithioc acid 3-cyano-3,3-diphenylpropyl ester hydrochloride in rats by high-performance liquid chromatography/electrospray ionization tandem mass spectrometry.

J Pharm Biomed Anal 2007 Sep 25;44(5):1127-32. Epub 2007 May 25.

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Xueyuan Road 38, Beijing 100083, China.

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http://dx.doi.org/10.1016/j.jpba.2007.05.026DOI Listing
September 2007

Studies on the metabolism of 4-methylpiperazine-1-carbodithioc acid 3-cyano-3,3- diphenylpropyl ester hydrochloride in rat bile by high-performance liquid chromatography/electrospray ionization tandem mass spectrometry.

Rapid Commun Mass Spectrom 2007 ;21(10):1599-605

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Beijing 100083, China.

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http://dx.doi.org/10.1002/rcm.3001DOI Listing
August 2007

Analysis of 4-methyl-piperazine-1-carbodithioic acid 3-cyano-3,3-diphenyl-propyl ester hydrochloride and its major metabolites in rat plasma and tissues by LC-MS/MS.

J Sep Sci 2007 Aug;30(13):2080-5

Department of Pharmaceutical Analysis, School of Pharmaceutical Sciences, Peking University, Beijing, China.

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http://doi.wiley.com/10.1002/jssc.200700081
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http://dx.doi.org/10.1002/jssc.200700081DOI Listing
August 2007

Embelin derivatives and their anticancer activity through microtubule disassembly.

Planta Med 2005 Oct;71(10):944-8

State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Xueyuan Road 38, 100083 Beijing, P.R. China.

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http://dx.doi.org/10.1055/s-2005-871250DOI Listing
October 2005

Novel pyrrolyllactone and pyrrolyllactam indolinones as potent cyclin-dependent kinase 2 inhibitors.

Bioorg Med Chem Lett 2003 Jun;13(11):1939-42

SUGEN, Inc., 230 East Grand Ave., South San Francisco, CA 94080, USA.

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http://dx.doi.org/10.1016/s0960-894x(03)00312-3DOI Listing
June 2003