Publications by authors named "Dominique Schols"

255Publications

Palladium-catalyzed cross-coupling reactions on a bromo-naphthalene scaffold in the search for novel human CC chemokine receptor 8 (CCR8) antagonists.

Bioorg Chem 2020 Dec 16;107:104560. Epub 2020 Dec 16.

KU Leuven, Department of Microbiology, Immunology and Transplantation, Rega Institute for Medical Research, Laboratory of Virology and Chemotherapy, Herestraat 49, box 1043, 3000 Leuven, Belgium. Electronic address:

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December 2020

Characterization of the Carbohydrate-Binding Agents HHA, GNA and UDA as Inhibitors of Influenza a and B Virus Replication.

Antimicrob Agents Chemother 2020 Dec 7. Epub 2020 Dec 7.

KU Leuven, Rega Institute for Medical Research, Laboratory of Virology and Chemotherapy, Leuven, Belgium.

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December 2020

Synthesis, Molecular Docking and Preliminary Antileukemic Activity of 4-Methoxybenzyl Derivatives Bearing Imidazo[2,1-b][1,3,4]thiadiazole.

Chem Biodivers 2020 Dec 4. Epub 2020 Dec 4.

Department of Pharmaceutical Chemistry, KLE College of Pharmacy (A Constituent Unit of KAHER-Belagavi), Bengaluru, 560010, Karnataka, India.

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December 2020

γ-Ketobenzyl-Modified Nucleoside Triphosphate Prodrugs as Potential Antivirals.

J Med Chem 2020 11 13;63(22):13745-13761. Epub 2020 Nov 13.

Organic Chemistry, Department of Chemistry, Faculty of Mathematics, Informatics and Natural Sciences, Universität Hamburg, Martin-Luther-King-Platz 6, D-20146 Hamburg, Germany.

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November 2020

Development of a Novel SPR Assay to Study CXCR4-Ligand Interactions.

Biosensors (Basel) 2020 Oct 21;10(10). Epub 2020 Oct 21.

Laboratory of Virology and Chemotherapy, Department of Microbiology, Immunology and Transplantation, Rega Institute, KU Leuven, Herestraat 49, P.O. Box 1030, 3000 Leuven, Belgium.

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October 2020

γ-Non-Symmetrically Dimasked TriPPPro Prodrugs as Potential Antiviral Agents against HIV.

ChemMedChem 2020 Oct 22. Epub 2020 Oct 22.

Organic Chemistry, Department of Chemistry, Faculty of Mathematics, Informatics and Natural Sciences, Universität Hamburg, Martin-Luther-King-Platz 6, 20146, Hamburg, Germany.

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October 2020

Thiophene-based water-soluble fullerene derivatives as highly potent antiherpetic pharmaceuticals.

Org Biomol Chem 2020 Nov;18(42):8702-8708

Skolkovo Institute of Science and Technology, Nobel St. 3, Moscow, 143026, Russia. and IPCP RAS, Semenov Prospect 1, Chernogolovka, 142432, Russia.

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November 2020

Itaconic acid hybrids as potential anticancer agents.

Mol Divers 2020 Oct 11. Epub 2020 Oct 11.

Department of Medicinal Chemistry, Faculty of Pharmacy and Biochemistry, University of Zagreb, 10 000, Zagreb, Croatia.

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October 2020

Membrane Permeable, Bioreversibly Modified Prodrugs of Nucleoside Diphosphate-γ-Phosphonates.

J Med Chem 2020 10 14;63(20):11990-12007. Epub 2020 Oct 14.

Organic Chemistry, Department of Chemistry, Faculty of Mathematics, Informatics and Natural Sciences, Universität Hamburg, Martin-Luther-King-Platz 6, D-20146 Hamburg, Germany.

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October 2020

Synthesis of new riboflavin modified ODNs: Effect of riboflavin moiety on the G-quadruplex arrangement and stability.

Bioorg Chem 2020 11 1;104:104213. Epub 2020 Sep 1.

Department of Chemical Sciences, University of Napoli Federico II, Complesso di Monte Sant'Angelo, Via Cintia 4, I-80126 Napoli, Italy. Electronic address:

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November 2020

Discovery of HIV entry inhibitors via a hybrid CXCR4 and CCR5 receptor pharmacophore-based virtual screening approach.

Eur J Pharm Sci 2020 Dec 2;155:105537. Epub 2020 Sep 2.

Medicinal Chemistry, Department of Pharmaceutical and Pharmacological Sciences, Rega Institute for Medical Research, KU Leuven, B-3000 Leuven, Belgium. Electronic address:

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December 2020

Synthesis, Molecular Docking and Molecular Dynamics Simulation of 2-thioxothiazolidin-4-one derivatives against Gp41.

Curr HIV Res 2020 Sep 3. Epub 2020 Sep 3.

Department of Medicinal Chemistry, School of Pharmacy and Pharmaceutical Sciences, Isfahan University of Medical Sciences, Isfahan. Iran.

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September 2020

Water-soluble fullerene-based nanostructures with promising antiviral and myogenic activity.

Chem Commun (Camb) 2020 Sep;56(70):10203-10206

Skolkovo Institute of Science and Technology, Nobel St. 3, Moscow, 143026, Russia. and IPCP RAS, Semenov Prospect 1, Chernogolovka, 142432, Russia.

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September 2020

Lipophilic Triphosphate Prodrugs of Various Nucleoside Analogues.

J Med Chem 2020 07 29;63(13):6991-7007. Epub 2020 Jun 29.

Organic Chemistry, Department of Chemistry, Faculty of Mathematics, Informatics and Natural Sciences, Universität Hamburg, Martin-Luther-King-Platz 6, D-20146 Hamburg, Germany.

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July 2020

Anti-HIV-Active Nucleoside Triphosphate Prodrugs.

J Med Chem 2020 06 3;63(11):6003-6027. Epub 2020 Jun 3.

Organic Chemistry, Department of Chemistry, Faculty of Mathematics, Informatics and Natural Sciences, Universität Hamburg, Martin-Luther-King-Platz 6, D-20146 Hamburg, Germany.

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June 2020