Frank E Kwarcinski

Frank E Kwarcinski

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Frank E Kwarcinski

Frank E Kwarcinski

Publications by authors named "Frank E Kwarcinski"

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Selective Proteolysis to Study the Global Conformation and Regulatory Mechanisms of c-Src Kinase.

ACS Chem Biol 2019 Jul 9;14(7):1556-1563. Epub 2019 Jul 9.

Department of Internal Medicine , University of Michigan , Ann Arbor , Michigan 48109 , United States.

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http://dx.doi.org/10.1021/acschembio.9b00306DOI Listing
July 2019

Conformation-Selective Analogues of Dasatinib Reveal Insight into Kinase Inhibitor Binding and Selectivity.

ACS Chem Biol 2016 05 1;11(5):1296-304. Epub 2016 Mar 1.

Department of Pharmacological Sciences, Stony Brook University , Stony Brook, New York 11794, United States.

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http://dx.doi.org/10.1021/acschembio.5b01018DOI Listing
May 2016

Discovery of Bivalent Kinase Inhibitors via Enzyme-Templated Fragment Elaboration.

ACS Med Chem Lett 2015 Aug 13;6(8):898-901. Epub 2015 Jul 13.

Departments of Medicinal Chemistry and Chemistry, University of Michigan , 930 North University Avenue, Ann Arbor, Michigan 48109, United States.

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http://dx.doi.org/10.1021/acsmedchemlett.5b00167DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4538437PMC
August 2015

Substrate activity screening with kinases: discovery of small-molecule substrate-competitive c-Src inhibitors.

Angew Chem Int Ed Engl 2014 Jul 2;53(27):7010-3. Epub 2014 May 2.

Departments of Medicinal Chemistry and Chemistry, University of Michigan, 930 N. University Avenue, Ann Arbor, MI 48109 (USA).

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http://dx.doi.org/10.1002/anie.201311096DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4108202PMC
July 2014

Irreversible inhibitors of c-Src kinase that target a nonconserved cysteine.

ACS Chem Biol 2012 Nov 5;7(11):1910-7. Epub 2012 Sep 5.

Department of Medicinal Chemistry, University of Michigan, 930 N. University Avenue, Ann Arbor, Michigan 48109, United States.

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http://pubs.acs.org/doi/abs/10.1021/cb300337u
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http://dx.doi.org/10.1021/cb300337uDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3500393PMC
November 2012