Publications by authors named "Dumrongsak Pekthong"

13Publications

Elucidation of Vasodilation Response and Structure Activity Relationships of ²,⁴Disubstituted Quinazoline 2,4-Diamines in a Rat Pulmonary Artery Model.

Authors:
Tamkeen Urooj Paracha Nattakarn Pobsuk Nattapas Salaloy Praphasri Suphakun Dumrongsak Pekthong Supa Hannongbua Kiattawee Choowongkomon Nantaka Khorana Prapapan Temkitthawon Kornkanok Ingkaninan M Paul Gleeson Krongkarn Chootip

Molecules 2019 Jan 14;24(2). Epub 2019 Jan 14.

Department of Physiology, Faculty of Medical Science, Naresuan University, Phitsanulok 65000, Thailand.

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January 2019

Design, synthesis and evaluation of N,N-diaminoquinazoline based inhibitors of phosphodiesterase type 5.

Authors:
Nattakarn Pobsuk Tamkeen Urooj Paracha Nattiya Chaichamnong Nattapas Salaloy Praphasri Suphakun Supa Hannongbua Kiattawee Choowongkomon Dumrongsak Pekthong Krongkarn Chootip Kornkanok Ingkaninan M Paul Gleeson

Bioorg Med Chem Lett 2019 01 22;29(2):267-270. Epub 2018 Nov 22.

Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang 10520, Thailand. Electronic address:

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January 2019

Suppressed lipogenesis by plasma membrane citrate transporter inhibitor promotes apoptosis in HepG2 cells.

Authors:
Phornpun Phokrai Wan-Angkan Poolsri Somrudee Suwankulanan Narinthorn Phakdeeto Worasak Kaewkong Dumrongsak Pekthong Lysiane Richert Piyarat Srisawang

FEBS Open Bio 2018 Jun 14;8(6):986-1000. Epub 2018 May 14.

Department of Physiology Faculty of Medical Science Naresuan University Phitsanulok Thailand.

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June 2018

Epistructured catechins, EGCG and EC facilitate apoptosis induction through targeting de novo lipogenesis pathway in HepG2 cells.

Authors:
Phuriwat Khiewkamrop Pattamaphron Phunsomboon Lysiane Richert Dumrongsak Pekthong Piyarat Srisawang

Cancer Cell Int 2018 21;18:46. Epub 2018 Mar 21.

1Department of Physiology, Faculty of Medical Science, Naresuan University, Phitsanulok, 65000 Thailand.

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March 2018

Combination of Mitochondrial and Plasma Membrane Citrate Transporter Inhibitors Inhibits De Novo Lipogenesis Pathway and Triggers Apoptosis in Hepatocellular Carcinoma Cells.

Authors:
Wan-Angkan Poolsri Phornpun Phokrai Somrudee Suwankulanan Narinthorn Phakdeeto Pattamaphorn Phunsomboon Dumrongsak Pekthong Lysiane Richert Sutatip Pongcharoen Piyarat Srisawang

Biomed Res Int 2018 9;2018:3683026. Epub 2018 Jan 9.

Department of Physiology, Faculty of Medical Science, Naresuan University, Phitsanulok 65000, Thailand.

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August 2018

Immunochromatographic determination of bacopaside I in biological samples.

Authors:
Sontaya Sookying Dumrongsak Pekthong Sarawut Oo-Puthinan Watoo Phrompittayarat Waraporn Putalun Hiroyuki Tanaka Jie Xing Zhaoqi Zhan Nantaka Khorana Nitra Nuengchamnong Kornkanok Ingkaninan

J Chromatogr B Analyt Technol Biomed Life Sci 2017 Jan 23;1040:60-66. Epub 2016 Nov 23.

Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand. Electronic address:

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January 2017

[6]-Gingerol inhibits de novo fatty acid synthesis and carnitine palmitoyltransferase-1 activity which triggers apoptosis in HepG2.

Authors:
Hathaichanok Impheng Lysiane Richert Dumrongsak Pekthong C Norman Scholfield Sutatip Pongcharoen Ittipon Pungpetchara Piyarat Srisawang

Am J Cancer Res 2015 15;5(4):1319-36. Epub 2015 Mar 15.

Department of Physiology, Faculty of Medical Science, Naresuan University Phitsanulok, Thailand 65000.

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June 2015

Prediction of drug induced liver injury using molecular and biological descriptors.

Authors:
Christophe Muller Dumrongsak Pekthong Eliane Alexandre Gilles Marcou Dragos Horvath Lysiane Richert Alexandre Varnek

Comb Chem High Throughput Screen 2015 ;18(3):315-22

Laboratory of Chemoinformatics, University of Strasbourg, 1, rue B. Pascal, Strasbourg, 67000, France.

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October 2015

The selective target of capsaicin on FASN expression and de novo fatty acid synthesis mediated through ROS generation triggers apoptosis in HepG2 cells.

Authors:
Hathaichanok Impheng Sutatip Pongcharoen Lysiane Richert Dumrongsak Pekthong Piyarat Srisawang

PLoS One 2014 25;9(9):e107842. Epub 2014 Sep 25.

Department of Physiology, Faculty of Medical Science, Naresuan University, Phitsanulok, Thailand.

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June 2015

Plateable cryopreserved human hepatocytes for the assessment of cytochrome P450 inducibility: experimental condition-related variables affecting their response to inducers.

Authors:
Eliane Alexandre Audrey Baze Céline Parmentier Coraline Desbans Dumrongsak Pekthong Brigitte Gerin Claudine Wack Philippe Bachellier Bruno Heyd Jean-Christophe Weber Lysiane Richert

Xenobiotica 2012 Oct 19;42(10):968-79. Epub 2012 Apr 19.

KaLy-Cell, 20A rue du Général Leclerc, Plobsheim, France.

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October 2012

Bupropion hydroxylation as a selective marker of rat CYP2B1 catalytic activity.

Authors:
Dumrongsak Pekthong Coraline Desbans Hélène Martin Lysiane Richert

Drug Metab Dispos 2012 Jan 30;40(1):32-8. Epub 2011 Sep 30.

KaLy-Cell, Bioparc, Boulevard Sébastien Brant, 67400 Illkirch Cedex, France.

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January 2012

Follow-up to the pre-validation of a harmonised protocol for assessment of CYP induction responses in freshly isolated and cryopreserved human hepatocytes with respect to culture format, treatment, positive reference inducers and incubation conditions.

Authors:
Catherine Abadie-Viollon Hélène Martin Nadège Blanchard Dumrongsak Pekthong Philippe Bachellier Georges Mantion Bruno Heyd Frantz Schuler Philippe Coassolo Eliane Alexandre Lysiane Richert

Toxicol In Vitro 2010 Feb 2;24(1):346-56. Epub 2009 Jun 2.

KaLy-Cell, Bioparc, Boulevard Sébastien Brant, Illkirch, France.

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February 2010

Effects of Andrographis paniculata extract and Andrographolide on hepatic cytochrome P450 mRNA expression and monooxygenase activities after in vivo administration to rats and in vitro in rat and human hepatocyte cultures.

Authors:
Dumrongsak Pekthong Nadège Blanchard Catherine Abadie Alexandre Bonet Bruno Heyd Georges Mantion Alain Berthelot Lysiane Richert Hélène Martin

Chem Biol Interact 2009 May 8;179(2-3):247-55. Epub 2008 Nov 8.

Laboratoire de Toxicologie Cellulaire, EA 4267, IFR 133, UFR Pharmacie, Place Saint-Jacques, 25030 Besançon, France.

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May 2009