Publications by authors named "Frederic Berst"

11Publications

An Amphiphilic Polymer-Supported Strategy Enables Chemical Transformations under Anhydrous Conditions for DNA-Encoded Library Synthesis.

ACS Comb Sci 2020 03 27;22(3):120-128. Epub 2020 Feb 27.

Novartis Institutes for BioMedical Research, Novartis Pharma AG, Novartis Campus, CH-4002, Basel, Switzerland.

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March 2020

Efficient copper-catalyzed amination of DNA-conjugated aryl iodides under mild aqueous conditions.

Medchemcomm 2018 Jul 17;9(7):1188-1193. Epub 2018 May 17.

Novartis Institutes for BioMedical Research , Novartis Pharma AG , Novartis Campus , 4002 Basel , Switzerland . Email:

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July 2018

Trypsin inhibitors for the treatment of pancreatitis.

Bioorg Med Chem Lett 2016 09 17;26(17):4340-4. Epub 2016 Jul 17.

Novartis Pharma AG, Cardio Metabolic Development Franchise, Novartis Campus, CH-4002 Basel, Switzerland.

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September 2016

Substrate profiling of IGF-1R and InsR: identification of a potent pentamer substrate.

Bioorg Med Chem Lett 2011 Dec 29;21(23):7030-3. Epub 2011 Sep 29.

Novartis Institutes for BioMedical Research, Basel, Switzerland.

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December 2011

Straightforward preparation and assay of aspartyl protease substrates with an internal thioester linkage.

Chembiochem 2007 Jun;8(9):981-4

Department of Chemistry, University of California, Berkeley, Berkley, CA 94720, USA.

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June 2007

The development and preparation of the 2,4-dimethoxybenzyl arylhydrazine (DMBAH) "latent" safety-catch linker: solid phase synthesis of ketopiperazines.

Org Biomol Chem 2003 May;1(10):1711-9

GSK Cambridge Technology Centre, University Chemical Laboratory, Lensfield Road, Cambridge, UK CB2 1EW.

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May 2003

Solid-phase synthesis of apicidin A and a cyclic tetrapeptoid analogue.

Chem Commun (Camb) 2002 Mar(5):508-9

GSK Cambridge Technology Centre, Lensfield Road, Cambridge, UK CB2 1EW.

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March 2002