Jigar A Makawana

Jigar A Makawana

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Jigar A Makawana

Jigar A Makawana

Publications by authors named "Jigar A Makawana"

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17Publications

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Recent Developments of Metal and Metal Oxide Nanocatalysts in Organic Synthesis.

Mini Rev Med Chem 2016 ;16(16):1303-1320

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210023, People's Republic of China.

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http://dx.doi.org/10.2174/1389557516666160823143243DOI Listing
March 2017

A Quinoline-Based Ratiometric and Reversible Fluorescent Probe for Cadmium Imaging in Living Cells.

Chem Pharm Bull (Tokyo) 2016 30;64(1):27-33. Epub 2015 Oct 30.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University.

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http://dx.doi.org/10.1248/cpb.c15-00579DOI Listing
September 2016

Design, synthesis and biological evaluation of novel 5-phenyl-1H-pyrazole derivatives as potential BRAF(V600E) inhibitors.

Bioorg Med Chem 2014 Nov 6;22(21):6201-8. Epub 2014 Sep 6.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2014.08.029DOI Listing
November 2014

Design, synthesis and biological evaluation of metronidazole-thiazole derivatives as antibacterial inhibitors.

Bioorg Med Chem Lett 2014 Nov;24(22):5279-83

State Key Laboratory of Pharmaceutical Biotechnology, School of Life Science Nanjing University, Nanjing 210093, People’s Republic of China.

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November 2014

Discovery and molecular modeling of novel 1-indolyl acetate--5-nitroimidazole targeting tubulin polymerization as antiproliferative agents.

Eur J Med Chem 2014 Oct 30;85:341-51. Epub 2014 Jul 30.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2014.07.082DOI Listing
October 2014

Design, synthesis and molecular modeling of biquinoline-pyridine hybrids as a new class of potential EGFR and HER-2 kinase inhibitors.

Bioorg Med Chem Lett 2014 Sep 9;24(18):4472-4476. Epub 2014 Aug 9.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X140082
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http://dx.doi.org/10.1016/j.bmcl.2014.07.094DOI Listing
September 2014

Design, synthesis and biological evaluation of metronidazole-thiazole derivatives as antibacterial inhibitors.

Bioorg Med Chem Lett 2014 Sep 28. Epub 2014 Sep 28.

State Key Laboratory of Pharmaceutical Biotechnology, School of Life Science Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X140100
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http://dx.doi.org/10.1016/j.bmcl.2014.09.054DOI Listing
September 2014

Synthesis, biological evaluation and molecular modeling of 1,3,4-thiadiazol-2-amide derivatives as novel antitubulin agents.

Bioorg Med Chem 2014 Aug 17;22(15):4312-22. Epub 2014 May 17.

State Key Laboratory of Pharmaceutical Biotechnology, School of Life Sciences, Nanjing University, Nanjing 210093, PR China; School of Medicine, Nanjing University, Nanjing 210093, PR China. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S09680896140036
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http://dx.doi.org/10.1016/j.bmc.2014.05.017DOI Listing
August 2014

Synthesis, biological evaluation, and molecular docking studies of novel 2-styryl-5-nitroimidazole derivatives containing 1,4-benzodioxan moiety as FAK inhibitors with anticancer activity.

Bioorg Med Chem 2014 Jun 13;22(11):2947-54. Epub 2014 Apr 13.

State Key Laboratory of Pharmaceutical Biotechnology, School of Life Sciences, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2014.04.005DOI Listing
June 2014

Design, synthesis and molecular modeling of pyrazole-quinoline-pyridine hybrids as a new class of antimicrobial and anticancer agents.

Eur J Med Chem 2014 Apr 25;76:549-57. Epub 2014 Jan 25.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, China. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S02235234140004
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http://dx.doi.org/10.1016/j.ejmech.2014.01.018DOI Listing
April 2014

Schiff's base derivatives bearing nitroimidazole and quinoline nuclei: new class of anticancer agents and potential EGFR tyrosine kinase inhibitors.

Bioorg Med Chem Lett 2014 Apr 28;24(7):1734-6. Epub 2014 Feb 28.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2014.02.041DOI Listing
April 2014

Schiff's base derivatives bearing nitroimidazole moiety: new class of antibacterial, anticancer agents and potential EGFR tyrosine kinase inhibitors.

Bioorg Med Chem Lett 2013 Dec 8;23(23):6264-8. Epub 2013 Oct 8.

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People's Republic of China.

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http://dx.doi.org/10.1016/j.bmcl.2013.09.086DOI Listing
December 2013

1,3,4-oxadiazole derivatives as potential biological agents.

Mini Rev Med Chem 2013 Oct;13(12):1725-43

State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, P.R. China.

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http://dx.doi.org/10.2174/13895575113139990071DOI Listing
October 2013

Synthesis and antimicrobial evaluation of new pyrano[4,3-b]pyran and Pyrano[3,2-c]chromene derivatives bearing a 2-thiophenoxyquinoline nucleus.

Arch Pharm (Weinheim) 2012 Apr 22;345(4):314-22. Epub 2011 Nov 22.

Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar, Gujarat, India.

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http://dx.doi.org/10.1002/ardp.201100203DOI Listing
April 2012

Microwave assisted synthesis and antimicrobial evaluation of new fused pyran derivatives bearing 2-morpholinoquinoline nucleus.

Bioorg Med Chem Lett 2011 Oct 6;21(20):6166-9. Epub 2011 Aug 6.

Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar 388120, Gujarat, India.

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http://dx.doi.org/10.1016/j.bmcl.2011.07.123DOI Listing
October 2011