Publications by authors named "Haridas B Rode"

20Publications

Synthesis of novel 4,5-dihydropyrrolo[1,2-a]quinoxalines, pyrrolo[1,2-a]quinoxalin]-2-ones and their antituberculosis and anticancer activity.

Arch Pharm (Weinheim) 2020 Aug 12:e2000192. Epub 2020 Aug 12.

Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Hyderabad, Telangana, India.

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http://dx.doi.org/10.1002/ardp.202000192DOI Listing
August 2020

Synthesis and efficacy of pyrvinium-inspired analogs against tuberculosis and malaria pathogens.

Bioorg Med Chem Lett 2020 04 14;30(8):127037. Epub 2020 Feb 14.

Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad 500 007, India; Academy of Scientific and Innovative Research, Ghaziabad, Uttar Pradesh 201 002, India. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2020.127037DOI Listing
April 2020

Catalyst-Free Regioselective [3+2] Cycloadditions of α,β-unsaturated N-arylnitrones with Alkenes to Access Functionalized Isoxazolidines: A DFT Study.

Chem Asian J 2020 Mar 24;15(6):899-903. Epub 2020 Feb 24.

Centre for Nano and Material Sciences, Jain University, Jain Global Campus, Bangalore, Karnataka, 562112, India.

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http://dx.doi.org/10.1002/asia.201901754DOI Listing
March 2020

Synthesis and biological evaluation of 2,4,5-trisubstituted thiazoles as antituberculosis agents effective against drug-resistant tuberculosis.

Eur J Med Chem 2019 Sep 4;178:315-328. Epub 2019 Jun 4.

Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad, 500007, India; Academy of Scientific and Innovative Research (AcSIR), Ghaziabad, Uttar Pradesh, 201 002, India. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2019.05.082DOI Listing
September 2019

Strategies towards the synthesis of anti-tuberculosis drugs.

Org Biomol Chem 2019 06;17(22):5428-5459

Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad-500007, India.

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http://dx.doi.org/10.1039/c9ob00817aDOI Listing
June 2019

Transition metal-free functionalized hydration of alkynes: one-pot synthesis of fluorinated β-keto-imidates using Selectfluor.

Org Biomol Chem 2019 05;17(18):4440-4445

Centre for Nano and Material Sciences, Jain Global Campus, JAIN (Deemed-to-be-University), Bangalore, Karnataka 562112, India.

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http://dx.doi.org/10.1039/c9ob00527gDOI Listing
May 2019

Novel 1,3,4-oxadiazoles as antitubercular agents with limited activity against drug-resistant tuberculosis.

Future Med Chem 2019 03 20;11(6):499-510. Epub 2019 Mar 20.

Department of Organic Synthesis & Process Chemistry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad 500 007, India.

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https://www.future-science.com/doi/10.4155/fmc-2018-0378
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http://dx.doi.org/10.4155/fmc-2018-0378DOI Listing
March 2019

Synthesis and evaluation of α-aminoacyl amides as antitubercular agents effective on drug resistant tuberculosis.

Eur J Med Chem 2019 Feb 3;164:665-677. Epub 2019 Jan 3.

Department of Organic Synthesis and Process Chemistry, CSIR-Indian Institute of Chemical Technology, Tarnaka, Hyderabad, 500 007, India; Academy of Scientific and Innovative Research, Ghaziabad, Uttar Pradesh, 201 002, India. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2019.01.002DOI Listing
February 2019

Crosslinked enzyme aggregates (CLEA) of phytase with soymilk proteins.

J Biotechnol 2018 Sep 4;282:67-69. Epub 2018 Jul 4.

Organic Synthesis and Process Chemistry Division, Indian Institute of Chemical Technology, Hyderabad, 500 007, India. Electronic address:

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http://dx.doi.org/10.1016/j.jbiotec.2018.07.003DOI Listing
September 2018

Methyl 3-[(1,1-dioxo-1λ(6),2-benzothiazol-3-yl)amino]-5-nitrothiophene-2-carboxyl-ate.

Acta Crystallogr Sect E Struct Rep Online 2012 Oct 19;68(Pt 10):o2951-2. Epub 2012 Sep 19.

Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, Ernst-Moritz-Arndt-University, Friedrich-Ludwig-Jahn-Str. 17, Greifswald, D-17489, Germany ; Council Scientific and Industrial Research (CSIR) Head Quarter, Anusandhan Bhavan, 2 Rafi Marg, Delhi-110001, India.

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http://scripts.iucr.org/cgi-bin/paper?S1600536812038378
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http://dx.doi.org/10.1107/S1600536812038378DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3470323PMC
October 2012

A chemical genetic approach for covalent inhibition of analogue-sensitive aurora kinase.

ACS Chem Biol 2012 Apr 1;7(4):723-31. Epub 2012 Feb 1.

Friedrich Miescher Laboratory of the Max Planck Society, Tübingen, Germany.

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http://dx.doi.org/10.1021/cb200465cDOI Listing
April 2012

Synthesis and biological evaluation of 7-substituted-1-(3-bromophenylamino)isoquinoline-4-carbonitriles as inhibitors of myosin light chain kinase and epidermal growth factor receptor.

Bioorg Med Chem 2011 Jan 10;19(1):429-39. Epub 2010 Nov 10.

Chemical Genomics Centre of the Max Planck Society, Otto-Hahn-Strasse 15, 44227 Dortmund, Germany.

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http://dx.doi.org/10.1016/j.bmc.2010.11.007DOI Listing
January 2011

Hybrid compound design to overcome the gatekeeper T338M mutation in cSrc.

J Med Chem 2009 Jul;52(13):3915-26

Chemical Genomics Centre of the Max Planck Society, D-44227 Dortmund, Germany.

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http://dx.doi.org/10.1021/jm9002928DOI Listing
July 2009

A new screening assay for allosteric inhibitors of cSrc.

Nat Chem Biol 2009 Jun 26;5(6):394-6. Epub 2009 Apr 26.

Chemical Genomics Centre of the Max Planck Society, Dortmund, Germany.

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http://dx.doi.org/10.1038/nchembio.162DOI Listing
June 2009

Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR.

Bioorg Med Chem 2008 Apr 20;16(7):3482-8. Epub 2008 Feb 20.

Chemical Genomics Centre of the Max-Planck-Society, Otto-Hahn-Strasse 15, 44227 Dortmund, Germany.

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https://linkinghub.elsevier.com/retrieve/pii/S09680896080017
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http://dx.doi.org/10.1016/j.bmc.2008.02.053DOI Listing
April 2008