Publications by authors named "Haiyan Bian"

8Publications

The discovery of azetidine-piperazine di-amides as potent, selective and reversible monoacylglycerol lipase (MAGL) inhibitors.

Authors:
Bin Zhu Peter J Connolly Yue-Mei Zhang Mark E McDonnell Haiyan Bian Shu-Chen Lin Li Liu Sui-Po Zhang Kristen M Chevalier Michael R Brandt Cynthia M Milligan Christopher M Flores Mark J Macielag

Bioorg Med Chem Lett 2020 07 7;30(14):127243. Epub 2020 May 7.

Janssen Research & Development, L.L.C., Welsh & McKean Roads, Spring House, PA 19477, USA.

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July 2020

Tuning isoform selectivity and bortezomib sensitivity with a new class of alkenyl indene PDI inhibitor.

Authors:
Reeder M Robinson Leticia Reyes Ravyn M Duncan Haiyan Bian Eric D Strobel Sarah L Hyman Allen B Reitz Nathan G Dolloff

Eur J Med Chem 2020 Jan 21;186:111906. Epub 2019 Nov 21.

Department of Cell and Molecular Pharmacology & Experimental Therapeutics, College of Medicine, Medical University of South Carolina, Charleston, SC, USA. Electronic address:

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January 2020

Inhibitors of the protein disulfide isomerase family for the treatment of multiple myeloma.

Authors:
Reeder M Robinson Leticia Reyes Ravyn M Duncan Haiyan Bian Allen B Reitz Yefim Manevich Jesse J McClure Matthew M Champion C James Chou Meahgen E Sharik Marta Chesi P Leif Bergsagel Nathan G Dolloff

Leukemia 2019 04 12;33(4):1011-1022. Epub 2018 Oct 12.

Department of Cell and Molecular Pharmacology & Experimental Therapeutics, College of Medicine, Medical University of South Carolina, Charleston, SC, USA.

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April 2019

Dipeptide Prodrugs of the Glutamate Modulator Riluzole.

Authors:
Jeffrey C Pelletier Suzie Chen Haiyan Bian Raj Shah Garry R Smith Jay E Wrobel Allen B Reitz

ACS Med Chem Lett 2018 Jul 15;9(7):752-756. Epub 2018 Jun 15.

Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, Pennsylvania 18902, United States.

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July 2018

High-Throughput Screening Uncovers Novel Botulinum Neurotoxin Inhibitor Chemotypes.

Authors:
Kristin M Bompiani Dejan Caglič Michelle C Krutein Galit Benoni Morgan Hrones Luke L Lairson Haiyan Bian Garry R Smith Tobin J Dickerson

ACS Comb Sci 2016 08 20;18(8):461-74. Epub 2016 Jul 20.

Department of Chemistry, The Scripps Research Institute , 10550 North Torrey Pines Road, La Jolla, California 92037, United States.

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August 2016

Anilino-monoindolylmaleimides as potent and selective JAK3 inhibitors.

Authors:
Mark E McDonnell Haiyan Bian Jay Wrobel Garry R Smith Shuguang Liang Haiching Ma Allen B Reitz

Bioorg Med Chem Lett 2014 Feb 9;24(4):1116-21. Epub 2014 Jan 9.

Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States.

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February 2014

Indole-glucosides as novel sodium glucose co-transporter 2 (SGLT2) inhibitors. Part 2.

Authors:
Xiaoyan Zhang Maud Urbanski Mona Patel Geoffrey G Cox Roxanne E Zeck Haiyan Bian Bruce R Conway Mary Pat Beavers Philip J Rybczynski Keith T Demarest

Bioorg Med Chem Lett 2006 Mar 27;16(6):1696-701. Epub 2005 Dec 27.

Johnson & Johnson Pharmaceutical Research and Development, L.L.C., 1000 Rt. 202, PO Box 300, Raritan, NJ 08869, USA.

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March 2006

Heteroaryl-O-glucosides as novel sodium glucose co-transporter 2 inhibitors. Part 1.

Authors:
Xiaoyan Zhang Maud Urbanski Mona Patel Roxanne E Zeck Geoffrey G Cox Haiyan Bian Bruce R Conway Mary Pat Beavers Philip J Rybczynski Keith T Demarest

Bioorg Med Chem Lett 2005 Dec 28;15(23):5202-6. Epub 2005 Sep 28.

Johnson & Johnson Pharmaceutical Research and Development, L.L.C., 1000 Rt. 202, PO Box 300, Raritan, NJ 08869, USA.

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December 2005