Publications by authors named "Jiantao Hu"

13Publications

Correction to: Targeted degradation of activating estrogen receptor α ligand-binding domain mutations in human breast cancer.

Authors:
Thomas L Gonzalez Molly Hancock Siqi Sun Christina L Gersch Jose M Larios Wadie David Jiantao Hu Daniel F Hayes Shaomeng Wang James M Rae

Breast Cancer Res Treat 2020 04;180(3):623

The University of Michigan Rogel Cancer Center, Ann Arbor, USA.

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April 2020

Targeted degradation of activating estrogen receptor α ligand-binding domain mutations in human breast cancer.

Authors:
Thomas L Gonzalez Molly Hancock Siqi Sun Christina L Gersch Jose M Larios Wadie David Jiantao Hu Daniel F Hayes Shaomeng Wang James M Rae

Breast Cancer Res Treat 2020 Apr 17;180(3):611-622. Epub 2020 Feb 17.

The University of Michigan Rogel Cancer Center, Ann Arbor, USA.

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April 2020

Discovery of ERD-308 as a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Estrogen Receptor (ER).

Authors:
Jiantao Hu Biao Hu Mingliang Wang Fuming Xu Bukeyan Miao Chao-Yie Yang Mi Wang Zhaomin Liu Daniel F Hayes Krishnapriya Chinnaswamy James Delproposto Jeanne Stuckey Shaomeng Wang

J Med Chem 2019 02 18;62(3):1420-1442. Epub 2019 Jan 18.

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February 2019

Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Inducing Complete and Durable Tumor Regression.

Authors:
Chong Qin Yang Hu Bing Zhou Ester Fernandez-Salas Chao-Yie Yang Liu Liu Donna McEachern Sally Przybranowski Mi Wang Jeanne Stuckey Jennifer Meagher Longchuan Bai Zhuo Chen Mei Lin Jiuling Yang Danya N Ziazadeh Fuming Xu Jiantao Hu Weiguo Xiang Liyue Huang Siwei Li Bo Wen Duxin Sun Shaomeng Wang

J Med Chem 2018 Aug 18;61(15):6685-6704. Epub 2018 Jul 18.

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August 2018

Learning from Natural Nacre: Constructing Layered Polymer Composites with High Thermal Conductivity.

Authors:
Guiran Pan Yimin Yao Xiaoliang Zeng Jiajia Sun Jiantao Hu Rong Sun Jian-Bin Xu Ching-Ping Wong

ACS Appl Mater Interfaces 2017 Sep 13;9(38):33001-33010. Epub 2017 Sep 13.

Shenzhen Institutes of Advanced Technology, Chinese Academy of Sciences , Shenzhen 518055, China.

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September 2017

Polymer Composite with Improved Thermal Conductivity by Constructing a Hierarchically Ordered Three-Dimensional Interconnected Network of BN.

Authors:
Jiantao Hu Yun Huang Yimin Yao Guiran Pan Jiajia Sun Xiaoliang Zeng Rong Sun Jian-Bin Xu Bo Song Ching-Ping Wong

ACS Appl Mater Interfaces 2017 Apr 5;9(15):13544-13553. Epub 2017 Apr 5.

Shenzhen Institutes of Advanced Technology, Chinese Academy of Sciences , Shenzhen 518055, China.

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April 2017

Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression.

Authors:
Bing Zhou Jiantao Hu Fuming Xu Zhuo Chen Longchuan Bai Ester Fernandez-Salas Mei Lin Liu Liu Chao-Yie Yang Yujun Zhao Donna McEachern Sally Przybranowski Bo Wen Duxin Sun Shaomeng Wang

J Med Chem 2018 01 24;61(2):462-481. Epub 2017 Mar 24.

University of Michigan Comprehensive Cancer Center, and Departments of ‡Internal Medicine, §Pathology, ∥Pharmaceutical Sciences, ⊥Medicinal Chemistry, and #Pharmacology, University of Michigan , Ann Arbor, Michigan 48109, United States.

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January 2018

Targeted Degradation of BET Proteins in Triple-Negative Breast Cancer.

Authors:
Longchuan Bai Bing Zhou Chao-Yie Yang Jiao Ji Donna McEachern Sally Przybranowski Hui Jiang Jiantao Hu Fuming Xu Yujun Zhao Liu Liu Ester Fernandez-Salas Jing Xu Yali Dou Bo Wen Duxin Sun Jennifer Meagher Jeanne Stuckey Daniel F Hayes Shunqiang Li Matthew J Ellis Shaomeng Wang

Cancer Res 2017 05 16;77(9):2476-2487. Epub 2017 Feb 16.

University of Michigan Comprehensive Cancer Center, University of Michigan, Ann Arbor, Michigan.

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May 2017

Interfacial Engineering of Silicon Carbide Nanowire/Cellulose Microcrystal Paper toward High Thermal Conductivity.

Authors:
Yimin Yao Xiaoliang Zeng Guiran Pan Jiajia Sun Jiantao Hu Yun Huang Rong Sun Jian-Bin Xu Ching-Ping Wong

ACS Appl Mater Interfaces 2016 Nov 4;8(45):31248-31255. Epub 2016 Nov 4.

Shenzhen Institutes of Advanced Technology, Chinese Academy of Sciences , Shenzhen 518055, China.

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November 2016

Unactivated C(sp(3))-H hydroxylation through palladium catalysis with H2O as the oxygen source.

Authors:
Jiantao Hu Tianlong Lan Yihua Sun Hui Chen Jiannian Yao Yu Rao

Chem Commun (Camb) 2015 Oct;51(80):14929-32

MOE Key Laboratory of Protein Sciences, Department of Pharmacology and Pharmaceutical Sciences, School of Medicine, Tsinghua University, Beijing, 100084, China.

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October 2015

Synthesis of indazoles and azaindazoles by intramolecular aerobic oxidative C-N coupling under transition-metal-free conditions.

Authors:
Jiantao Hu Huacheng Xu Pengju Nie Xiaobo Xie Zongxiu Nie Yu Rao

Chemistry 2014 Apr 3;20(14):3932-8. Epub 2014 Mar 3.

MOE Key Laboratory of Protein Sciences, Department of Pharmacology and Pharmaceutical Sciences, School of Medicine and School of Life Sciences, Tsinghua University, Beijing 100084 (China).

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April 2014

Synthesis of tri- and tetrasubstituted pyrazoles via Ru(II) catalysis: intramolecular aerobic oxidative C-N coupling.

Authors:
Jiantao Hu Shi Chen Yonghui Sun Jing Yang Yu Rao

Org Lett 2012 Oct 18;14(19):5030-3. Epub 2012 Sep 18.

Department of Pharmacology and Pharmaceutical Sciences, School of Medicine, Tsinghua University, Beijing 100084, China.

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October 2012

A general and efficient approach to 2H-indazoles and 1H-pyrazoles through copper-catalyzed intramolecular N-N bond formation under mild conditions.

Authors:
Jiantao Hu Yongfeng Cheng Yiqing Yang Yu Rao

Chem Commun (Camb) 2011 Sep 9;47(36):10133-5. Epub 2011 Aug 9.

Department of Pharmacology and Pharmaceutical Sciences, School of Life Sciences, Tsinghua University, Beijing 100084, China.

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September 2011