Publications by authors named "Florian Thaler"

22Publications

Novel potent inhibitors of the histone demethylase KDM1A (LSD1), orally active in a murine promyelocitic leukemia model.

Future Med Chem 2017 07 19;9(11):1161-1174. Epub 2017 Jul 19.

Department of Experimental Oncology, Academic Drug Discovery, European Institute of Oncology, Ifom-IEO-Campus, via Adamello 16, 20139 Milan, Italy.

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July 2017

Compounds and methods for inhibiting histone demethylases: a patent evaluation of US20160102096A1.

Expert Opin Ther Pat 2016 Dec 21;26(12):1367-1370. Epub 2016 Oct 21.

a Experimental Therapeutics Unit , IFOM - The FIRC Institute of Molecular Oncology , Milan , Italy.

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December 2016

Current trends in the development of histone deacetylase inhibitors: a review of recent patent applications.

Authors:
Florian Thaler

Pharm Pat Anal 2012 Mar;1(1):75-90

Drug Discovery Unit, European Institute of Oncology, Via Adamello 16, 20139 Milan, Italy.

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March 2012

Next generation histone deacetylase inhibitors: the answer to the search for optimized epigenetic therapies?

Expert Opin Drug Discov 2011 Apr 23;6(4):393-404. Epub 2011 Feb 23.

European Institute of Oncology, Drug Discovery Unit, Department of Experimental Oncology, Via Celoria 26, 20133 Milan, Italy.

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April 2011

Polymer-supported scavengers for purification of labeled proteins.

Anal Biochem 2005 Jun;341(2):379-81

DIBIT-Laboratory of Dynamic Fluorescence Spectroscopy, Scientific Institute San Raffaele, Via Olgettina 58, 20132 Milan, Italy.

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June 2005

Reaction behaviour of dinuclear copper(I) complexes with m-xylyl-based ligands towards dioxygen.

Dalton Trans 2004 Aug 30(15):2321-8. Epub 2004 Jun 30.

Institut fur Anorganische und Analytische Chemie, Justus-Liebig-Universitat Giessen, Heinrich-Buff-Ring 58, 35392 Giessen, Germany.

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August 2004