Francis C Colpaert

Francis C Colpaert

UNVERIFIED PROFILE

Are you Francis C Colpaert?   Register this Author

Register author
Francis C Colpaert

Francis C Colpaert

Publications by authors named "Francis C Colpaert"

Are you Francis C Colpaert?   Register this Author

31Publications

144Reads

44Profile Views

[(3)H]-F13640, a novel, selective and high-efficacy serotonin 5-HT(1A) receptor agonist radioligand.

Naunyn Schmiedebergs Arch Pharmacol 2010 Oct 27;382(4):321-30. Epub 2010 Aug 27.

Department of Cellular and Molecular Biology, Centre de Recherche Pierre Fabre, Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1007/s00210-010-0551-4DOI Listing
October 2010

F15599, a preferential post-synaptic 5-HT1A receptor agonist: activity in models of cognition in comparison with reference 5-HT1A receptor agonists.

Eur Neuropsychopharmacol 2010 Sep 21;20(9):641-54. Epub 2010 May 21.

Neurobiology 2 Division, Centre de Recherche Pierre Fabre, 17, avenue Jean Moulin, 81106 Castres, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.euroneuro.2010.04.005DOI Listing
September 2010

Long-lasting descending and transitory short-term spinal controls on deep spinal dorsal horn nociceptive-specific neurons in response to persistent nociception.

Brain Res Bull 2008 Jan 6;75(1):34-41. Epub 2007 Aug 6.

Department of Physiology and Pathophysiology, Xi'an Jiaotong University School of Medicine, Xi'an, Shaanxi 710061, PR China.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.brainresbull.2007.07.015DOI Listing
January 2008

Curative-like analgesia in a neuropathic pain model: parametric analysis of the dose and the duration of treatment with a high-efficacy 5-HT(1A) receptor agonist.

Eur J Pharmacol 2007 Jul 22;568(1-3):134-41. Epub 2007 Apr 22.

Laboratory of Anesthesiology, University of Antwerp, Universiteitsplein 1, 2610 Antwerp, Belgium.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.ejphar.2007.04.022DOI Listing
July 2007

High-efficacy 5-hydroxytryptamine 1A receptor activation counteracts opioid hyperallodynia and affective conditioning.

J Pharmacol Exp Ther 2006 Feb 27;316(2):892-9. Epub 2005 Oct 27.

Centre de Recherche Pierre Fabre, Castres, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1124/jpet.105.095109DOI Listing
February 2006

5-HT(1A) receptor activation: new molecular and neuroadaptive mechanisms of pain relief.

Curr Opin Investig Drugs 2006 Jan;7(1):40-7

Institut de Recherche Pierre Fabre, 3 rue des Satellites, BP 94244, 31432 Toulouse 4, France.

View Article

Download full-text PDF

Source
January 2006

Differential ion current activation by human 5-HT(1A) receptors in Xenopus oocytes: evidence for agonist-directed trafficking of receptor signalling.

Neuropharmacology 2005 Dec 17;49(7):963-76. Epub 2005 Jun 17.

Centre de Recherche Pierre Fabre, 17, Avenue Jean Moulin, F-81106 Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.neuropharm.2005.05.001DOI Listing
December 2005

The novel analgesic, F 13640, produces intra- and postoperative analgesia in a rat model of surgical pain.

Eur J Pharmacol 2005 Oct 13;523(1-3):29-39. Epub 2005 Oct 13.

Klinik für Anästhesie, Intensivmedizin und Schmerztherapie, Alfried Krupp Krankenhaus, 45117 Essen, Germany.

View Article

Download full-text PDF

Source
http://linkinghub.elsevier.com/retrieve/pii/S001429990500907
Publisher Site
http://dx.doi.org/10.1016/j.ejphar.2005.09.003DOI Listing
October 2005

Nociceptive spinal withdrawal reflexes but not spinal dorsal horn wide-dynamic range neuron activities are specifically inhibited by halothane anaesthesia in spinalized rats.

Eur J Neurosci 2005 Jul;22(2):354-60

Center for Sensory-Motor Interaction (SMI), Laboratory for Experimental Pain Research, Aalborg University, Fredrik Bajers Vej 7 D-3, DK-9220 Aalborg, Denmark.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1111/j.1460-9568.2005.04234.xDOI Listing
July 2005

The novel analgesic and high-efficacy 5-HT1A receptor agonist F 13640 inhibits nociceptive responses, wind-up, and after-discharges in spinal neurons and withdrawal reflexes.

Exp Neurol 2005 Jan;191(1):174-83

Center for Sensory-Motor Interaction, Laboratory for Experimental Pain Research Aalborg University, Aalborg 9220, Denmark.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.expneurol.2004.08.031DOI Listing
January 2005

Effects of the combined continuous administration of morphine and the high-efficacy 5-HT1A agonist, F 13640 in a rat model of trigeminal neuropathic pain.

Eur J Pain 2004 Dec;8(6):547-54

Laboratory of Anesthesiology, University of Antwerp, Universiteitsplein 1, B-2610 Antwerp, Belgium.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.ejpain.2004.01.002DOI Listing
December 2004

High-efficacy 5-HT1A receptor activation causes a curative-like action on allodynia in rats with spinal cord injury.

Eur J Pharmacol 2004 Aug;497(1):29-33

Centre de Recherche Pierre Fabre, 17 Avenue Jean Moulin, 81100 Castres, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.ejphar.2004.06.026DOI Listing
August 2004

KC 12291: an atypical sodium channel blocker with myocardial antiischemic properties.

Cardiovasc Drug Rev 2004 ;22(1):17-26

Centre de Recherche Pierre Fabre, 17, Avenue Jean Moulin, 81100 Castres, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1111/j.1527-3466.2004.tb00129.xDOI Listing
July 2004

Role of spinal 5-HT(1A) receptors in morphine analgesia and tolerance in rats.

Eur J Pain 2004 Jun;8(3):253-61

Centre de Recherche Pierre-Fabre, 17 Avenue Jean Moulin, Castres Cédex F-81106, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.ejpain.2003.09.002DOI Listing
June 2004

Ability of dopamine antagonists to inhibit the locomotor effects of cocaine in sensitized and non-sensitized C57BL/6 mice depends on the challenge dose.

Psychopharmacology (Berl) 2004 Apr 11;172(4):409-14. Epub 2003 Dec 11.

Centre de Recherche Pierre Fabre, 17 Avenue Jean Moulin, 81106 Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1007/s00213-003-1691-8DOI Listing
April 2004

Noradrenergic mechanisms in neurodegenerative diseases: a theory.

Brain Res Brain Res Rev 2004 Apr;45(1):38-78

Centre de Recherche Pierre Fabre, Neurobiology I, 17 Avenue Jean Moulin, 81106 Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.brainresrev.2004.02.002DOI Listing
April 2004

Ca2+ responses in Chinese hamster ovary-K1 cells demonstrate an atypical pattern of ligand-induced 5-HT1A receptor activation.

J Pharmacol Exp Ther 2003 Nov 11;307(2):608-14. Epub 2003 Sep 11.

Centre d'Immunologie Pierre Fabre, 5 avenue Napoléon III-BP 497, F 74164 Saint-Julien-en-Genevois Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1124/jpet.103.055871DOI Listing
November 2003

The very-high-efficacy 5-HT1A receptor agonist, F 13640, preempts the development of allodynia-like behaviors in rats with spinal cord injury.

Eur J Pharmacol 2003 Oct;478(2-3):131-7

Division of Clinical Neurophysiology, Department of Medical Laboratory Sciences and Technology, Huddinge University Hospital, Huddinge, Sweden.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.ejphar.2003.08.047DOI Listing
October 2003

Discovering risperidone: the LSD model of psychopathology.

Nat Rev Drug Discov 2003 04;2(4):315-20

Centre de Recherche Pierre Fabre, 17 avenue Jean Moulin, 81106 Castres Cédex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1038/nrd1062DOI Listing
April 2003

Tolerance and inverse tolerance to the hyperalgesic and analgesic actions, respectively, of the novel analgesic, F 13640.

Eur J Pharmacol 2003 Apr;466(3):271-9

Centre de Recherche Pierre Fabre, 17 Avenue Jean Moulin, 81106 Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/s0014-2999(03)01566-8DOI Listing
April 2003

Tacrine-scopolamine interactions on state-dependent retrieval.

Psychopharmacology (Berl) 2003 Feb 19;166(1):33-9. Epub 2002 Dec 19.

Centre de Recherche Pierre Fabre, 17 avenue Jean Moulin, 81106 Castres Cedex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1007/s00213-002-1292-yDOI Listing
February 2003

Constitutive coupling of a chimeric dopamine D2/alpha 1B receptor to the phospholipase C pathway: inverse agonism to silent antagonism by neuroleptic drugs.

J Pharmacol Exp Ther 2003 Jan;304(1):380-90

Department of Cellular and Molecular Biology, Centre de Recherche Pierre Fabre, Castres Cédex, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1124/jpet.102.040535DOI Listing
January 2003

The 5-HT(1A) receptor agonist F 13640 attenuates mechanical allodynia in a rat model of trigeminal neuropathic pain.

Eur J Pharmacol 2002 Dec;456(1-3):51-7

Laboratory of Anesthesiology S4, University of Antwerp, Universiteitsplein 1, B-2610 Antwerp, Belgium.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/s0014-2999(02)02640-7DOI Listing
December 2002

5-HT1A receptor activation and anti-cataleptic effects: high-efficacy agonists maximally inhibit haloperidol-induced catalepsy.

Eur J Pharmacol 2002 Oct;453(2-3):217-21

Centre de Recherche Pierre Fabre, 17 Avenue Jean Moulin, F-81106 cedex, Castres, France.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/s0014-2999(02)02430-5DOI Listing
October 2002