Anil K Saxena

Anil K Saxena

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Synthesis, SAR and docking studies of substituted aryl phenylthiazolyl phenylcarboxamide as potential protein tyrosine phosphatase 1B (PTP1B) inhibitors.

Chem Biol Drug Des 2019 Jul 5;94(1):1378-1389. Epub 2019 Jun 5.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow, India.

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http://dx.doi.org/10.1111/cbdd.13515DOI Listing
July 2019

Synthesis of primaquine glyco-conjugates as potential tissue schizontocidal antimalarial agents.

Chem Biol Drug Des 2017 08 22;90(2):254-261. Epub 2017 Feb 22.

Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Lucknow, UP, India.

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http://dx.doi.org/10.1111/cbdd.12944DOI Listing
August 2017

Insight into stereoselective disposition of enantiomers of a potent antithrombotic agent, S002-333 following administration of the racemic compound to mice.

Eur J Pharm Sci 2017 Apr 9;101:107-114. Epub 2017 Feb 9.

Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow 226032, Uttar Pradesh, India; Academy of Scientific and Innovative Research, New Delhi 110001, India. Electronic address:

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http://dx.doi.org/10.1016/j.ejps.2017.02.012DOI Listing
April 2017

Design, Synthesis, and Biological Evaluation of Novel 1,2,4-Trioxanes as Potential Antimalarial Agents.

Arch Pharm (Weinheim) 2017 Apr 16;350(3-4). Epub 2017 Feb 16.

Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow, India.

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http://dx.doi.org/10.1002/ardp.201600335DOI Listing
April 2017

Taxonomic and functional diversity of the culturable microbiomes of epigeic earthworms and their prospects in agriculture.

J Basic Microbiol 2016 Sep 2;56(9):1009-20. Epub 2016 May 2.

ICAR - Indian Veterinary Research Institute, Izatnagar, Bareilly, Uttar Pradesh, India.

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http://dx.doi.org/10.1002/jobm.201500779DOI Listing
September 2016

Pre-clinical investigation of plasma pharmacokinetics and biodistribution of a novel antithrombotic agent S002-333 in mice using LC-MS/MS.

J Chromatogr B Analyt Technol Biomed Life Sci 2016 Sep 18;1031:154-162. Epub 2016 Jul 18.

Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow, Uttar Pradesh 226032, India; Academy of Scientific and Innovative Research, New Delhi 110001, India. Electronic address:

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http://dx.doi.org/10.1016/j.jchromb.2016.07.030DOI Listing
September 2016

Enantioselective inhibition of Cytochrome P450-mediated drug metabolism by a novel antithrombotic agent, S002-333: Major effect on CYP2B6.

Chem Biol Interact 2016 Aug 4;256:257-65. Epub 2016 Jul 4.

Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Lucknow 226032, Uttar Pradesh, India; Academy of Scientific and Innovative Research, New Delhi 110001, India. Electronic address:

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http://dx.doi.org/10.1016/j.cbi.2016.07.001DOI Listing
August 2016

First high quality draft genome sequence of a plant growth promoting and cold active enzyme producing psychrotrophic Arthrobacter agilis strain L77.

Stand Genomic Sci 2016 26;11(1):54. Epub 2016 Aug 26.

Division of Microbiology, ICAR-Indian Agricultural Research Institute, New Delhi, 110012 India ; Present Address: ICAR-National Bureau of Agriculturally Important Microorganisms, Kushmaur, Mau, 275103 Uttar Pradesh India.

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http://dx.doi.org/10.1186/s40793-016-0176-4DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC5000428PMC
August 2016

Pharmacokinetics, dose proportionality and permeability of S002-333 and its enantiomers, a potent antithrombotic agent, in rabbits.

Xenobiotica 2015 18;45(11):1016-23. Epub 2015 Jun 18.

a Pharmacokinetics and Metabolism Division, CSIR - Central Drug Research Institute , Lucknow , India .

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http://dx.doi.org/10.3109/00498254.2015.1034224DOI Listing
June 2016

Metabolic profiling of a novel antithrombotic compound, S002-333 and enantiomers: metabolic stability, species comparison and in vitro-in vivo extrapolation.

Biopharm Drug Dispos 2016 May;37(4):185-99

Pharmacokinetics and Metabolism Division, CSIR - Central Drug Research Institute, Lucknow, 226031, India.

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http://dx.doi.org/10.1002/bdd.1995DOI Listing
May 2016

Pharmacophore Modeling, Docking and Molecular Dynamics Studies on Caspase-3 Activators Binding at β-Tubulin Site.

Curr Comput Aided Drug Des 2015 ;11(1):72-83

Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Lucknow 226031, India.

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April 2016

Novel Glycoconjugate of 8-Fluoro Norfloxacin Derivatives as Gentamicin-resistant Staphylococcus aureus Inhibitors: Synthesis and Molecular Modelling Studies.

Chem Biol Drug Des 2015 Oct 20;86(4):440-6. Epub 2015 Jan 20.

Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Lucknow, UP, 226031, India.

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http://dx.doi.org/10.1111/cbdd.12503DOI Listing
October 2015

Molecular modelling based target identification for endo-peroxides class of antimalarials.

Comb Chem High Throughput Screen 2015 ;18(2):199-207

Academy of Sciences and Innovative Research, India.

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September 2015

Taxonomic and functional annotation of gut bacterial communities of Eisenia foetida and Perionyx excavatus.

Microbiol Res 2015 Jun 10;175:48-56. Epub 2015 Mar 10.

Division of Microbiology, ICAR-Indian Agricultural Research Institute, New Delhi 110012, India.. Electronic address:

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http://dx.doi.org/10.1016/j.micres.2015.03.003DOI Listing
June 2015

Novel, potent, orally bioavailable and selective mycobacterial ATP synthase inhibitors that demonstrated activity against both replicating and non-replicating M. tuberculosis.

Bioorg Med Chem 2015 Feb 2;23(4):742-52. Epub 2015 Jan 2.

Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, B.S. 10/1, Sector 10, Jankipuram Extension, Sitapur Road, Lucknow 226031, India. Electronic address:

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http://dx.doi.org/10.1016/j.bmc.2014.12.060DOI Listing
February 2015

Culturable diversity and functional annotation of psychrotrophic bacteria from cold desert of Leh Ladakh (India).

World J Microbiol Biotechnol 2015 Jan 5;31(1):95-108. Epub 2014 Nov 5.

Division of Microbiology, Indian Agricultural Research Institute, New Delhi, 110012, India.

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http://dx.doi.org/10.1007/s11274-014-1768-zDOI Listing
January 2015

Purification and physicochemical characterization of a trypsin inhibitor from Cassia absus Linn.

Protein Pept Lett 2014 ;21(2):108-14

Department of Biotechnology, Indian Institute of Technology Roorkee, Roorkee-247 667, India.

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September 2014

Pharmacokinetic and metabolism studies of rohitukine in rats by high performance liquid-chromatography with tandem mass spectrometry.

Fitoterapia 2014 Sep 16;97:34-42. Epub 2014 May 16.

Pharmacokinetics & Metabolism Div., CSIR - Central Drug Research Institute, Lucknow 226031, India; Academy of Scientific and Innovative Research (AcSIR), Anusandhan Bhawan, Rafi Marg, New Delhi 110 001, India. Electronic address:

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http://dx.doi.org/10.1016/j.fitote.2014.05.004DOI Listing
September 2014

Genetic and functional diversity of fluorescent Pseudomonas from rhizospheric soils of wheat crop.

J Basic Microbiol 2014 May 17;54(5):425-37. Epub 2013 May 17.

National Bureau of Agriculturally Important Microorganisms, Mau Nath Bhanjan, Mau, Uttar Pradesh, India.

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http://dx.doi.org/10.1002/jobm.201200384DOI Listing
May 2014

In vitro metabolism of a novel antithrombotic compound, S002-333, and its enantiomers: quantitative cytochrome P450 phenotyping, metabolic profiling and enzyme kinetic studies.

Xenobiotica 2014 Apr 30;44(4):295-308. Epub 2013 Aug 30.

Pharmacokinetics and Metabolism Division, CSIR - Central Drug Research Institute , Lucknow, Uttar Pradesh , India .

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http://dx.doi.org/10.3109/00498254.2013.831958DOI Listing
April 2014

Metal-free, mild, nonepimerizing, chemo- and enantio- or diastereoselective N-alkylation of amines by alcohols via oxidation/imine-iminium formation/reductive amination: a pragmatic synthesis of octahydropyrazinopyridoindoles and higher ring analogues.

J Org Chem 2013 Dec 17;78(23):11656-69. Epub 2013 Sep 17.

Laboratory No. 101, Medicinal and Process Chemistry Division (MPC), CSIR-Central Drug Research Institute (CDRI) , Chattar Manzil Palace, Lucknow, Uttar Pradesh 226-001, India.

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http://dx.doi.org/10.1021/jo4012249DOI Listing
December 2013

Drug/drug interaction of common NSAIDs with antiplatelet effect of aspirin in human platelets.

Eur J Pharmacol 2013 Dec 25;721(1-3):215-24. Epub 2013 Sep 25.

Institut für Pharmakologie und Klinische Pharmakologie, Heinrich-Heine-Universität Düsseldorf, Moorenstraße 5, 40225 Düsseldorf, Germany.

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http://dx.doi.org/10.1016/j.ejphar.2013.09.032DOI Listing
December 2013

Antidyslipidemic and antioxidant effects of novel Lupeol-derived chalcones.

Lipids 2013 Oct 14;48(10):1017-27. Epub 2013 Aug 14.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow, 226 001, India.

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http://dx.doi.org/10.1007/s11745-013-3824-0DOI Listing
October 2013

Cold-active hydrolases producing bacteria from two different sub-glacial Himalayan lakes.

J Basic Microbiol 2013 Aug 7;53(8):703-14. Epub 2012 Sep 7.

National Bureau of Agriculturally Important Microorganisms (NBAIM), Kusmaur, Mau, Uttar Pradesh, India.

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http://dx.doi.org/10.1002/jobm.201200126DOI Listing
August 2013

Optimization of media components for chitinase production by chickpea rhizosphere associated Lysinibacillus fusiformis B-CM18.

J Basic Microbiol 2013 May 26;53(5):451-60. Epub 2012 Jun 26.

National Bureau of Agriculturally Important Microorganisms, Mau, Uttar Pradesh, India -275101.

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http://dx.doi.org/10.1002/jobm.201100590DOI Listing
May 2013

Biological evaluation of novel substituted chloroquinolines targeting mycobacterial ATP synthase.

Int J Antimicrob Agents 2013 Jan 8;41(1):41-6. Epub 2012 Nov 8.

Division of Microbiology, Council of Scientific and Industrial Research (CSIR)-Central Drug Research Institute, Lucknow, India.

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http://dx.doi.org/10.1016/j.ijantimicag.2012.09.012DOI Listing
January 2013

Identification of novel amino acid derived CCK-2R antagonists as potential antiulcer agent: homology modeling, design, synthesis, and pharmacology.

J Chem Inf Model 2013 Jan 4;53(1):176-87. Epub 2013 Jan 4.

Medicinal and Process Chemistry Division, CSIR-Central Drug Research Institute, Lucknow, 226001, India.

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http://dx.doi.org/10.1021/ci3003655DOI Listing
January 2013

Exploration and characterization of agriculturally and industrially important haloalkaliphilic bacteria from environmental samples of hypersaline Sambhar lake, India.

World J Microbiol Biotechnol 2012 Nov 25;28(11):3207-17. Epub 2012 Jul 25.

National Bureau of Agriculturally Important Microorganisms, Kusmaur, Mau 275101, Uttar Pradesh, India.

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http://dx.doi.org/10.1007/s11274-012-1131-1DOI Listing
November 2012

Lead optimization studies towards the discovery of novel carbamates as potent AChE inhibitors for the potential treatment of Alzheimer's disease.

Bioorg Med Chem 2012 Nov 12;20(21):6313-20. Epub 2012 Sep 12.

Division of Medicinal and Process Chemistry, CSIR Central Drug Research Institute, Lucknow 226 001, India.

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http://dx.doi.org/10.1016/j.bmc.2012.09.005DOI Listing
November 2012

End-Stage Sickle Cell Nephropathy: Determinants of Reduced Survival of Patients on Long-term Hemodialysis.

Saudi J Kidney Dis Transpl 2004 Apr-Jun;15(2):174-5

Division of Nephrology, Post-graduate Department of Medicine, Hofuf, Al-Hasa-31982, Saudi Arabia.

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October 2012

The Prevalence of Nasal Carriage of Staphylococcus aureus and Associated Vascular Access-Related Septicemia Among Patients on Hemodialysis in Al-Hasa Region of Saudi Arabia.

Saudi J Kidney Dis Transpl 2003 Jan-Mar;14(1):30-8

Division of Nephrology, King Fahad Hospital, Hofuf, Al-Hasa, Saudi Arabia.

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October 2012

Hemodynamic factors and oxidative stress: a unifying concept in the progression of renal disease?

Authors:
Anil K Saxena

Saudi J Kidney Dis Transpl 2003 Oct-Dec;14(4):531-4

Post-graduate Department of Medicine, King Fahad Hospital and Tertiary Care Center, Hofuf, Al-Hasa-31982, Saudi Arabia.

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October 2012

The new molecular revelations of recurrent focal segmental glomerulosclerosis in renal allografts.

Authors:
Anil K Saxena

Saudi J Kidney Dis Transpl 2002 October-December;13(4):511-2

Post-Graduate Department of Medicine, King Fahad Hospital, Hofuf, Al-Hasa 31982, Saudi Arabia.

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October 2012

Antibiotic-Heparin Lock Technique: A Potentially Precious Tool to Prevent Hemodialysis Catheter-related Septicemia.

Saudi J Kidney Dis Transpl 2004 Jan-Mar;15(1):67-9

Post-graduate Department of Medicine, King Fahad Hospital & Tertiary Care Center, Hofuf, Al-Hasa-31982, Saudi Arabia.

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October 2012

Vascular access related septicemia in hemodialysis: a focus on bacterial flora and antibiotic access salvage.

Saudi J Kidney Dis Transpl 2002 Jan-Mar;13(1):29-34

Department of Microbiology, King Fahad Hospital, Hofuf, Al-Hasa, Saudi Arabia.

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October 2012

How Harmless are Herbal Remedies on Human Kidneys?

Authors:
Anil K Saxena

Saudi J Kidney Dis Transpl 2003 Apr-Jun;14(2):205-6

Division of Nephrology, Post-graduate Department of Medicine, King Fahad Hospital and Tertiary Care Center, Hofuf, Al-Hasa-31982, Saudi Arabia.

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October 2012

Vascular access related infections in hemodialysis patients.

Saudi J Kidney Dis Transpl 2005 Jan-Mar;16(1):46-71

Division of Nephrology, Postgraduate Department of Medicine, King Fahd Hospital & Territory Care Center, Hofuf, Al-Hasa, Saudi Arabia.

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October 2012

Synthesis, structure-activity relationship and docking studies of substituted aryl thiazolyl phenylsulfonamides as potential protein tyrosine phosphatase 1B inhibitors.

ChemMedChem 2012 Jul 21;7(7):1185-90. Epub 2012 May 21.

Division of Medicinal and Process Chemistry, Council of Scientific and Industrial Research (CSIR), Central Drug Research Institute (CDRI), Chattar Manzil Palace, M G Marg, Lucknow, Uttar Pardesh 226001, India.

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http://dx.doi.org/10.1002/cmdc.201200197DOI Listing
July 2012

Cefotaxime-heparin lock prophylaxis against hemodialysis catheter-related sepsis among Staphylococcus aureus nasal carriers.

Saudi J Kidney Dis Transpl 2012 Jul;23(4):743-54

Al-Rahba Hospital-Johns Hopkins Medicine International, Abu Dhabi, United Arab Emirates.

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http://www.sjkdt.org/text.asp?2012/23/4/743/98154
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http://dx.doi.org/10.4103/1319-2442.98154DOI Listing
July 2012

Epiphytic pink-pigmented methylotrophic bacteria enhance germination and seedling growth of wheat (Triticum aestivum) by producing phytohormone.

Antonie Van Leeuwenhoek 2012 May 27;101(4):777-86. Epub 2011 Dec 27.

National Bureau of Agriculturally Important Microorganisms, Kushmaur, Maunath Bhanjan, India.

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http://dx.doi.org/10.1007/s10482-011-9692-9DOI Listing
May 2012

Toward the identification of a reliable 3D QSAR pharmacophore model for the CCK2 receptor antagonism.

J Chem Inf Model 2012 May 4;52(5):1376-90. Epub 2012 May 4.

Medicinal and Process Chemistry Division, C.S.I.R.-Central Drug Research Institute, Lucknow 226001, India.

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http://dx.doi.org/10.1021/ci300094eDOI Listing
May 2012

Genetic and functional diversity of Bacillus strains in the soils long-term irrigated with paper and pulp mill effluent.

J Gen Appl Microbiol 2011 ;57(4):183-95

National Bureau of Agriculturally Important Microorganisms, Mau Nath Bhanjan, India.

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January 2012

Fragment-based design, docking, synthesis, biological evaluation and structure-activity relationships of 2-benzo/benzisothiazolimino-5-aryliden-4-thiazolidinones as cycloxygenase/lipoxygenase inhibitors.

Eur J Med Chem 2012 Jan 25;47(1):111-24. Epub 2011 Oct 25.

Department of Medical Laboratory Studies, School of Health and Medical Care, Alexander Technological Education Institute of Thessaloniki, Thessaloniki 57400, Greece.

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http://dx.doi.org/10.1016/j.ejmech.2011.10.029DOI Listing
January 2012

Synthesis and 2D QSAR of O-sulphonated β-aminols derivatives as novel antifungal and antibacterial agents.

Bioorg Med Chem Lett 2011 Nov 23;21(21):6476-81. Epub 2011 Aug 23.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226 001, India.

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http://dx.doi.org/10.1016/j.bmcl.2011.08.078DOI Listing
November 2011

CoMFA, CoMSIA, and docking studies on thiolactone-class of potent anti-malarials: identification of essential structural features modulating anti-malarial activity.

Chem Biol Drug Des 2011 Sep 13;78(3):483-93. Epub 2011 Jul 13.

Division of Medicinal and Process Chemistry, Central Drug Research Institute CSIR, Lucknow-226001, India.

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http://dx.doi.org/10.1111/j.1747-0285.2011.01158.xDOI Listing
September 2011

Synthesis and biological evaluation of substituted 4-arylthiazol-2-amino derivatives as potent growth inhibitors of replicating Mycobacterium tuberculosis H₃₇Rv.

Bioorg Med Chem Lett 2011 Sep 2;21(18):5589-93. Epub 2011 Jul 2.

Division of Medicinal and Process Chemistry, Central Drug Research Institute, CSIR, Lucknow 226 001, India.

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https://linkinghub.elsevier.com/retrieve/pii/S0960894X110085
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http://dx.doi.org/10.1016/j.bmcl.2011.06.076DOI Listing
September 2011

Profiling the structural determinants for the selectivity of representative factor-Xa and thrombin inhibitors using combined ligand-based and structure-based approaches.

J Chem Inf Model 2011 Aug 1;51(8):1966-85. Epub 2011 Aug 1.

Division of Medicinal and Process Chemistry, Central Drug Research Institute, CSIR, Lucknow, India.

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http://dx.doi.org/10.1021/ci200185qDOI Listing
August 2011

Structural basis for the β-adrenergic receptor subtype selectivity of the representative agonists and antagonists.

J Chem Inf Model 2011 Jun 13;51(6):1405-22. Epub 2011 May 13.

Division of Medicinal and Process Chemistry, Central Drug Research Institute, CSIR, Lucknow, India.

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http://dx.doi.org/10.1021/ci2000874DOI Listing
June 2011

Integration-mediated prediction enrichment of quantitative model for Hsp90 inhibitors as anti-cancer agents: 3D-QSAR study.

Mol Divers 2011 May 26;15(2):477-89. Epub 2010 Aug 26.

Division of Medicinal and Process Chemistry, Central Drug Research Institute, CSIR, Lucknow, 226001, India.

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http://dx.doi.org/10.1007/s11030-010-9269-yDOI Listing
May 2011

Diversity and phylogeny of plant growth-promoting bacilli from moderately acidic soil.

J Basic Microbiol 2011 Feb 12;51(1):98-106. Epub 2010 Nov 12.

National Bureau of Agriculturally Important Microorganisms, Mau Nath Bhanjan, Uttar Pradesh, India.

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http://dx.doi.org/10.1002/jobm.201000098DOI Listing
February 2011

Cloning, overexpression and characterization of Leishmania donovani squalene synthase.

FEMS Microbiol Lett 2010 Oct 16;311(1):82-92. Epub 2010 Aug 16.

Division of Biochemistry, Central Drug Research Institute, Lucknow, UP, India.

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http://dx.doi.org/10.1111/j.1574-6968.2010.02071.xDOI Listing
October 2010

Design, synthesis and docking studies on phenoxy-3-piperazin-1-yl-propan-2-ol derivatives as protein tyrosine phosphatase 1B inhibitors.

Bioorg Med Chem Lett 2010 Oct 7;20(19):5732-4. Epub 2010 Aug 7.

Medicinal and Process Chemistry Division, Central Drug Research Institute, CSIR, Lucknow 226001, India.

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http://linkinghub.elsevier.com/retrieve/pii/S0960894X1001118
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http://dx.doi.org/10.1016/j.bmcl.2010.08.008DOI Listing
October 2010

Pharmacophore modeling of substituted 1,2,4-Trioxanes for quantitative prediction of their antimalarial activity.

J Chem Inf Model 2010 Aug;50(8):1510-20

Medicinal and Process Chemistry Division and Parasitology Division, Central Drug Research Institute, CSIR, Lucknow, 226001, India.

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http://pubs.acs.org/doi/abs/10.1021/ci100180e
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http://dx.doi.org/10.1021/ci100180eDOI Listing
August 2010

Substituted hydrazinecarbothioamide as potent antitubercular agents: synthesis and quantitative structure-activity relationship (QSAR).

Bioorg Med Chem Lett 2010 Apr 23;20(8):2597-600. Epub 2010 Feb 23.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226 001, India.

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http://dx.doi.org/10.1016/j.bmcl.2010.02.081DOI Listing
April 2010

Consensus superiority of the pharmacophore-based alignment, over maximum common substructure (MCS): 3D-QSAR studies on carbamates as acetylcholinesterase inhibitors.

J Chem Inf Model 2009 Jun;49(6):1590-601

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow, India 226001.

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http://dx.doi.org/10.1021/ci900049eDOI Listing
June 2009

Synthesis of protein tyrosine phosphatase 1B inhibitors: model validation and docking studies.

Bioorg Med Chem Lett 2009 Apr 21;19(8):2320-3. Epub 2009 Feb 21.

Central Drug Research Institute, Medicinal and Process Chemistry, Chattar Manzil Palace, Mahatma Gandhi Marg, Lucknow, Uttar Pradesh, India.

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http://dx.doi.org/10.1016/j.bmcl.2009.02.058DOI Listing
April 2009

Substituted 1,2,3,4-tetrahydroquinolin-6-yloxypropanes as beta3-adrenergic receptor agonists: design, synthesis, biological evaluation and pharmacophore modeling.

Bioorg Med Chem 2009 Jan 19;17(2):830-47. Epub 2008 Nov 19.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226001, India.

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http://dx.doi.org/10.1016/j.bmc.2008.11.030DOI Listing
January 2009

An investigation of structurally diverse carbamates for acetylcholinesterase (AChE) inhibition using 3D-QSAR analysis.

J Mol Graph Model 2008 Sep 24;27(2):197-208. Epub 2008 Apr 24.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226001, UP, India.

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http://dx.doi.org/10.1016/j.jmgm.2008.04.006DOI Listing
September 2008

Identification and detection of Macrophomina phaseolina by using species-specific oligonucleotide primers and probe.

Mycologia 2007 Nov-Dec;99(6):797-803

National Bureau of Agriculturally Important Microorganisms, Mau Nath Bhanjan, Post bag no.-6, Uttar Pradesh-2 75101, India.

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April 2008

Computer-aided discovery of anti-inflammatory thiazolidinones with dual cyclooxygenase/lipoxygenase inhibition.

J Med Chem 2008 Mar 27;51(6):1601-9. Epub 2008 Feb 27.

Department of Pharmaceutical Chemistry, School of Pharmacy, Aristotle University, Thessaloniki, Greece.

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http://dx.doi.org/10.1021/jm701496hDOI Listing
March 2008

QSAR analysis of PPAR-gamma agonists as anti-diabetic agents.

Eur J Med Chem 2008 Jan 18;43(1):73-80. Epub 2007 Mar 18.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Chattar Manzil Palace, MG Marg, Lucknow, Uttar Pradesh 226001, India.

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http://dx.doi.org/10.1016/j.ejmech.2007.03.004DOI Listing
January 2008

N-acetylcysteine for preventing ototoxicity in hemodialysis patients receiving gentamicin.

Authors:
Anil K Saxena

Nat Clin Pract Nephrol 2007 Sep 31;3(9):478-9. Epub 2007 Jul 31.

Al-Rahba Hospital, Health Authority of Abu Dhabi, Department of Medicine/Nephrology, Abu Dhabi, United Arab Emirates.

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http://dx.doi.org/10.1038/ncpneph0572DOI Listing
September 2007

alpha-Amino acid derivatives as proton pump inhibitors and potent anti-ulcer agents.

Eur J Med Chem 2007 Mar 11;42(3):386-93. Epub 2006 Oct 11.

Medicinal Chemistry Division, Central Drug Research Institute, Chattar Manzil Palace, Lucknow 226 001, India.

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http://dx.doi.org/10.1016/j.ejmech.2006.08.016DOI Listing
March 2007

Synthesis and QSAR studies on hypotensive 1-[3-(4-substituted phenylthio) propyl]-4-(substituted phenyl) piperazines.

Bioorg Med Chem Lett 2007 Mar 23;17(6):1708-12. Epub 2006 Dec 23.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226001, India.

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http://dx.doi.org/10.1016/j.bmcl.2006.12.072DOI Listing
March 2007

3D QSAR studies on protein tyrosine phosphatase 1B inhibitors: comparison of the quality and predictivity among 3D QSAR models obtained from different conformer-based alignments.

J Chem Inf Model 2006 Nov-Dec;46(6):2579-90

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow, India.

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http://dx.doi.org/10.1021/ci600224nDOI Listing
February 2007

Synthesis of some substituted pyrazinopyridoindoles and 3D QSAR studies along with related compounds: piperazines, piperidines, pyrazinoisoquinolines, and diphenhydramine, and its semi-rigid analogs as antihistamines (H1).

Bioorg Med Chem 2006 Dec 28;14(24):8249-58. Epub 2006 Sep 28.

Medicinal and Process Chemistry Division, Central Drug Research Institute, Lucknow 226001, India.

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http://dx.doi.org/10.1016/j.bmc.2006.09.018DOI Listing
December 2006

Enhancing the survival of tunneled haemodialysis catheters using an antibiotic lock in the elderly: a randomised, double-blind clinical trial.

Nephrology (Carlton) 2006 Aug;11(4):299-305

Division of Nephrology, Postgraduate Department of Medicine, King Fahad Hospital and Tertiary Care Centre, Hofuf, Eastern Province, Saudi Arabia.

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http://dx.doi.org/10.1111/j.1440-1797.2006.00563.xDOI Listing
August 2006

Evaluation of binary QSAR models derived from LUDI and MOE scoring functions for structure based virtual screening.

J Chem Inf Model 2006 Jan-Feb;46(1):39-51

Medicinal and Process Chemistry Division, Central Drug Research Institute, Chatter Manzil Palace, Lucknow, India.

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http://dx.doi.org/10.1021/ci050120wDOI Listing
April 2006

The impact of catheter-restricted filling with cefotaxime and heparin on the lifespan of temporary hemodialysis catheters: a case controlled study.

J Nephrol 2005 Nov-Dec;18(6):755-63

Division of Nephrology, Post-graduate Department of Medicine, King Fahad Hospital and Tertiary Care Center, King Faisal University, Eastern Province - Saudi Arabia.

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January 2006

Prevalence of methicillin-resistant and methicillin-sensitive Staphylococcus aureus nasal colonization among patients at the time of admission to the hospital.

Ann Saudi Med 2005 Jul-Aug;25(4):304-8

Department of Infection Control, King Fahad Hospital & Tertiary Care Centre, Al Hofuf, Al Hasa, Saudi Arabia.

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http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6148020PMC
http://dx.doi.org/10.5144/0256-4947.2005.304DOI Listing
December 2005

Cardiovascular mortality and dialysis access-related infections: is there a link?

Am J Kidney Dis 2005 Dec;46(6):1149-50

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http://dx.doi.org/10.1053/j.ajkd.2005.08.035DOI Listing
December 2005

Utility of cefoxitin resistance determination by disk diffusion method for routine detection of methicillin resistant Staphylococcus aureus.

Saudi Med J 2005 Dec;26(12):1999-2000

Department of Infection Control, Internal Medicine, Surgery, King Fahad Hospital, Al-Hofuf, Al-Hasa 31982, Kingdom of Saudi Arabia.

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December 2005

"Uremic pruritus": a misnomer.

Authors:
Anil K Saxena

Hemodial Int 2005 Oct;9(4):416-7

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http://dx.doi.org/10.1111/j.1542-4758.2005.01161.xDOI Listing
October 2005

Contamination of patients' files in intensive care units: an indication of strict handwashing after entering case notes.

Am J Infect Control 2005 Sep;33(7):398-401

Department of Infection Control, King Fahad Hospital, Al-Hofuf, Saudi Arabia.

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http://dx.doi.org/10.1016/j.ajic.2004.12.009DOI Listing
September 2005

Chloramphenicol susceptible methicillin resistant Staphylococcus aureus in eastern region of Saudi Arabia.

Saudi Med J 2005 Jul;26(7):1149-51

Department of Infection Control, King Fahad Hospital, Al-Hofuf, Al-Hasa 31982, Kingdom of Saudi Arabia.

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July 2005

Prevention of catheter-related bloodstream infections: an appraisal of developments in designing an infection-resistant 'dream dialysis-catheter'.

Nephrology (Carlton) 2005 Jun;10(3):240-8

Division of Nephrology, Postgraduate Department of Medicine and Microbiology, King Fahad Hospital & Tertiary Care Centre, Hofuf, King Faisal University, Al-Hasa, Saudi Arabia.

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http://dx.doi.org/10.1111/j.1440-1797.2005.00382.xDOI Listing
June 2005

Haemodialysis catheter-related bloodstream infections: current treatment options and strategies for prevention.

Swiss Med Wkly 2005 Mar;135(9-10):127-38

Division of Nephrology, King Faizal University, King Fahad Hospital, Hofuf, Al-Hasa, Saudi Arabia.

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http://dx.doi.org/2005/09/smw-10860DOI Listing
March 2005

Characterization of beta3-adrenergic receptor: determination of pharmacophore and 3D QSAR model for beta3 adrenergic receptor agonism.

J Comput Aided Mol Des 2005 Feb;19(2):93-110

Division of Medicinal and Process Chemistry, Central Drug Research Institute, 226001, Lucknow, India.

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http://dx.doi.org/10.1007/s10822-005-1558-7DOI Listing
February 2005