Publications by authors named "Ernst Blum"

4Publications

Modulating ADME Properties by Fluorination: MK2 Inhibitors with Improved Oral Exposure.

Authors:
Juraj Velcicky Achim Schlapbach Richard Heng Laszlo Revesz Daniel Pflieger Ernst Blum Stuart Hawtin Christine Huppertz Roland Feifel Rene Hersperger

ACS Med Chem Lett 2018 Apr 20;9(4):392-396. Epub 2018 Mar 20.

Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.

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April 2018

Pyrazoloheteroaryls: novel p38alpha MAP kinase inhibiting scaffolds with oral activity.

Authors:
Laszlo Revesz Ernst Blum Franco E Di Padova Thomas Buhl Roland Feifel Hermann Gram Peter Hiestand Ute Manning Ulf Neumann Gerard Rucklin

Bioorg Med Chem Lett 2006 Jan 24;16(2):262-6. Epub 2005 Oct 24.

Novartis Institutes for BioMedical Research, Global Discovery Chemistry, CH-4002 Basel, Switzerland.

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January 2006

SAR of benzoylpyridines and benzophenones as p38alpha MAP kinase inhibitors with oral activity.

Authors:
Laszlo Revesz Ernst Blum Franco E Di Padova Thomas Buhl Roland Feifel Hermann Gram Peter Hiestand Ute Manning Gerard Rucklin

Bioorg Med Chem Lett 2004 Jul;14(13):3601-5

Novartis Institutes for BioMedical Research, Arthritis and Bone Metabolism, CH-4002 Basel, Switzerland.

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July 2004

Novel p38 inhibitors with potent oral efficacy in several models of rheumatoid arthritis.

Authors:
Laszlo Revesz Ernst Blum Franco E Di Padova Thomas Buhl Roland Feifel Hermann Gram Peter Hiestand Ute Manning Gerard Rucklin

Bioorg Med Chem Lett 2004 Jul;14(13):3595-9

Novartis Institutes for BioMedical Research, Arthritis & Bone Metabolism, CH-4002 Basel, Switzerland.

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July 2004