47 Publications
Bioorg Med Chem Lett 2020 11 29;30(22):127589. Epub 2020 Sep 29.
Discovery Chemistry, Janssen Pharmaceutical Research & Development, 1400 McKean Rd, Spring House, PA 19477, USA. Electronic address:
J Antimicrob Chemother 2020 09;75(9):2526-2534
Janssen Research and Development, Turnhoutseweg 30, 2340 Beerse, Belgium.
Methods Mol Biol 2018 ;1825:425-450
Life Science Informatics Research Unit, Laboratory of Molecular Biosciences, Kyoto University Graduate School of Medicine, Kyoto, Japan.
Methods Mol Biol 2018 ;1787:183-193
Janssen Research and Development, Beerse, Belgium.
Mol Inform 2018 05 8;37(5):e1700119. Epub 2017 Nov 8.
Janssen Research & Development, Turnhoutseweg 30, 2340, Beerse, Belgium.
J Med Chem 2016 07 6;59(14):6973. Epub 2016 Jul 6.
PLoS One 2016 8;11(1):e0146100. Epub 2016 Jan 8.
Evotec (München) GmbH, Martinsried, Germany.
J Proteome Res 2015 Oct 25;14(10):4179-93. Epub 2015 Aug 25.
Department of Medical Protein Research, VIB , A. Baertsoenkaai 3, 9000 Ghent, Belgium.
Bioorg Med Chem Lett 2015 Sep 23;25(17):3621-5. Epub 2015 Jun 23.
Novartis Institutes for BioMedical Research, WKL-136.P.12, CH-4002 Basel, Switzerland. Electronic address:
J Proteome Res 2015 Apr 12;14(4):1987-90. Epub 2015 Mar 12.
†Department of Medical Protein Research, VIB, Albert Baertsoenkaai 3, B-9000 Ghent, Belgium.
J Med Chem 2015 Feb 10;58(4):1818-31. Epub 2015 Feb 10.
Institut de Chimie Organique et Analytique, UMR CNRS-Université d'Orléans 7311 , Université d'Orléans BP 6759, Orléans 45067 Cedex 2, France.
Drug Discov Today 2015 Jun 14;20(6):652-8. Epub 2015 Jan 14.
Janssen Research & Development, Turnhoutseweg 30, 2340 Beerse, Belgium. Electronic address:
PLoS One 2014 18;9(12):e115460. Epub 2014 Dec 18.
Swiss Institute of Bioinformatics, CALIPHO Group, CMU - Rue Michel-Servet 1, 1211 Geneva 4, Switzerland.
Drug Discov Today 2013 Sep 20;18(17-18):843-52. Epub 2013 May 20.
Novartis Institutes for BioMedical Research, Novartis Pharma AG, Forum 1 Novartis Campus, CH-4056 Basel, Switzerland.
J Med Chem 2013 Mar 15;56(6):2207-17. Epub 2013 Mar 15.
Novartis Pharma AG, Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
J Med Chem 2013 Mar 15;56(6):2196-206. Epub 2013 Mar 15.
J Biomol Screen 2013 Jan 1;18(1):1-13. Epub 2012 Aug 1.
Informatics and Technology, Novartis Pharma AG, Institutes for BioMedical Research, Basel, Switzerland.
J Chem Inf Model 2012 May 19;52(5):1167-78. Epub 2012 Apr 19.
Novartis Institutes for BioMedical Research, Novartis Pharma AG, Forum 1, Novartis Campus, CH-4056 Basel, Switzerland.
J Chem Inf Model 2011 Dec 11;51(12):3093-8. Epub 2011 Nov 11.
Future Med Chem 2011 Apr;3(6):751-66
Novartis Institutes for BioMedical Research, Center for Proteomic Chemistry, Forum 1, Novartis Campus, CH-4056 Basel, Switzerland.
Curr Opin Chem Biol 2011 Aug 14;15(4):540-6. Epub 2011 Mar 14.
Novartis Institutes for BioMedical Research, Inc., 250 Massachusetts Avenue, Cambridge, MA 02139, USA.
Methods Mol Biol 2009 ;575:173-94
Novartis Institutes for BioMedical Research, Novartis Pharma AG, Basel, Switzerland.
Antimicrob Agents Chemother 2009 May 17;53(5):1823-31. Epub 2009 Feb 17.
Novartis Institute for Tropical Diseases, 10 Biopolis Rd., Chromos Building, Singapore 138670, Singapore.
Curr Opin Drug Discov Devel 2008 May;11(3):327-37
Lead Finding Platform, Novartis Institutes for Biomedical Research, Cambridge, MA 02139, USA.
ChemMedChem 2007 Jun;2(6):874-80
CPC/LFP/MLI, Novartis Institutes for Biomedical Research, Novartis Pharma AG, Postfach, 4002 Basel, Switzerland.
J Chem Inf Model 2007 May-Jun;47(3):1171-81. Epub 2007 May 10.
M.M. Shemyakin & Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Ul. Miklukho-Maklaya, 16/10, 117997 GSP, Moscow V-437, Russia.
J Mol Model 2007 Aug 9;13(8):897-905. Epub 2007 May 9.
Novartis Institutes for BioMedical Research, Discovery Technologies, Basel, Switzerland.
Curr Med Chem 2007 ;14(4):393-415
M.M. Shemyakin and Yu.A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Ul. Miklukho-Maklaya, 16/10, Moscow V-437, 117997 GSP, Russia.
Mini Rev Med Chem 2006 Nov;6(11):1217-29
Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
Proteins 2007 Feb;66(2):388-98
M.M. Shemyakin & Yu. A. Ovchinnikov Institute of Bioorganic Chemistry, Russian Academy of Sciences, Ul. Miklukho-Maklaya, 16/10, 117997 GSP, Moscow V-437, Russia.