Publications by authors named "Chahrazade El Amri"

26Publications

Insights into the activity control of the kallikrein-related peptidase 6: small-molecule modulators and allosterism.

Biol Chem 2018 09;399(9):1073-1078

Sorbonne University, Faculty of Sciences and Engineering, IBPS, UMR 8256 CNRS-UPMC, ERL INSERM U1164, Biological Adaptation and Ageing, F-75252 Paris, France.

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http://www.degruyter.com/view/j/bchm.2018.399.issue-9/hsz-20
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http://dx.doi.org/10.1515/hsz-2017-0336DOI Listing
September 2018

Piperlongumine and some of its analogs inhibit selectively the human immunoproteasome over the constitutive proteasome.

Biochem Biophys Res Commun 2018 02 2;496(3):961-966. Epub 2018 Feb 2.

Sorbonne Université, UPMC Univ Paris 06-CNRS, IBPS, UMR 8256, Inserm ERL1164, B2A, 7 Quai Saint Bernard, F75005 Paris, France. Electronic address:

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http://dx.doi.org/10.1016/j.bbrc.2018.01.100DOI Listing
February 2018

Serine protease inhibitors to treat inflammation: a patent review (2011-2016).

Expert Opin Ther Pat 2018 02 5;28(2):93-110. Epub 2017 Dec 5.

a B2A, Biological Adaptation and Ageing, Integrated Cellular Ageing and Inflammation, Molecular & Functional Enzymology , Sorbonne Universités , UPMC Univ Paris 06, UMR 8256 , Paris , France.

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http://dx.doi.org/10.1080/13543776.2018.1406478DOI Listing
February 2018

Phenoxypropanolamine derivatives as selective inhibitors of the 20S proteasome β1 and β5 subunits.

Bioorg Med Chem Lett 2017 12 23;27(23):5172-5178. Epub 2017 Oct 23.

Sorbonne Universités, UPMC Univ Paris 06, IBPS, CNRS UMR 8256, Biological Adaptation and Ageing (B2A), Integrated Cellular Ageing and Inflammation, 7 Quai St Bernard, 75005 Paris, France. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2017.10.055DOI Listing
December 2017

Inhibitors of kallikrein-related peptidases: An overview.

Med Res Rev 2018 03 13;38(2):655-683. Epub 2017 Jun 13.

Institut des Biomolécules Max Mousseron, UMR 5247, CNRS, Université de Montpellier, ENSCM, UFR des Sciences Pharmaceutiques et Biologiques, Montpellier Cedex, France.

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http://dx.doi.org/10.1002/med.21451DOI Listing
March 2018

Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.

Eur J Med Chem 2015 Mar 7;93:202-13. Epub 2015 Feb 7.

Sorbonne Universités, UPMC Univ Paris 06, UMR 8256, B2A, Biological Adaptation and Ageing, Integrated Cellular Ageing and Inflammation, Molecular & Functional Enzymology, 7 Quai St Bernard, F-75005 Paris, France. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S02235234150009
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http://dx.doi.org/10.1016/j.ejmech.2015.02.008DOI Listing
March 2015

Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7.

Eur J Med Chem 2015 Mar 7;93:202-13. Epub 2015 Feb 7.

Sorbonne Universités, UPMC Univ Paris 06, UMR 8256, B2A, Biological Adaptation and Ageing, Integrated Cellular Ageing and Inflammation, Molecular & Functional Enzymology, 7 Quai St Bernard, F-75005 Paris, France. Electronic address:

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https://linkinghub.elsevier.com/retrieve/pii/S02235234150009
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http://dx.doi.org/10.1016/j.ejmech.2015.02.008DOI Listing
March 2015

Investigating the role of GXXXG motifs in helical folding and self-association of plasticins, Gly/Leu-rich antimicrobial peptides.

Biophys Chem 2015 Jan 28;196:40-52. Epub 2014 Sep 28.

Sorbonne Universités, UPMC Univ Paris 06, Ecole Normale Supérieure-PSL Research University, Département de chimie, CNRS UMR 7203 Laboratoire des Biomolécules, 4 place Jussieu, F-75005 Paris, France. Electronic address:

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http://dx.doi.org/10.1016/j.bpc.2014.09.004DOI Listing
January 2015

Synthesis of {[5-(adenin-9-yl)-2-furyl]methoxy}methyl phosphonic acid and evaluations against human adenylate kinases.

Bioorg Med Chem Lett 2014 Sep 17;24(17):4227-30. Epub 2014 Jul 17.

Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 CNRS-UM 1-UM 2, cc 1705, Université Montpellier 2, Place Eugène Bataillon, 34095 Montpellier cedex 5, France.

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X140076
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http://dx.doi.org/10.1016/j.bmcl.2014.07.036DOI Listing
September 2014

Identification by in silico and in vitro screenings of small organic molecules acting as reversible inhibitors of kallikreins.

Eur J Med Chem 2013 22;70:661-8. Epub 2013 Oct 22.

Enzymologie Moléculaire et Fonctionnelle, UR4, Université Pierre et Marie Curie - Sorbonne Universités (UPMC), case courrier 256, 7, quai St Bernard, 75252 Paris Cedex 05, France.

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http://dx.doi.org/10.1016/j.ejmech.2013.10.040DOI Listing
September 2014

1,2,4-Triazole derivatives as transient inactivators of kallikreins involved in skin diseases.

Bioorg Med Chem Lett 2013 Aug 24;23(16):4547-51. Epub 2013 Jun 24.

Enzymologie Moléculaire et Fonctionnelle, UR4, Université Pierre et Marie Curie-Sorbonne Universités (UPMC), Case Courrier 256, 7, Quai St Bernard, 75252 Paris Cedex 05, France.

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http://dx.doi.org/10.1016/j.bmcl.2013.06.039DOI Listing
August 2013

Borononucleotides as substrates/binders for human NMP kinases: enzymatic and spectroscopic evaluation.

Chembiochem 2012 Jul 25;13(11):1605-12. Epub 2012 Jun 25.

Groupe d'Enzymologie Moléculaire et Fonctionnelle, UR4-UPMC, Université Pierre et Marie Curie, Sorbonne Universités, case courrier 256, 7, quai St Bernard, 75252 Paris Cedex 05, France.

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http://dx.doi.org/10.1002/cbic.201200199DOI Listing
July 2012

5',6'-nucleoside phosphonate analogues architecture: synthesis and comparative evaluation towards metabolic enzymes.

ChemMedChem 2011 Jun 12;6(6):1094-106. Epub 2011 May 12.

Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 CNRS-UM1&2, Université Montpellier 2, cc1705, Place E. Bataillon, 34095 Montpellier Cedex 5, France.

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http://dx.doi.org/10.1002/cmdc.201100068DOI Listing
June 2011

Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: structural and catalytic properties.

Antiviral Res 2010 Apr;86(1):101-20

Enzymologie Moléculaire et Fonctionnelle, UR4 Université Pierre et Marie Curie, 7 quai St Bernard, 75252 Paris Cedex 05, France.

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http://dx.doi.org/10.1016/j.antiviral.2010.02.001DOI Listing
April 2010

C-terminal domain of the Uup ATP-binding cassette ATPase is an essential folding domain that binds to DNA.

Biochim Biophys Acta 2010 Apr 27;1804(4):755-61. Epub 2009 Nov 27.

Unité des Membranes Bactériennes-CNRS URA2172, Département de Microbiologie, Institut Pasteur, 75724 Paris Cedex 15, France.

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http://dx.doi.org/10.1016/j.bbapap.2009.11.017DOI Listing
April 2010

Comparative study of two plasticins: specificity, interfacial behavior, and bactericidal activity.

Biochemistry 2009 Oct;48(40):9372-83

Universite Pierre et Marie Curie, ER3-Biogenese des signaux peptidiques, 75251 Paris Cedex 05, France.

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http://dx.doi.org/10.1021/bi901222pDOI Listing
October 2009

Lipid reorganization induced by membrane-active peptides probed using differential scanning calorimetry.

Biochim Biophys Acta 2009 Sep 7;1788(9):1772-81. Epub 2009 May 7.

UPMC Univ Paris 06, FRE 2852 Peptidome de la Peau d'Amphibiens, Paris F-75005, France.

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http://dx.doi.org/10.1016/j.bbamem.2009.05.001DOI Listing
September 2009

The dermaseptin superfamily: a gene-based combinatorial library of antimicrobial peptides.

Biochim Biophys Acta 2009 Aug 26;1788(8):1537-50. Epub 2008 Sep 26.

Equipe peptidome de la Peau des Amphibiens, FRE 2852 Université Pierre et Marie Curie - Paris 6, Tour 43, 2, Place Jussieu 75252 Paris cedex 05, France.

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http://dx.doi.org/10.1016/j.bbamem.2008.09.006DOI Listing
August 2009

Structural requirements for antimicrobial versus chemoattractant activities for dermaseptin S9.

FEBS J 2008 Aug 10;275(16):4134-51. Epub 2008 Jul 10.

UPMC Université de Paris 06, CNRS FRE 2852, Peptidome de la Peau des Amphibiens, Paris Cedex 5, France.

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http://dx.doi.org/10.1111/j.1742-4658.2008.06554.xDOI Listing
August 2008

The plasticins: membrane adsorption, lipid disorders, and biological activity.

Biochemistry 2006 Dec;45(48):14285-97

Peptidome de la Peau d'Amphibiens, FRE 2852, CNRS, Université Pierre et Marie Curie (Paris-6), Tour 43, 2 Place Jussieu, 75251 Paris Cedex 05, France.

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http://dx.doi.org/10.1021/bi060999oDOI Listing
December 2006

Assessment of adenyl residue reactivity within model nucleic acids by surface enhanced Raman spectroscopy.

Biopolymers 2006 May;82(1):6-28

Laboratoire de Dynamique Interactions et Réactivité, UMR 7075, Université Paris 6 CNRS, 2 rue Henri Dunant, 94320, Thiais, France.

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http://dx.doi.org/10.1002/bip.20455DOI Listing
May 2006

The micro-distribution of carbonaceous matter in the Murchison meteorite as investigated by Raman imaging.

Spectrochim Acta A Mol Biomol Spectrosc 2005 Jul;61(9):2049-56

Laboratoire de Bioactivation des Peptides, Institut Jacques-Monod, Université Paris VI, tour 43, 2, place Jussieu, Paris Cedex 75251, France.

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http://dx.doi.org/10.1016/j.saa.2004.08.005DOI Listing
July 2005

Adenine and RNA in mineral samples. Surface-enhanced Raman spectroscopy (SERS) for picomole detections.

Spectrochim Acta A Mol Biomol Spectrosc 2003 Sep;59(11):2645-54

Laboratoire de Biochimie de l'Evolution et Adaptabilité Moléculaire, Institut Jacques Monod, Université Paris-6, tour 43, 2, place Jussieu, 75251 Paris Cedex 05, France.

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http://dx.doi.org/10.1016/s1386-1425(03)00034-9DOI Listing
September 2003