Amol Gupte

Amol Gupte

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Amol Gupte

Amol Gupte

Publications by authors named "Amol Gupte"

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Synthesis and evaluation of cyclohexane carboxylic acid head group containing isoxazole and thiazole analogs as DGAT1 inhibitors.

Eur J Med Chem 2014 May 28;79:203-15. Epub 2014 Mar 28.

Department of Medicinal Chemistry, Piramal Enterprises Limited, 1-Nirlon Complex, Goregaon (E), Mumbai 400063, India. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2014.03.077DOI Listing
May 2014

Copper(II)-Catalyzed Conversion of Aryl/Heteroaryl Boronic Acids, Boronates, and Trifluoroborates into the Corresponding Azides: Substrate Scope and Limitations.

Synthesis (Stuttg) 2010 May;2010(9):1441-1448

Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN 55455, USA, Fax +1(612)6265173;

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http://dx.doi.org/10.1055/s-0029-1218683DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2879648PMC
May 2010

Synthesis and biological evaluation of phloridzin analogs as human concentrative nucleoside transporter 3 (hCNT3) inhibitors.

Bioorg Med Chem Lett 2009 Feb 6;19(3):917-21. Epub 2008 Dec 6.

Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Sciences Center, 847 Monroe Avenue Suite 327, Memphis, TN 38163, USA.

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http://dx.doi.org/10.1016/j.bmcl.2008.11.112DOI Listing
February 2009

CoMFA and CoMSIA 3D-QSAR studies on S(6)-(4-nitrobenzyl)mercaptopurine riboside (NBMPR) analogs as inhibitors of human equilibrative nucleoside transporter 1 (hENT1).

Bioorg Med Chem Lett 2009 Jan 27;19(2):314-8. Epub 2008 Nov 27.

Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Sciences Center, 847 Monroe Avenue Suite 327, Memphis, TN 38163, USA.

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http://dx.doi.org/10.1016/j.bmcl.2008.11.092DOI Listing
January 2009

Synthesis of deuterium-labelled 5'-O-[N-(Salicyl)sulfamoyl]adenosine (Sal-AMS-d(4)) as an internal standard for quantitation of Sal-AMS.

J Labelled Comp Radiopharm 2008 Feb;51(2):118-122

Center for Drug Design, Academic Health Center, University of Minnesota, Minneapolis, MN 55455, USA.

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http://dx.doi.org/10.1002/jlcr.1490DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2367327PMC
February 2008

Novel C2-purine position analogs of nitrobenzylmercaptopurine riboside as human equilibrative nucleoside transporter 1 inhibitors.

Bioorg Med Chem 2007 Dec 1;15(24):7726-37. Epub 2007 Sep 1.

Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Sciences Center, 847 Monroe Avenue Suite 327, Memphis, TN 38163, USA.

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http://dx.doi.org/10.1016/j.bmc.2007.08.058DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2692207PMC
December 2007

6-Benzylthioinosine analogues: promising anti-toxoplasmic agents as inhibitors of the mammalian nucleoside transporter ENT1 (es).

Biochem Pharmacol 2005 Dec 23;71(1-2):69-73. Epub 2005 Nov 23.

Department of Pharmaceutical Sciences, College of Pharmacy, 847 Monroe Avenue, Suite 327, University of Tennessee Health Sciences Center, Memphis, TN 38163, USA.

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http://linkinghub.elsevier.com/retrieve/pii/S000629520500702
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http://dx.doi.org/10.1016/j.bcp.2005.10.031DOI Listing
December 2005

Novel halogenated nitrobenzylthioinosine analogs as es nucleoside transporter inhibitors.

Bioorg Med Chem Lett 2004 May;14(9):2257-60

Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Sciences Center, 847 Monroe Avenue Suite 327, Memphis, TN 38163, USA.

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http://dx.doi.org/10.1016/j.bmcl.2004.02.016DOI Listing
May 2004