Publications by authors named "Abderrahman El Bouakher"

8Publications

Pyrrolo-imidazo[1,2-]pyridine Scaffolds through a Sequential Coupling of -Tosylhydrazones with Imidazopyridines and Reductive Cadogan Annulation, Synthetic Scope, and Application.

J Org Chem 2019 11 9;84(21):13807-13823. Epub 2019 Oct 9.

BioCIS UMR 8076, Université Paris-Sud, CNRS, Université Paris-Saclay, Equipe Labellisée Ligue Contre Le Cancer, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie , 5 rue J.-B. Clément , F-92296 Châtenay-Malabry , France.

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http://dx.doi.org/10.1021/acs.joc.9b02018DOI Listing
November 2019

α-Halogenoacetamides: versatile and efficient tools for the synthesis of complex aza-heterocycles.

Org Biomol Chem 2019 09;17(37):8467-8485

Normandie Univ, UNILEHAVRE, FR 3038 CNRS, URCOM, 76600 Le Havre, France.

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http://xlink.rsc.org/?DOI=C9OB01683J
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http://dx.doi.org/10.1039/c9ob01683jDOI Listing
September 2019

Synthetic Modification of 9α- and 9β-Hydroxyparthenolide by Heck or Acylation Reactions and Evaluation of Cytotoxic Activities.

Planta Med 2017 May 5;83(7):661-671. Epub 2016 Dec 5.

Laboratoire de Chimie Physique & de Chimie Bioorganique, URAC 22, Université Hassan II Casablanca, Mohammedia, Morocco.

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http://dx.doi.org/10.1055/s-0042-119864DOI Listing
May 2017

Synthesis of Oxazolidin-4-ones: Domino O-Alkylation/Aza-Michael/Intramolecular Retro-Claisen Condensation.

Org Lett 2016 05 29;18(10):2383-6. Epub 2016 Apr 29.

Normandie Université , UNIHAVRE, URCOM, 76600 Le Havre 25, Rue Philipe Lebon, BP 540, F-76600 Le Havre, France.

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http://dx.doi.org/10.1021/acs.orglett.6b00851DOI Listing
May 2016

Sequential Friedel-Crafts-Type α-Amidoalkylation/Intramolecular Hydroarylation: Distinct Advantage of Combined Tf2NH/Cationic LAu(I) as a Consecutive or Binary Bicatalytic System.

Org Lett 2015 May 15;17(9):2130-3. Epub 2015 Apr 15.

†Unité de Recherche en Chimie Organique et Macromoléculaire (URCOM, EA 3221, FR CNRS 3038), Faculté des Sciences et Techniques, l'Université du Havre, 25 rue Philippe Lebon, BP 540, Le Havre 76058 Cedex, France.

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http://dx.doi.org/10.1021/acs.orglett.5b00718DOI Listing
May 2015

Synthesis and biological evaluation of 9α- and 9β-hydroxyamino-parthenolides as novel anticancer agents.

Bioorg Med Chem Lett 2014 Aug 14;24(16):4014-8. Epub 2014 Jun 14.

Laboratoire de Chimie Physique & de Chimie Bioorganique, URAC 22, Université Hassan II Mohammedia-Casablanca, BP 146, 28800 Mohammedia, Morocco. Electronic address:

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http://dx.doi.org/10.1016/j.bmcl.2014.06.019DOI Listing
August 2014