Publications by authors named "Jean Quancard"

22Publications

The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes.

ChemMedChem 2020 Dec 3;15(24):2388-2390. Epub 2020 Sep 3.

Pharmaceutical&Medicinal Chemistry, Institute of Pharmacy&Biochemistry, Tübingen Center for Academic Drug Discovery, Auf der Morgenstelle 8 D, 72070 Tuebingen, Germany.

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December 2020

A lead discovery strategy driven by a comprehensive analysis of proteases in the peptide substrate space.

Protein Sci 2010 Nov;19(11):2096-109

Lead Discovery Informatics, Lead Finding Platform, Novartis Institutes for BioMedical Research, Inc., 250 Massachusetts Avenue, Cambridge, Massachusetts 02139, USA.

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November 2010

Prolinoamino acids as tools to build bifunctionalized, stable beta-turns in water.

Chembiochem 2010 Jan;11(1):55-8

UPMC Université de Paris 06, UMR 7203 CNRS-UPMC-ENS, Laboratoire des Biomolécules, UPMC, 4 Place Jussieu, Paris Cedex 05, France.

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January 2010

Palladium-catalyzed enantioselective C-3 allylation of 3-substituted-1H-indoles using trialkylboranes.

J Am Chem Soc 2006 May;128(19):6314-5

Department of Chemistry, Stanford University, Stanford, California 94305-5080, USA.

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May 2006

Conformational analysis of the C-terminal Gly-Leu-Met-NH2 tripeptide of substance P bound to the NK-1 receptor.

Chem Biol 2005 May;12(5):555-65

Synthèse, Structure et Fonction de Molécules Bioactives, Unite Mixte de Recherche 7613, Centre National de la Recherche Scientifique-Université Paris 6, Paris, France.

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May 2005

Asymmetric synthesis of 3-substituted proline chimeras bearing polar side chains of proteinogenic amino acids.

J Org Chem 2004 Nov;69(23):7940-8

Synthèse, Structure et Fonction de Molécules Bioactives, CNRS/UMR 7613, Université Pierre et Marie Curie, 4 Place Jussieu, 75252 Paris Cedex 05, France.

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November 2004

Development of potent inhibitors of botulinum neurotoxin type B.

J Med Chem 2003 Oct;46(22):4648-56

Département de Pharmacochimie Moléculaire et Structurale, INSERM U266--CNRS FRE2463, UFR des Sciences Pharmaceutiques et Biologiques 4, Avenue de l'Observatoire--75270 Paris Cedex 06, France.

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October 2003

Purification and inactivation of 3-hydroxyanthranilic acid 3,4-dioxygenase from beef liver.

Int J Biochem Cell Biol 2003 Jul;35(7):1085-97

Department of Chemistry, Northwestern University, Evanston IL 60208-3113, USA.

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July 2003