Publications by authors named "Bruno Catalanotti"

34Publications

Hijacking SARS-CoV-2/ACE2 Receptor Interaction by Natural and Semi-synthetic Steroidal Agents Acting on Functional Pockets on the Receptor Binding Domain.

Authors:
Adriana Carino Federica Moraca Bianca Fiorillo Silvia Marchianò Valentina Sepe Michele Biagioli Claudia Finamore Silvia Bozza Daniela Francisci Eleonora Distrutti Bruno Catalanotti Angela Zampella Stefano Fiorucci

Front Chem 2020 23;8:572885. Epub 2020 Oct 23.

Department of Surgical and Biomedical Sciences, University of Perugia, Perugia, Italy.

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October 2020

Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen.

Authors:
Alessandro Deplano Jessica Karlsson Mona Svensson Federica Moraca Bruno Catalanotti Christopher J Fowler Valentina Onnis

J Enzyme Inhib Med Chem 2020 Dec;35(1):815-823

Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences, Department of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy.

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December 2020

Targeting multiple G-quadruplex-forming DNA sequences: Design, biophysical and biological evaluations of indolo-naphthyridine scaffold derivatives.

Authors:
Raffaella Catalano Federica Moraca Jussara Amato Camilla Cristofari Riccardo Rigo Lisa Dalla Via Roberta Rocca Antonio Lupia Annalisa Maruca Giosuè Costa Bruno Catalanotti Anna Artese Bruno Pagano Antonio Randazzo Claudia Sissi Ettore Novellino Stefano Alcaro

Eur J Med Chem 2019 Nov 16;182:111627. Epub 2019 Aug 16.

Dipartimento di Scienze della Salute, Università "Magna Græcia", Campus Salvatore Venuta, Viale Europa, 88100, Catanzaro, Italy; Net4Science srl, Università "Magna Græcia", Campus Salvatore Venuta, Viale Europa, 88100, Catanzaro, Italy.

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November 2019

Feedback inhibition of cAMP effector signaling by a chaperone-assisted ubiquitin system.

Authors:
Laura Rinaldi Rossella Delle Donne Bruno Catalanotti Omar Torres-Quesada Florian Enzler Federica Moraca Robert Nisticò Francesco Chiuso Sonia Piccinin Verena Bachmann Herbert H Lindner Corrado Garbi Antonella Scorziello Nicola Antonino Russo Matthis Synofzik Ulrich Stelzl Lucio Annunziato Eduard Stefan Antonio Feliciello

Nat Commun 2019 06 12;10(1):2572. Epub 2019 Jun 12.

Department of Molecular Medicine and Medical Biotechnologies, University Federico II, 80131, Naples, Italy.

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June 2019

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors.

Authors:
Alessandro Deplano Mariateresa Cipriano Federica Moraca Ettore Novellino Bruno Catalanotti Christopher J Fowler Valentina Onnis

J Enzyme Inhib Med Chem 2019 Dec;34(1):562-576

a Department of Life and Environmental Sciences - Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences , University of Cagliari , Cagliari , Italy.

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December 2019

Synthesis and Biological Evaluation of a New Structural Simplified Analogue of cADPR, a Calcium-Mobilizing Secondary Messenger Firstly Isolated from Sea Urchin Eggs.

Authors:
Stefano D'Errico Nicola Borbone Bruno Catalanotti Agnese Secondo Tiziana Petrozziello Ilaria Piccialli Anna Pannaccione Valeria Costantino Luciano Mayol Gennaro Piccialli Giorgia Oliviero

Mar Drugs 2018 Mar 10;16(3). Epub 2018 Mar 10.

SYSBIO, Centre of Systems Biology, University of Milano-Bicocca, Piazza della Scienza 2, 20126 Milano, Italy.

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March 2018

Peptide Nucleic Acids as miRNA Target Protectors for the Treatment of Cystic Fibrosis.

Authors:
Federica Zarrilli Felice Amato Carmine Marco Morgillo Brunella Pinto Giuliano Santarpia Nicola Borbone Stefano D'Errico Bruno Catalanotti Gennaro Piccialli Giuseppe Castaldo Giorgia Oliviero

Molecules 2017 Jul 8;22(7). Epub 2017 Jul 8.

Department of Molecular Medicine and Medical Biotechnologies, University of Naples Federico II, 80131 Napoli, Italy.

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July 2017

Novel propanamides as fatty acid amide hydrolase inhibitors.

Authors:
Alessandro Deplano Carmine Marco Morgillo Monica Demurtas Emmelie Björklund Mariateresa Cipriano Mona Svensson Sanaz Hashemian Giovanni Smaldone Emilia Pedone F Javier Luque Maria G Cabiddu Ettore Novellino Christopher J Fowler Bruno Catalanotti Valentina Onnis

Eur J Med Chem 2017 Aug 12;136:523-542. Epub 2017 May 12.

Department of Life and Environmental Sciences, Unit of Pharmaceutical, Pharmacological and Nutraceutical Sciences, University of Cagliari, via Ospedale 72, Cagliari I-09124, Italy.

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August 2017

Hyodeoxycholic acid derivatives as liver X receptor α and G-protein-coupled bile acid receptor agonists.

Authors:
Simona De Marino Adriana Carino Dario Masullo Claudia Finamore Silvia Marchianò Sabrina Cipriani Francesco Saverio Di Leva Bruno Catalanotti Ettore Novellino Vittorio Limongelli Stefano Fiorucci Angela Zampella

Sci Rep 2017 02 24;7:43290. Epub 2017 Feb 24.

Department of Pharmacy, University of Naples "Federico II", Via D. Montesano, 49, I-80131 Naples, Italy.

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February 2017

Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode.

Authors:
Jessica Karlsson Carmine M Morgillo Alessandro Deplano Giovanni Smaldone Emilia Pedone F Javier Luque Mona Svensson Ettore Novellino Cenzo Congiu Valentina Onnis Bruno Catalanotti Christopher J Fowler

PLoS One 2015 13;10(11):e0142711. Epub 2015 Nov 13.

Department of Pharmacology and Clinical Neuroscience, Pharmacology Unit, Umeå University, Umeå, Sweden.

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June 2016

Structural model of the hUbA1-UbcH10 quaternary complex: in silico and experimental analysis of the protein-protein interactions between E1, E2 and ubiquitin.

Authors:
Stefania Correale Ivan de Paola Carmine Marco Morgillo Antonella Federico Laura Zaccaro Pierlorenzo Pallante Aldo Galeone Alfredo Fusco Emilia Pedone F Javier Luque Bruno Catalanotti

PLoS One 2014 6;9(11):e112082. Epub 2014 Nov 6.

Dipartimento di Farmacia, Università degli Studi di Napoli Federico II, Napoli, Italy.

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July 2015

Exploitation of a very small peptide nucleic acid as a new inhibitor of miR-509-3p involved in the regulation of cystic fibrosis disease-gene expression.

Authors:
Felice Amato Rossella Tomaiuolo Fabrizia Nici Nicola Borbone Ausilia Elce Bruno Catalanotti Stefano D'Errico Carmine Marco Morgillo Giuseppe De Rosa Laura Mayol Gennaro Piccialli Giorgia Oliviero Giuseppe Castaldo

Biomed Res Int 2014 15;2014:610718. Epub 2014 Apr 15.

Dipartimento di Medicina Molecolare e Biotecnologie Mediche, Via Pansini 5, 80131 Napoli, Italy ; CEINGE-Biotecnologie Avanzate, 80131 Napoli, Italy.

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December 2014

Insight into the mechanism of action of plakortins, simple 1,2-dioxane antimalarials.

Authors:
Orazio Taglialatela-Scafati Ernesto Fattorusso Adriana Romano Fernando Scala Vincenzo Barone Paola Cimino Emiliano Stendardo Bruno Catalanotti Marco Persico Caterina Fattorusso

Org Biomol Chem 2010 Feb 16;8(4):846-56. Epub 2009 Dec 16.

Dipartimento di Chimica delle Sostanze Naturali, Università di Napoli Federico II, Via D. Montesano 49, I-80131 Napoli, Italy.

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February 2010

Full relative stereochemistry assignment and conformational analysis of 13,19-didesmethyl spirolide C via NMR- and molecular modeling-based techniques. A step towards understanding spirolide's mechanism of action.

Authors:
Patrizia Ciminiello Bruno Catalanotti Carmela Dell'aversano Caterina Fattorusso Ernesto Fattorusso Martino Forino Laura Grauso Angela Leo Luciana Tartaglione

Org Biomol Chem 2009 Sep 16;7(18):3674-81. Epub 2009 Jul 16.

Dipartimento di Chimica delle Sostanze Naturali, Università di Napoli Federico II, via D. Montesano, 49, 80131 Napoli, Italy.

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September 2009

Specific targeting of peripheral serotonin 5-HT(3) receptors. Synthesis, biological investigation, and structure-activity relationships.

Authors:
Elena Morelli Sandra Gemma Roberta Budriesi Giuseppe Campiani Ettore Novellino Caterina Fattorusso Bruno Catalanotti Salvatore Sanna Coccone Sindu Ros Giuseppe Borrelli Marco Persico Isabella Fiorini Vito Nacci Pierfranco Ioan Alberto Chiarini Michel Hamon Alfredo Cagnotto Tiziana Mennini Claudia Fracasso Milena Colovic Silvio Caccia Stefania Butini

J Med Chem 2009 Jun;52(11):3548-62

European Research Centre for Drug Discovery and Development, Siena, Italy.

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June 2009

Exploiting protein fluctuations at the active-site gorge of human cholinesterases: further optimization of the design strategy to develop extremely potent inhibitors.

Authors:
Stefania Butini Giuseppe Campiani Marianna Borriello Sandra Gemma Alessandro Panico Marco Persico Bruno Catalanotti Sindu Ros Margherita Brindisi Marianna Agnusdei Isabella Fiorini Vito Nacci Ettore Novellino Tatyana Belinskaya Ashima Saxena Caterina Fattorusso

J Med Chem 2008 Jun 15;51(11):3154-70. Epub 2008 May 15.

European Research Centre for Drug Discovery and Development (NatSynDrugs), Università di Siena, Siena, Italy.

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June 2008

Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling.

Authors:
Sandra Gemma Gagan Kukreja Giuseppe Campiani Stefania Butini Matteo Bernetti Bhupendra P Joshi Luisa Savini Nicoletta Basilico Donatella Taramelli Vanessa Yardley Alessia Bertamino Ettore Novellino Marco Persico Bruno Catalanotti Caterina Fattorusso

Bioorg Med Chem Lett 2007 Jul 29;17(13):3535-9. Epub 2007 Apr 29.

European Research Centre for Drug Discovery & Development, Università di Siena, via Aldo Moro, 53100 Siena, Italy.

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July 2007

Design and synthesis of potent antimalarial agents based on clotrimazole scaffold: exploring an innovative pharmacophore.

Authors:
Sandra Gemma Giuseppe Campiani Stefania Butini Gagan Kukreja Bhupendra P Joshi Marco Persico Bruno Catalanotti Ettore Novellino Ernesto Fattorusso Vito Nacci Luisa Savini Donatella Taramelli Nicoletta Basilico Giulia Morace Vanessa Yardley Caterina Fattorusso

J Med Chem 2007 Feb 31;50(4):595-8. Epub 2007 Jan 31.

Dipartimento Farmaco Chimico Tecnologico and European Research Centre for Drug Discovery and Development, Universita' di Siena, via Aldo Moro, 53100 Siena, Italy.

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February 2007

Endoperoxide derivatives from marine organisms: 1,2-dioxanes of the plakortin family as novel antimalarial agents.

Authors:
Caterina Fattorusso Giuseppe Campiani Bruno Catalanotti Marco Persico Nicoletta Basilico Silvia Parapini Donatella Taramelli Claudio Campagnuolo Ernesto Fattorusso Adriana Romano Orazio Taglialatela-Scafati

J Med Chem 2006 Nov;49(24):7088-94

Dipartimento di Chimica delle Sostanze Naturali, Università di Napoli Federico II, Via D. Montesano 49, 80131 Napoli, Italy.

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November 2006

Discovery of huperzine A-tacrine hybrids as potent inhibitors of human cholinesterases targeting their midgorge recognition sites.

Authors:
Sandra Gemma Emanuele Gabellieri Paul Huleatt Caterina Fattorusso Marianna Borriello Bruno Catalanotti Stefania Butini Meri De Angelis Ettore Novellino Vito Nacci Tatyana Belinskaya Ashima Saxena Giuseppe Campiani

J Med Chem 2006 Jun;49(11):3421-5

Dipartimento Farmaco Chimico Tecnologico, Via Aldo Moro, Universita' di Siena, 53100 Siena, Italy.

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June 2006