Publications by authors named "Antonella Goggiamani"

30Publications

Synthesis of functionalised 2,3-dihydroquinolin-4(1)-ones quinoline or -alkenylindole derivatives through sequential reactions of 2-alkynylanilines with ketones.

Authors:
Vincenzo Marsicano Antonio Arcadi Marco Chiarini Giancarlo Fabrizi Antonella Goggiamani Antonia Iazzetti

Org Biomol Chem 2020 Dec 14. Epub 2020 Dec 14.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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December 2020

Naturally-Occurring Alkaloids of Plant Origin as Potential Antimicrobials against Antibiotic-Resistant Infections.

Authors:
Bruno Casciaro Laura Mangiardi Floriana Cappiello Isabella Romeo Maria Rosa Loffredo Antonia Iazzetti Andrea Calcaterra Antonella Goggiamani Francesca Ghirga Maria Luisa Mangoni Bruno Botta Deborah Quaglio

Molecules 2020 Aug 9;25(16). Epub 2020 Aug 9.

Department of Chemistry and Technology of Drugs, "Department of Excellence 2018-2022", Sapienza University of Rome, P.le Aldo Moro 5, 00185 Rome, Italy.

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August 2020

Synthesis of pyrano[2,3-f]chromen-2-ones vs. pyrano[3,2-g]chromen-2-ones through site controlled gold-catalyzed annulations.

Authors:
Antonio Arcadi Alessia Ciogli Giancarlo Fabrizi Andrea Fochetti Roberta Franzini Francesca Ghirga Antonella Goggiamani Antonia Iazzetti

Org Biomol Chem 2019 12;17(47):10065-10072

Dipartimento di Scienze Fisiche e Chimiche Università degli Studi di L'Aquila, Via Vetoio, 67100 Coppito (AQ), Italy.

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December 2019

Stereo- and regioselective gold(i)-catalyzed hydroamination of 2-(arylethynyl)pyridines with anilines.

Authors:
Sandro Cacchi Giancarlo Fabrizi Andrea Fochetti Francesca Ghirga Antonella Goggiamani Antonia Iazzetti

Org Biomol Chem 2019 01;17(3):527-532

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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January 2019

Synthesis of indolo[1,2-]quinazolines from 2-alkynylaniline derivatives through Pd-catalyzed indole formation/cyclization with ,-dimethylformamide dimethyl acetal.

Authors:
Antonio Arcadi Sandro Cacchi Giancarlo Fabrizi Francesca Ghirga Antonella Goggiamani Antonia Iazzetti Fabio Marinelli

Beilstein J Org Chem 2018 14;14:2411-2417. Epub 2018 Sep 14.

Dipartimento di Scienze Fisiche e Chimiche, Università di L'Aquila, Via Vetoio, 671010 Coppito (AQ), Italy.

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September 2018

Design, Palladium-Catalyzed Synthesis, and Biological Investigation of 2-Substituted 3-Aroylquinolin-4(1H)-ones as Inhibitors of the Hedgehog Signaling Pathway.

Authors:
Romina Alfonsi Bruno Botta Sandro Cacchi Lucia Di Marcotullio Giancarlo Fabrizi Roberta Faedda Antonella Goggiamani Antonia Iazzetti Mattia Mori

J Med Chem 2017 02 10;60(4):1469-1477. Epub 2017 Feb 10.

Center for Life Nano Science@Sapienza, Istituto Italiano di Tecnologia , Viale Regina Elena 291, 00161 Rome, Italy.

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February 2017

Construction of the 1,5-Benzodiazepine Skeleton from o-Phenylendiamine and Propargylic Alcohols via a Domino Gold-Catalyzed Hydroamination/Cyclization Process.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Antonia Iazzetti

Org Lett 2016 08 28;18(15):3511-3. Epub 2016 Jul 28.

Dipartimento di Chimica e Tecnologie del Farmaco, La Sapienza, Università di Roma , P.le A. Moro 5, 00185 Rome, Italy.

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August 2016

Pd- and Rh-Catalyzed Hydroarylation of γ-(2-Methoxycarbonylphenyl)propargylic Alcohols: Approaches to 4- or 5-Substituted Seven-Membered Benzolactones and 3,3-Disubstituted Phthalides.

Authors:
Antonio Arcadi Giancarlo Fabrizi Antonella Goggiamani Fabio Marinelli

J Org Chem 2015 Jul 6;80(14):6986-95. Epub 2015 Jul 6.

†Dipartimento di Scienze Fisiche e Chimiche, Università di L'Aquila, Via Vetoio - 67010 Coppito (AQ), Italy.

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July 2015

Palladium-catalyzed synthesis of 2-(aminomethyl)indoles from 3-(o-trifluoroacetamidoaryl)-1-propargylic alcohols and amines.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Carmela Molinaro Rosanna Verdiglione

J Org Chem 2014 Jan 18;79(1):401-7. Epub 2013 Dec 18.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma , P.le A. Moro 5, 00185 Rome, Italy.

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January 2014

Palladium-catalyzed cascade reactions of 1-(3-arylprop-2-ynyloxy)-2-bromo benzene derivatives with organoboron compounds.

Authors:
Antonio Arcadi Federico Blesi Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Fabio Marinelli

J Org Chem 2013 May 22;78(9):4490-8. Epub 2013 Apr 22.

Dipartimento di Scienze Fisiche e Chimiche, Università di L'Aquila, Via Vetoio, 67010, Coppito (AQ), Italy.

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May 2013

2-Substituted 3-arylindoles through palladium-catalyzed arylative cyclization of 2-alkynyltrifluoroacetanilides with arylboronic acids under oxidative conditions.

Authors:
Antonio Arcadi Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Antonia Iazzetti Fabio Marinelli

Org Biomol Chem 2013 Jan 6;11(4):545-8. Epub 2012 Dec 6.

Dipartimento di Scienze Fisiche e Chimiche, Università degli Studi di L'Aquila, Via Vetoio, 67010 Coppito, L'Aquila, Italy.

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January 2013

Gold versus silver catalyzed intramolecular hydroarylation reactions of [(3-arylprop-2-ynyl)oxy]benzene derivatives.

Authors:
Antonio Arcadi Federico Blesi Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Fabio Marinelli

Org Biomol Chem 2012 Dec 13;10(48):9700-8. Epub 2012 Nov 13.

Dipartimento di Scienze Fisiche e Chimiche, Università degli Studi di L'Aquila, Via Vetoio, 67010 Coppito, L'Aquila, Italy.

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December 2012

Dibenzo[a,c]carbazoles from 2-(2-bromoaryl)-3-arylindoles via a palladium-catalyzed intramolecular C-H functionalization/C-C bond formation process.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Antonia Iazzetti

Org Biomol Chem 2012 Dec 29;10(46):9142-7. Epub 2012 Oct 29.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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December 2012

One-pot gold-catalyzed synthesis of azepino[1,2-a]indoles.

Authors:
Gianpiero Cera Stefano Piscitelli Michel Chiarucci Giancarlo Fabrizi Antonella Goggiamani Rubén S Ramón Steven P Nolan Marco Bandini

Angew Chem Int Ed Engl 2012 Sep 3;51(39):9891-5. Epub 2012 Sep 3.

Dipartimento di Chimica G. Ciamician, Alma Mater Studiorum-Università di Bologna, Bologna, Italy.

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September 2012

Palladium-catalyzed synthesis of 2-amino ketones from propargylic carbonates and secondary amines.

Authors:
Sandro Cacchi Giancarlo Fabrizi Eleonora Filisti Antonella Goggiamani Antonia Iazzetti Loredana Maurone

Org Biomol Chem 2012 Jun 18;10(24):4699-703. Epub 2012 May 18.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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June 2012

4-Aryl-2-quinolones from 3,3-diarylacrylamides through intramolecular copper-catalyzed C-H functionalization/C-N bond formation.

Authors:
Roberta Berrino Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani

J Org Chem 2012 Mar 22;77(5):2537-42. Epub 2012 Feb 22.

Dipartimento di Chimica e Tecnologie del Farmaco, La Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, Italy.

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March 2012

Functionalized 2,3-dihydrofurans via palladium-catalyzed oxyarylation of α-allyl-β-ketoesters.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Antonia Iazzetti David Madec Giovanni Poli Guillaume Prestat

Org Biomol Chem 2011 Dec 1;9(24):8233-6. Epub 2011 Nov 1.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Roma, Italy.

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December 2011

Heck reaction of arenediazonium salts with N,N-diprotected allylamines. Synthesis of cinnamylamines and indoles.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Alessio Sferrazza

Org Biomol Chem 2011 Mar 11;9(6):1727-30. Epub 2011 Feb 11.

Dipartimento di Chimica e Tecnologie del Farmaco, La Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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March 2011

Copper catalysis in the construction of indole and benzo[b]furan rings.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani

Org Biomol Chem 2011 Feb 2;9(3):641-52. Epub 2010 Dec 2.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185, Rome, Italy.

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February 2011

Arenediazonium tetrafluoroborates in palladium-catalyzed C-P bond-forming reactions. Synthesis of arylphosphonates, -phosphine oxides, and -phosphines.

Authors:
Roberta Berrino Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Paolo Stabile

Org Biomol Chem 2010 Oct 13;8(20):4518-20. Epub 2010 Aug 13.

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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October 2010

2,3-Disubstituted indoles via palladium-catalyzed reaction of 2-alkynyltrifluoroacetanilides with arenediazonium tetrafluoroborates.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Alcide Perboni Alessio Sferrazza Paolo Stabile

Org Lett 2010 Jul;12(14):3279-81

Dipartimento di Chimica e Tecnologie del Farmaco, La Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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July 2010

Sonogashira cross-coupling of arenediazonium salts.

Authors:
Giancarlo Fabrizi Antonella Goggiamani Alessio Sferrazza Sandro Cacchi

Angew Chem Int Ed Engl 2010 Jun;49(24):4067-70

Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P.le A. Moro 5, 00185 Rome, Italy.

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June 2010

Diastereoselective synthesis of hexahydro-3H-pyrrolyzin-3-ones through Pd-catalyzed carboamination.

Authors:
Luana Bagnoli Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Catalina Scarponi Marcello Tiecco

J Org Chem 2010 Mar;75(6):2134-7

Dipartimento di Chimica e Tecnologia del Farmaco, Sezione di Chimica Organica, Università di Perugia, 06123 Perugia, Italy.

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March 2010

Palladium-catalyzed hydroarylation of alkynes with arenediazonium salts.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Daniela Persiani

Org Lett 2008 Apr 20;10(8):1597-600. Epub 2008 Mar 20.

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi La Sapienza, Piazzale A. Moro 5, 00185 Rome, Italy.

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April 2008

Synthesis of N,N-Dialkyl-N'-arylhydrazines via palladium-catalyzed N-arylation by using N,N-dialkylhydrazines/2LiCl adducts.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Emanuela Licandro Stefano Maiorana Dario Perdicchia

Org Lett 2005 Apr;7(8):1497-500

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi La Sapienza, P.le A. Moro 5, 00185 Roma, Italy.

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April 2005

Palladium-catalyzed synthesis of aldehydes from aryl iodides and acetic formic anhydride.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani

J Comb Chem 2004 Sep-Oct;6(5):692-4

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi "La Sapienza", P.le A. Moro 5, 00185 Rome, Italy.

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January 2006

Unsymmetrical diaryl sulfones and aryl vinyl sulfones through palladium-catalyzed coupling of aryl and vinyl halides or triflates with sulfinic acid salts.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Luca M Parisi Roberta Bernini

J Org Chem 2004 Aug;69(17):5608-14

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi "La Sapienza", P. le A. Moro 5, 00185 Rome, Italy.

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August 2004

Palladium-catalyzed hydroxycarbonylation of aryl and vinyl halides or triflates by acetic anhydride and formate anions.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani

Org Lett 2003 Nov;5(23):4269-72

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi La Sapienza, P.le A. Moro 5, 00185 Rome, Italy.

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November 2003

Palladium-catalyzed reaction of aryl iodides with acetic anhydride. A carbon monoxide-free synthesis of acetophenones.

Authors:
Sandro Cacchi Giancarlo Fabrizi Federica Gavazza Antonella Goggiamani

Org Lett 2003 Feb;5(3):289-91

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi La Sapienza, Ple A Moro 5, 00185 Roma, Italy.

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February 2003

Unsymmetrical diaryl sulfones through palladium-catalyzed coupling of aryl iodides and arenesulfinates.

Authors:
Sandro Cacchi Giancarlo Fabrizi Antonella Goggiamani Luca M Parisi

Org Lett 2002 Dec;4(26):4719-21

Dipartimento di Studi di Chimica e Tecnologia delle Sostanze Biologicamente Attive, Università degli Studi La Sapienza, P. le A. Moro 5, 00185 Rome, Italy.

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December 2002