Alan Whitehead

Alan Whitehead

UNVERIFIED PROFILE

Are you Alan Whitehead?   Register this Author

Register author
Alan Whitehead

Alan Whitehead

Publications by authors named "Alan Whitehead"

Are you Alan Whitehead?   Register this Author

10Publications

118Reads

44Profile Views

Selective Formation of Functionalized α-Quaternary Malononitriles toward 5,5-Disubstituted Pyrrolopyrimidinones.

Org Lett 2017 09 16;19(17):4448-4451. Epub 2017 Aug 16.

Discovery Chemistry, Merck & Co., Inc. , 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/acs.orglett.7b01930DOI Listing
September 2017

Synthesis of the Paralytic Shellfish Poisons (+)-Gonyautoxin 2, (+)-Gonyautoxin 3, and (+)-11,11-Dihydroxysaxitoxin.

J Am Chem Soc 2016 05 3;138(18):5994-6001. Epub 2016 May 3.

Department of Chemistry, Stanford University , Stanford, California 94305-0080, United States.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/jacs.6b02343DOI Listing
May 2016

Evaluation of selective inhibitors of 11β-HSD1 for the treatment of hypertension.

Bioorg Med Chem Lett 2013 Jun 22;23(12):3650-3. Epub 2013 Mar 22.

Department of Medicinal Chemistry, Merck & Co., Inc., PO Box 2000, Rahway, NJ 07065, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1016/j.bmcl.2013.03.011DOI Listing
June 2013

Total synthesis of dolabelide C: a phosphate-mediated approach.

J Org Chem 2011 Jun 29;76(11):4358-70. Epub 2011 Apr 29.

Department of Chemistry, University of Kansas, Lawrence, Kansas 66045, United States.

View Article

Download full-text PDF

Source
http://pubs.acs.org/doi/abs/10.1021/jo2003506
Publisher Site
http://dx.doi.org/10.1021/jo2003506DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC3150593PMC
June 2011

A multifaceted phosphate tether: application to the C15-C30 subunit of dolabelides A-D.

Org Lett 2008 Apr 7;10(7):1421-4. Epub 2008 Mar 7.

Department of Chemistry, University of Kansas, 1251 Wescoe Hall Drive, Lawrence, Kansas 66045, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/ol8001865DOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2641022PMC
April 2008

Synthesis of novel and uniquely shaped 3-azabicyclo[4.2.0]octan-4-one derivatives by sequential Ugi/[2+2] ene-enone photocycloadditions.

Org Lett 2007 Mar 27;9(7):1299-302. Epub 2007 Feb 27.

Scaffold Oriented Synthesis and Structural Chemistry, Abbott Laboratories, R4CP, AP10, Abbott Park, IL 60064-6099, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/ol070164lDOI Listing
March 2007

Divalent activation in temporary phosphate tethers: highly selective cuprate displacement reactions.

Org Lett 2006 Oct;8(22):5025-8

Department of Chemistry, University of Kansas, 1251 Wescoe Hall Drive, Lawrence, KS 66045-7582, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/ol061756rDOI Listing
October 2006

Multivalent activation in temporary phosphate tethers: a new tether for small molecule synthesis.

Org Lett 2005 Jul;7(15):3375-8

Department of Chemistry, University of Kansas, Lawrence, 66045-7582, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/ol0512886DOI Listing
July 2005

P-heterocyclic building blocks: application to the stereoselective synthesis of P-sugars.

J Org Chem 2005 Jul;70(15):5880-9

Department of Chemistry, 1251 Wescoe Hall Drive, Malott Hall, University of Kansas, Lawrence, KS 66045-7582, USA.

View Article

Download full-text PDF

Source
http://dx.doi.org/10.1021/jo0505122DOI Listing
July 2005