Bernard Delpech

mTOR Inhibition via Displacement of Phosphatidic Acid Induces Enhanced Cytotoxicity Specifically in Cancer Cells.

Cancer Res 2018 09 27;78(18):5384-5397. Epub 2018 Jul 27.

Institut de Chimie des Substances Naturelles, CNRS UPR 2301, Gif-sur-Yvette, France.

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September 2018

Correction: Comparison of the reactivity of β-thiolactones and β-lactones toward ring-opening by thiols and amines.

Authors:

Amandine Noel Bernard Delpech David Crich

Org Biomol Chem 2015 Sep 20;13(35):9324. Epub 2015 Aug 20.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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September 2015

Chemistry of the β-thiolactones: substituent and solvent effects on thermal decomposition and comparison with the β-lactones.

Authors:

Amandine Noel Bernard Delpech David Crich

J Org Chem 2014 May 21;79(9):4068-77. Epub 2014 Apr 21.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS , Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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May 2014

A concise formation of N-substituted 3,4-diarylpyrroles--synthesis and cytotoxic activity.

Authors:

Maxim Egorov Bernard Delpech Geneviève Aubert Thierry Cresteil Maria Concepcion Garcia-Alvarez Pascal Collin Christian Marazano

Org Biomol Chem 2014 Mar;12(9):1518-24

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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March 2014

The Saraine Alkaloids.

Authors:

Bernard Delpech

Alkaloids Chem Biol 2014;73:223-329. Epub 2013 Dec 25.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette Cedex, France. Electronic address:

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December 2013

Formation of N-heterocyclic carbene-boryl radicals through electrochemical and photochemical cleavage of the B-S bond in N-heterocyclic carbene-boryl sulfides.

Authors:

Sofia Telitel Anne-Laure Vallet Stéphane Schweizer Bernard Delpech Nicolas Blanchard Fabrice Morlet-Savary Bernadette Graff Dennis P Curran Marc Robert Emmanuel Lacôte Jacques Lalevée

J Am Chem Soc 2013 Nov 29;135(45):16938-47. Epub 2013 Oct 29.

Institut de Science des Matériaux de Mulhouse IS2M (UMR CNRS 7361), Université de Haute Alsace , 15 rue Jean Starcky, 68057 Mulhouse Cedex, France.

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November 2013

Se-(9-Fluorenylmethyl) selenoesters; preparation, reactivity, and use as convenient synthons for selenoacids.

Authors:

Fabien Fécourt Bernard Delpech Oleg Melnyk David Crich

Org Lett 2013 Jul 1;15(14):3758-61. Epub 2013 Jul 1.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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July 2013

Synthesis and evaluation of 3-deoxy and 3-deoxy-3-fluoro derivatives of gluco- and manno-configured tetrahydropyridoimidazole glycosidase inhibitors.

Authors:

Cécile Ouairy Thierry Cresteil Bernard Delpech David Crich

Carbohydr Res 2013 Aug 21;377:35-43. Epub 2013 May 21.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette, France.

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August 2013

Mechanistic and preparative studies of radical chain homolytic substitution reactions of N-heterocyclic carbene boranes and disulfides.

Authors:

Xiangcheng Pan Anne-Laure Vallet Stéphane Schweizer Karim Dahbi Bernard Delpech Nicolas Blanchard Bernadette Graff Steven J Geib Dennis P Curran Jacques Lalevée Emmanuel Lacôte

J Am Chem Soc 2013 Jul 3;135(28):10484-91. Epub 2013 Jul 3.

Department of Chemistry, University of Pittsburgh, Pittsburgh, Pennsylvania 15260, United States.

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July 2013

Exploration of an imide capture/N,N-acyl shift sequence for asparagine native peptide bond formation.

Authors:

Reda Mhidia Emmanuelle Boll Fabien Fécourt Mikhail Ermolenko Nathalie Ollivier Kaname Sasaki David Crich Bernard Delpech Oleg Melnyk

Bioorg Med Chem 2013 Jun 24;21(12):3479-85. Epub 2013 Mar 24.

CNRS UMR 8161, Univ. Lille Nord de France, Institut Pasteur de Lille, 59021 Lille, France.

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June 2013

Highly stereoselective synthesis of primary, secondary, and tertiary α-S-sialosides under Lewis acidic conditions.

Authors:

Amandine Noel Bernard Delpech David Crich

Org Lett 2012 Aug 30;14(16):4138-41. Epub 2012 Jul 30.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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August 2012

Comparison of the reactivity of β-thiolactones and β-lactones toward ring-opening by thiols and amines.

Authors:

Amandine Noel Bernard Delpech David Crich

Org Biomol Chem 2012 Aug 2;10(32):6480-3. Epub 2012 Jul 2.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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August 2012

Stereoselective, electrophilic α-C-sialidation.

Authors:

Amandine Noel Bernard Delpech David Crich

Org Lett 2012 Mar 15;14(5):1342-5. Epub 2012 Feb 15.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91190 Gif-sur-Yvette, France.

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March 2012

Concise construction of sarain A core according to a biosynthetic proposal: cyclization through an intramolecular Mannich-type reaction involving an endocyclic N-acyliminium ion.

Authors:

Sabrina Peixoto Marie-Thérèse Martin David Crich Bernard Delpech Christian Marazano

Chemistry 2011 Aug 2;17(36):9907-10. Epub 2011 Aug 2.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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August 2011

One-pot formation of piperidine- and pyrrolidine-substituted pyridinium salts via addition of 5-alkylaminopenta-2,4-dienals to N-acyliminium ions: application to the synthesis of (±)-nicotine and analogs.

Authors:

Sabrina Peixoto Tuan Minh Nguyen David Crich Bernard Delpech Christian Marazano

Org Lett 2010 Nov;12(21):4760-3

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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November 2010

Synthesis of N-acyl-5-aminopenta-2,4-dienals via base-induced ring-opening of N-acylated furfurylamines: scope and limitations.

Authors:

Cécile Ouairy Patrick Michel Bernard Delpech David Crich Christian Marazano

J Org Chem 2010 Jun;75(12):4311-4

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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June 2010

Antiplasmodial benzophenone derivatives from the root barks of Symphonia globulifera (Clusiaceae).

Authors:

Guillaume Marti Véronique Eparvier Christian Moretti Soizic Prado Philippe Grellier Nathalie Hue Odile Thoison Bernard Delpech Françoise Guéritte Marc Litaudon

Phytochemistry 2010 Jun 29;71(8-9):964-74. Epub 2010 Mar 29.

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Gif-sur-Yvette, France.

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June 2010

Concise access to a model of the marine alkaloid halicyclamine A through macrocycle-forming addition of a 5-aminopenta-2,4-dienal onto a 2,3-dihydropyridinium salt.

Authors:

Isabelle Sinigaglia Tuan Minh Nguyen Jean-Charles Wypych Bernard Delpech Christian Marazano

Chemistry 2010 Mar;16(12):3594-7

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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March 2010

Enhancement of 5-aminopenta-2,4-dienals electrophilicity via activation by O,N-bistrifluoroacetylation. application to an N-acyl Pictet-Spengler reaction.

Authors:

Philippe Nuhant Sanjay B Raikar Jean-Charles Wypych Bernard Delpech Christian Marazano

J Org Chem 2009 Dec;74(24):9413-21

Centre de Recherche de Gif, Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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December 2009

Alpha,alpha'-annulation of 2,6-prenyl-substituted cyclohexanone derivatives with malonyl chloride: application to a short synthesis of (+/-)-clusianone. Formation and rearrangement of a biogenetic-like intermediate.

Authors:

Philippe Nuhant Marc David Thomas Pouplin Bernard Delpech Christian Marazano

Org Lett 2007 Jan;9(2):287-9

Institut de Chimie des Substances Naturelles, CNRS, 1 Avenue de la Terrasse, 91198 Gif-sur-Yvette, France.

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January 2007

Oblongifolins A-D, polyprenylated benzoylphloroglucinol derivatives from Garcinia oblongifolia.

Authors:

Wafaa Hamed Solenn Brajeul Florence Mahuteau-Betzer Odile Thoison Stéphane Mons Bernard Delpech Van Hung Nguyen Thierry Sévenet Christian Marazano

J Nat Prod 2006 May;69(5):774-7

Institut de Chimie des Substances Naturelles, CNRS, Avenue de la Terrasse, 91198 Gif-sur-Yvette Cedex, France.

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May 2006

Publications by authors named "Bernard Delpech"

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