Publications by authors named "Dale F Mierke"

78Publications

The IKK-binding domain of NEMO is an irregular coiled coil with a dynamic binding interface.

Sci Rep 2019 02 27;9(1):2950. Epub 2019 Feb 27.

Department of Chemistry, Dartmouth College, Hanover, NH, 03755, USA.

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http://dx.doi.org/10.1038/s41598-019-39588-2DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6393490PMC
February 2019

New Monocyclic, Bicyclic, and Tricyclic Ethynylcyanodienones as Activators of the Keap1/Nrf2/ARE Pathway and Inhibitors of Inducible Nitric Oxide Synthase.

J Med Chem 2015 Jun 20;58(11):4738-48. Epub 2015 May 20.

†Institute of Chemical Biology and Drug Discovery, Stony Brook University, Stony Brook, New York 11794, United States.

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http://dx.doi.org/10.1021/acs.jmedchem.5b00393DOI Listing
June 2015

A novel caspase 8 selective small molecule potentiates TRAIL-induced cell death.

Sci Rep 2015 May 11;5:9893. Epub 2015 May 11.

1] Department of Pathology, Beth Israel Deaconess Medical Center and Harvard Medical School, Boston, MA, USA [2] Department of Biological and Biomedical Sciences Program, Harvard Medical School, Boston, MA, USA.

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http://dx.doi.org/10.1038/srep09893DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4426715PMC
May 2015

Modulating the dysregulated migration of pulmonary arterial hypertensive smooth muscle cells with motif mimicking cell permeable peptides.

Curr Top Pept Protein Res 2015;16:1-17

Tupper Research Institute and Pulmonary, Critical Care, and Sleep Division, Tufts Medical Center, Boston, Massachusetts 02111, USA.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4888800PMC
January 2015

Small-molecule inhibitors of JC polyomavirus infection.

J Pept Sci 2015 Mar 19;21(3):236-42. Epub 2014 Dec 19.

Department of Chemistry, Dartmouth College, Hanover, NH, 03755, USA.

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http://doi.wiley.com/10.1002/psc.2731
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http://dx.doi.org/10.1002/psc.2731DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4478595PMC
March 2015

Computational design of selective peptides to discriminate between similar PDZ domains in an oncogenic pathway.

J Mol Biol 2015 Jan 30;427(2):491-510. Epub 2014 Oct 30.

Department of Biological Sciences, Dartmouth College, Hanover, NH 03755, USA; Department of Computer Science, Dartmouth College, Hanover, NH 03755, USA. Electronic address:

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http://dx.doi.org/10.1016/j.jmb.2014.10.014DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4970318PMC
January 2015

Protein engineering of the N-terminus of NEMO: structure stabilization and rescue of IKKβ binding.

Biochemistry 2014 Nov 23;53(43):6776-85. Epub 2014 Oct 23.

Department of Chemistry, Dartmouth College , Hanover, New Hampshire 03755, United States.

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http://dx.doi.org/10.1021/bi500861xDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4222529PMC
November 2014

Small molecule inhibition of the Na(+)/H(+) exchange regulatory factor 1 and parathyroid hormone 1 receptor interaction.

Biochemistry 2014 Sep 15;53(37):5916-22. Epub 2014 Sep 15.

Department of Chemistry and Department of Molecular and Cellular Biology, Dartmouth College , Hanover, New Hampshire 03755, United States.

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http://dx.doi.org/10.1021/bi500368kDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4172209PMC
September 2014

Monitoring ATP hydrolysis and ATPase inhibitor screening using (1)H NMR.

Chem Commun (Camb) 2014 Oct;50(81):12037-9

Department of Chemistry, Dartmouth College, Hanover 03755, USA.

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http://dx.doi.org/10.1039/c4cc04399eDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4262093PMC
October 2014

Gallic acid-based small-molecule inhibitors of JC and BK polyomaviral infection.

Virus Res 2014 Aug 21;189:280-5. Epub 2014 Jun 21.

Department of Molecular Biology, Cell Biology and Biochemistry, Brown University, Providence, RI 02912, United States. Electronic address:

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http://dx.doi.org/10.1016/j.virusres.2014.06.008DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4144447PMC
August 2014

Engineering a soluble parathyroid hormone GPCR mimetic.

Proteins 2014 Jul 15;82(7):1370-5. Epub 2014 Jan 15.

Department of Chemistry, Dartmouth College, Hanover, New Hampshire, 03755.

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http://dx.doi.org/10.1002/prot.24503DOI Listing
July 2014

Recombinant production of TEV cleaved human parathyroid hormone.

J Pept Sci 2013 Aug 23;19(8):504-10. Epub 2013 Jun 23.

Department of Chemistry, Dartmouth College, Hanover, New Hampshire 03755, USA.

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http://dx.doi.org/10.1002/psc.2528DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3755510PMC
August 2013

AUF1-RGG peptides up-regulate the VEGF antagonist, soluble VEGF receptor-1 (sFlt-1).

Cytokine 2013 Oct 14;64(1):337-42. Epub 2013 Jun 14.

Veterans Administration Research Service, White River Junction, VT 05009, USA; Department of Medicine, Geisel School of Medicine at Dartmouth, Hanover, NH 03755, USA.

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http://dx.doi.org/10.1016/j.cyto.2013.05.019DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3770750PMC
October 2013

Peptides modeled on the RGG domain of AUF1/hnRNP-D regulate 3' UTR-dependent gene expression.

Int Immunopharmacol 2013 Sep 5;17(1):132-41. Epub 2013 Jun 5.

Veterans Administration Research Service, White River Junction, VT 05009, USA.

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http://dx.doi.org/10.1016/j.intimp.2013.05.014DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3711235PMC
September 2013

C-terminus of ETA/ETB receptors regulate endothelin-1 signal transmission.

J Pept Sci 2013 Apr 25;19(4):257-62. Epub 2013 Feb 25.

Department of Chemistry, Dartmouth College, Hanover, NH 03755, USA.

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http://dx.doi.org/10.1002/psc.2499DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3770155PMC
April 2013

Ligand binding site identification by higher dimension molecular dynamics.

J Chem Inf Model 2013 Mar 20;53(3):674-80. Epub 2013 Feb 20.

Department of Chemistry, Dartmouth College , Hanover, New Hampshire 03755, United States.

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http://dx.doi.org/10.1021/ci300561bDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3706581PMC
March 2013

Hydrophobic residues in helix 8 of cannabinoid receptor 1 are critical for structural and functional properties.

Biochemistry 2010 Jan;49(3):502-11

Department of Molecular and Cell Biology, University of Connecticut, Storrs, Connecticut 06269, USA.

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http://dx.doi.org/10.1021/bi901619rDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2904477PMC
January 2010

Dual role of the second extracellular loop of the cannabinoid receptor 1: ligand binding and receptor localization.

Mol Pharmacol 2009 Oct 30;76(4):833-42. Epub 2009 Jul 30.

Department of Molecular and Cell Biology, University of Connecticut, Storrs, CT 06269-3125, USA.

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http://dx.doi.org/10.1124/mol.109.057356DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2769047PMC
October 2009

Structural analysis of the human cannabinoid receptor one carboxyl-terminus identifies two amphipathic helices.

Biopolymers 2009 Jul;91(7):565-73

Department of Molecular and Cell Biology, University of Connecticut, Storrs, CT 06269, USA.

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http://dx.doi.org/10.1002/bip.21179DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2698224PMC
July 2009

PTH and PTH antagonist induce different conformational changes in the PTHR1 receptor.

J Bone Miner Res 2009 May;24(5):925-34

Department of Physiology, Tufts University School of Medicine, Boston, Massachusetts, USA.

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http://dx.doi.org/10.1359/jbmr.081228DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2672208PMC
May 2009

Residue 17 of sauvagine cross-links to the first transmembrane domain of corticotropin-releasing factor receptor 1 (CRFR1).

J Biol Chem 2008 Dec 27;283(51):35644-51. Epub 2008 Oct 27.

Endocrine Division, Department of Internal Medicine, Wayne State University School of Medicine, University Health Center, Detroit, Mighigan 48201, USA.

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http://dx.doi.org/10.1074/jbc.M806351200DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2602896PMC
December 2008

Mapping peptide hormone-receptor interactions using a disulfide-trapping approach.

Biochemistry 2008 Jun 7;47(22):5889-95. Epub 2008 May 7.

Department of Physiology, Tufts University School of Medicine, Boston, Massachusetts 02111, USA.

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http://pubs.acs.org/doi/abs/10.1021/bi800122f
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http://dx.doi.org/10.1021/bi800122fDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2570702PMC
June 2008

Conformational changes in the parathyroid hormone receptor associated with activation by agonist.

Mol Endocrinol 2008 May 7;22(5):1154-62. Epub 2008 Feb 7.

Department of Physiology, Tufts University School of Medicine, Boston, Massachusetts 02111, USA.

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https://academic.oup.com/mend/article-lookup/doi/10.1210/me.
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http://dx.doi.org/10.1210/me.2007-0520DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2366190PMC
May 2008

Conformational preference and potential templates of N-methylated cyclic pentaalanine peptides.

Chemistry 2008 ;14(5):1508-17

Center for Integrated Protein Science at the Department Chemie, Lehrstuhl für Organische Chemie II, Technische Universität München, Lichtenbergstrasse 4, Garching, Germany.

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http://dx.doi.org/10.1002/chem.200701029DOI Listing
May 2008

Further evidence for a C-terminal structural motif in CCK2 receptor active peptide hormones.

Peptides 2007 Nov 22;28(11):2211-22. Epub 2007 Sep 22.

Department of Chemistry, University of Cape Town, Rondebosch 7701, Cape Town, South Africa.

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http://dx.doi.org/10.1016/j.peptides.2007.09.008DOI Listing
November 2007

Evidence for a C-terminal structural motif in gastrin and its bioactive fragments in membrane mimetic media.

Peptides 2007 Aug 17;28(8):1561-71. Epub 2007 Jul 17.

Department of Chemistry, University of Cape Town, Private Bag, Rondebosch 7701, Cape Town, South Africa.

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http://dx.doi.org/10.1016/j.peptides.2007.07.009DOI Listing
August 2007

Identification of amino acid residues in BK virus VP1 that are critical for viability and growth.

J Virol 2007 Nov 15;81(21):11798-808. Epub 2007 Aug 15.

Department of Molecular Biology, Cell Biology and Biochemistry, Brown University, 70 Ship Street, Providence, RI 02903, USA.

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http://dx.doi.org/10.1128/JVI.01316-07DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2168807PMC
November 2007

Architecture of the 99 bp DNA-six-protein regulatory complex of the lambda att site.

Mol Cell 2006 Nov;24(4):569-80

Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1016/j.molcel.2006.10.006DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1866956PMC
November 2006

The conformation of cyclo(-D-Pro-Ala4-) as a model for cyclic pentapeptides of the DL4 type.

J Am Chem Soc 2006 Oct;128(42):13806-14

Department Chemie, Technische Universität München, Lichtenbergstrasse 4, 85747 Garching, Germany.

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http://dx.doi.org/10.1021/ja063174aDOI Listing
October 2006

Structural features of parathyroid hormone receptor coupled to Galpha(s)-protein.

Biophys J 2007 Jan 13;92(2):535-40. Epub 2006 Oct 13.

Department of Chemistry, and Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1529/biophysj.106.094813DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1751412PMC
January 2007

Targeting the PDZ domains of molecular scaffolds of transmembrane ion channels.

AAPS J 2006 Jun 2;8(2):E396-401. Epub 2006 Jun 2.

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, 171 Meeting Street, Providence, RI 02912, USA.

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http://www.aapsj.org/view.asp?art=aapsj080245
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http://dx.doi.org/10.1007/BF02854911DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3231575PMC
June 2006

The role of sialic acid in human polyomavirus infections.

Glycoconj J 2006 Feb;23(1-2):19-26

Department of Molecular Biology, Cell Biology and Biochemistry, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1007/s10719-006-5434-zDOI Listing
February 2006

Methionine acts as a "magnet" in photoaffinity crosslinking experiments.

FEBS Lett 2006 Mar 28;580(7):1872-6. Epub 2006 Feb 28.

Department of Physiology, Tufts University School of Medicine, 136 Harrison Ave, M&V 7, Boston, MA 02111, USA.

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http://doi.wiley.com/10.1016/j.febslet.2006.02.050
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http://dx.doi.org/10.1016/j.febslet.2006.02.050DOI Listing
March 2006

The mid-region of parathyroid hormone (1-34) serves as a functional docking domain in receptor activation.

Biochemistry 2006 Feb;45(7):2027-34

Department of Physiology, Tufts University School of Medicine, 136 Harrison Avenue, Boston, Massachusetts 02111, USA.

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http://pubs.acs.org/doi/abs/10.1021/bi051833a
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http://dx.doi.org/10.1021/bi051833aDOI Listing
February 2006

Association of the cystic fibrosis transmembrane regulator with CAL: structural features and molecular dynamics.

Biochemistry 2005 Dec;44(49):16158-66

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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https://pubs.acs.org/doi/10.1021/bi0516475
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http://dx.doi.org/10.1021/bi0516475DOI Listing
December 2005

Defining the retinoid binding site in the rod cyclic nucleotide-gated channel.

J Gen Physiol 2005 Nov 17;126(5):453-60. Epub 2005 Oct 17.

Department of Molecular Pharmacology, Physiology, and Biotechnology, Brown Medical School, Providence, RI 02912, USA.

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http://dx.doi.org/10.1085/jgp.200509387DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2266610PMC
November 2005

Structural characterization of the intermolecular interactions of synapse-associated protein-97 with the NR2B subunit of N-methyl-D-aspartate receptors.

J Biol Chem 2005 Jul 1;280(29):26992-6. Epub 2005 Jun 1.

Department of Physics, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://www.jbc.org/lookup/doi/10.1074/jbc.M503555200
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http://dx.doi.org/10.1074/jbc.M503555200DOI Listing
July 2005

Bradykinin B2 receptor signaling: structural and functional characterization of the C-terminus.

Biopolymers 2005 ;80(2-3):367-73

Department of Molecular Pharmacology, Division of Biology & Medicine, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1002/bip.20220DOI Listing
June 2005

Modeling a sialic acid binding pocket in the external loops of JC virus VP1.

J Biol Chem 2004 Nov 3;279(47):49172-6. Epub 2004 Sep 3.

Graduate Program in Molecular and Cell Biology and Biochemistry and Department of Molecular Microbiology and Immunology, Brown University, Providence, Rhode Island 02912, USA.

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http://www.jbc.org/lookup/doi/10.1074/jbc.M409326200
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http://dx.doi.org/10.1074/jbc.M409326200DOI Listing
November 2004

A steroid modulatory domain on NR2B controls N-methyl-D-aspartate receptor proton sensitivity.

Proc Natl Acad Sci U S A 2004 May 18;101(21):8198-203. Epub 2004 May 18.

Laboratory of Molecular Neurobiology, Department of Pharmacology, Boston University School of Medicine, 715 Albany Street, Boston, MA 02118, USA.

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http://dx.doi.org/10.1073/pnas.0401838101DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC419580PMC
May 2004

Targeting specific PDZ domains of PSD-95; structural basis for enhanced affinity and enzymatic stability of a cyclic peptide.

Chem Biol 2004 Apr;11(4):469-73

Department of Chemistry, Division of Biology & Medicine, Brown University, Providence, RI 02912 USA.

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http://linkinghub.elsevier.com/retrieve/pii/S107455210400089
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http://dx.doi.org/10.1016/j.chembiol.2004.03.013DOI Listing
April 2004

Cooperative interaction of arginine-19 and the N-terminal signaling domain in the affinity and potency of parathyroid hormone.

Biochemistry 2004 Mar;43(12):3459-70

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi036127tDOI Listing
March 2004

Conformational and molecular modeling studies of beta-cyclodextrin-heptagastrin and the third extracellular loop of the cholecystokinin 2 receptor.

Biochemistry 2004 Mar;43(10):2724-31

Department of Chemistry, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi035509wDOI Listing
March 2004

Toward parathyroid hormone minimization: conformational studies of cyclic PTH(1-14) analogues.

Biochemistry 2004 Jan;43(3):690-9

Department of Molecular Pharmacology, Division of Biology & Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi035703iDOI Listing
January 2004

Intermolecular interactions between peptidic and nonpeptidic agonists and the third extracellular loop of the cholecystokinin 1 receptor.

J Med Chem 2003 Jul;46(16):3476-82

Department of Chemistry, Division of Biology & Medicine, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1021/jm030144zDOI Listing
July 2003

Determination of ligand-receptor interactions of cholecystokinin by nuclear magnetic resonance.

Life Sci 2003 Jun;73(6):705-13

Department of Chemistry, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1016/s0024-3205(03)00391-6DOI Listing
June 2003

Extracellular domains of the neurokinin-1 receptor: structural characterization and interactions with substance P.

Biopolymers 2002 ;66(5):339-49

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, RI 02912, USA.

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http://doi.wiley.com/10.1002/bip.10312
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http://dx.doi.org/10.1002/bip.10312DOI Listing
March 2003

Residue 19 of the parathyroid hormone: structural consequences.

Biochemistry 2002 Nov;41(44):13217-23

Department of Chemistry, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi0261600DOI Listing
November 2002

Mechanisms regulating the expression, self-maintenance, and signaling-function of the bradykinin B2 and B1 receptors.

J Cell Physiol 2002 Dec;193(3):275-86

Department of Biochemistry, Boston University School of Medicine, Boston, Massachusetts 02118, USA.

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http://dx.doi.org/10.1002/jcp.10175DOI Listing
December 2002

Cannabinoid receptor-G protein interactions: G(alphai1)-bound structures of IC3 and a mutant with altered G protein specificity.

Protein Sci 2002 Oct;11(10):2526-31

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2373710PMC
http://dx.doi.org/10.1110/ps.0218402DOI Listing
October 2002

Structure of the third intracellular loop of the human cannabinoid 1 receptor.

Biochemistry 2002 Sep;41(38):11344-50

Department of Molecular Pharmacology, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi0259610DOI Listing
September 2002

Ni-to-Ni+ 3-ethylene-bridged partially modified retro-inverso tetrapeptide beta-turn mimetic: design, synthesis, and structural characterization.

J Org Chem 2002 Jul;67(15):5085-97

Department of Medicine, Bone and Mineral Metabolism Unit, Charles A. Dana and Thorndike Laboratories, Beth Israel Deaconess Medical Center-Harvard Medical School, Boston, Massachusetts 02215, USA.

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http://dx.doi.org/10.1021/jo011041wDOI Listing
July 2002

Selective ligand-induced stabilization of active and desensitized parathyroid hormone type 1 receptor conformations.

J Biol Chem 2002 Oct 9;277(41):38524-30. Epub 2002 Jul 9.

Department of Medicine, Division of Endocrinology and Metabolism, University of Pittsburgh School of Medicine, Pittsburgh, Pennsylvania 15261, USA.

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http://www.jbc.org/lookup/doi/10.1074/jbc.M202544200
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http://dx.doi.org/10.1074/jbc.M202544200DOI Listing
October 2002

Identification of the principal binding site for RGD-containing ligands in the alpha(V)beta(3) integrin: a photoaffinity cross-linking study.

Biochemistry 2002 Jul;41(26):8321-31

Bone and Mineral Metabolism Unit, Charles A. Dana and Thorndike Laboratories, Department of Medicine, Beth Israel Deaconess Medical Center and Harvard Medical School, 330 Brookline Avenue, Boston, Massachusetts 02215, USA.

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http://dx.doi.org/10.1021/bi025690tDOI Listing
July 2002

NMR studies of CCK-8/CCK1 complex support membrane-associated pathway for ligand-receptor interaction.

Can J Physiol Pharmacol 2002 May;80(5):383-7

Department of Chemistry, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1139/y02-031DOI Listing
May 2002

Conformational and molecular modeling studies of sulfated cholecystokinin-15.

Biochem Biophys Res Commun 2002 May;293(3):1053-9

Department of Chemistry, Division of Biology & Medicine, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1016/S0006-291X(02)00334-0DOI Listing
May 2002

Structural characterization of a cyclic dipeptidomimetic: the effect of ring size on a 1,2,5-trisubstituted-3-oxo-1,4-diazepine system.

Biopolymers 2002 Jun;64(1):16-25

Department of Chemistry, Brown University, Providence, RI 02912, USA.

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http://doi.wiley.com/10.1002/bip.10080
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http://dx.doi.org/10.1002/bip.10080DOI Listing
June 2002

Homologs of 1,2,5-hexahydro-3-one-1H-1,4-diazepine (DAP) as novel dipeptidomimetics and molecular scaffolds: efficient preparation of synthons.

Biopolymers 2002 Jun;64(1):1-15

Department of Medicine, Beth Israel Deaconess Medical Center, Harvard Medical School, 330 Brookline Avenue (HIM 944), Boston, MA 02215, USA.

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http://dx.doi.org/10.1002/bip.10079DOI Listing
June 2002

Intermolecular interactions between cholecystokinin-8 and the third extracellular loop of the cholecystokinin-2 receptor.

Biochemistry 2002 Apr;41(14):4560-6

Department of Chemistry, Division of Biology and Medicine, Brown University, Providence, Rhode Island 02912, USA.

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http://dx.doi.org/10.1021/bi0160009DOI Listing
April 2002

Molecular characterization of a ligand-tethered parathyroid hormone receptor.

Biophys Chem 2002 Feb;95(2):165-72

Department of Molecular Pharmacology, Division of Biology and Medicine, Box G-B4, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1016/s0301-4622(02)00005-4DOI Listing
February 2002

The PDZ1 domain of SAP90. Characterization of structure and binding.

J Biol Chem 2002 Mar 14;277(9):6967-73. Epub 2001 Dec 14.

Department of Chemistry, Division of Biology and Medicine, Brown University, Providence, RI 02912, USA.

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http://dx.doi.org/10.1074/jbc.M109453200DOI Listing
March 2002

Synthesis of a Trisubstituted 1,4-Diazepin-3-one-Based Dipeptidomimetic as a Novel Molecular Scaffold.

J Org Chem 1997 Apr;62(8):2527-2534

Department of Pharmaceutical Chemistry, School of Pharmacy, Faculty of Medicine, The Hebrew University of Jerusalem, Jerusalem 91120, Israel, Carlson School of Chemistry, Clark University, 950 Main Street, Worcester, Massachusetts 01610, and Division of Bone & Mineral Metabolism, Department of Medicine, Beth Israel Deaconess Medical Center, Harvard Medical School, 330 Brookline Avenue (HIM 944), Boston, Massachusetts 02215.

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http://dx.doi.org/10.1021/jo962257eDOI Listing
April 1997