Publications by authors named "Daniel Wyss"

39Publications

NMR Binding and Functional Assays for Detecting Inhibitors of S. aureus MnaA.

J Biomol Screen 2016 Jul 29;21(6):579-89. Epub 2016 Mar 29.

Structural Chemistry, Merck Research Laboratories, Kenilworth, NJ, USA

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July 2016

NMR screening in fragment-based drug design: a practical guide.

Methods Mol Biol 2015 ;1263:197-208

Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ, 07033, USA,

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September 2015

Effective progression of nuclear magnetic resonance-detected fragment hits.

Methods Enzymol 2011 ;493:447-68

Global Structural Chemistry, Merck Research Laboratories, Kenilworth, New Jersey, USA.

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June 2011

Pyridine Carboxamides: Potent Palm Site Inhibitors of HCV NS5B Polymerase.

ACS Med Chem Lett 2010 Dec 17;1(9):466-71. Epub 2010 Aug 17.

Department of Infectious Diseases, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033.

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December 2010

Pharmacological characterisation of anti-inflammatory compounds in acute and chronic mouse models of cigarette smoke-induced inflammation.

Respir Res 2010 Sep 18;11:126. Epub 2010 Sep 18.

Respiratory Disease Area, Novartis Institutes for BioMedical Research, Wimblehurst Road, Horsham RH12 5AB, UK.

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September 2010

Characterization of autocatalytic conversion of precursor BACE1 by heteronuclear NMR spectroscopy.

Biochemistry 2005 Dec;44(50):16594-601

Schering-Plough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033, USA.

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December 2005

Effect of adenosine A2A receptor activation in murine models of respiratory disorders.

Am J Physiol Lung Cell Mol Physiol 2006 May 9;290(5):L1036-43. Epub 2005 Dec 9.

Respiratory Diseases Area, Novartis Institutes for BioMedical Research, Horsham, England, UK.

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May 2006

Screening of protein kinases by ATP-STD NMR spectroscopy.

J Am Chem Soc 2005 Jun;127(22):7978-9

Schering-Plough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033, USA.

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June 2005

Mast cell involvement in the adenosine mediated airway hyper-reactivity in a murine model of ovalbumin-induced lung inflammation.

Br J Pharmacol 2005 Aug;145(7):845-52

Novartis Institutes for BioMedical Research, Respiratory Diseases Area, Horsham RH12 5AB, UK.

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August 2005