Publications by authors named "Abdallah Hamze"

57Publications

Sequential One-Pot Synthesis of 3-Arylbenzofurans from -Tosylhydrazones and Bromophenol Derivatives.

J Org Chem 2020 Nov 22;85(21):13664-13673. Epub 2020 Oct 22.

Université Paris-Saclay, CNRS, BioCIS, 92290 Châtenay-Malabry, France.

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http://dx.doi.org/10.1021/acs.joc.0c01835DOI Listing
November 2020

Cyclic bridged analogs of isoCA-4: Design, synthesis and biological evaluation.

Eur J Med Chem 2020 Oct 4;209:112873. Epub 2020 Oct 4.

Université Paris-Saclay, CNRS, BioCIS, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2020.112873DOI Listing
October 2020

An update on the use of sulfinate derivatives as versatile coupling partners in organic chemistry.

Org Biomol Chem 2020 Nov;18(45):9136-9159

Université Paris-Saclay, CNRS, BioCIS, 92290, Châtenay-Malabry, France.

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http://dx.doi.org/10.1039/d0ob01718cDOI Listing
November 2020

Identification of a new series of flavopiridol-like structures as kinase inhibitors with high cytotoxic potency.

Eur J Med Chem 2020 Aug 5;199:112355. Epub 2020 May 5.

BioCIS, Equipe Labellisée Ligue Contre le Cancer, Univ. Paris-Sud, CNRS, University Paris-Saclay, F-92290, Châtenay Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2020.112355DOI Listing
August 2020

How do we improve histone deacetylase inhibitor drug discovery?

Authors:
Abdallah Hamze

Expert Opin Drug Discov 2020 May 2;15(5):527-529. Epub 2020 Mar 2.

Equipe Labellisée Ligue Contre Le Cancer, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, BioCIS UMR 8076, Université Paris-Sud, CNRS, Université Paris-Saclay, Chatenay-Malabry, France.

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http://dx.doi.org/10.1080/17460441.2020.1736032DOI Listing
May 2020

Developments of isoCombretastatin A-4 derivatives as highly cytotoxic agents.

Eur J Med Chem 2020 Mar 30;190:112110. Epub 2020 Jan 30.

Université Paris-Saclay, CNRS, BioCIS, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2020.112110DOI Listing
March 2020

Toward a Greener Barluenga-Valdés Cross-Coupling: Microwave-Promoted C-C Bond Formation with a Pd/PEG/HO Recyclable Catalytic System.

Org Lett 2019 11 16;21(21):8708-8712. Epub 2019 Oct 16.

BioCIS UMR 8076 , Université Paris-Sud, CNRS, Université Paris-Saclay, Equipe Labellisée Ligue Contre Le Cancer, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie , rue J.-B. Clément , F-92296 Châtenay-Malabry , France.

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http://dx.doi.org/10.1021/acs.orglett.9b03310DOI Listing
November 2019

Pyrrolo-imidazo[1,2-]pyridine Scaffolds through a Sequential Coupling of -Tosylhydrazones with Imidazopyridines and Reductive Cadogan Annulation, Synthetic Scope, and Application.

J Org Chem 2019 11 9;84(21):13807-13823. Epub 2019 Oct 9.

BioCIS UMR 8076, Université Paris-Sud, CNRS, Université Paris-Saclay, Equipe Labellisée Ligue Contre Le Cancer, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie , 5 rue J.-B. Clément , F-92296 Châtenay-Malabry , France.

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http://dx.doi.org/10.1021/acs.joc.9b02018DOI Listing
November 2019

N,N-bis-heteroaryl methylamines: Potent anti-mitotic and highly cytotoxic agents.

Eur J Med Chem 2019 Apr 16;168:176-188. Epub 2019 Feb 16.

BioCIS, Univ. Paris-Sud, CNRS, Université Paris-Saclay, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2019.02.038DOI Listing
April 2019

One-Pot Reaction between N-Tosylhydrazones and 2-Nitrobenzyl Bromide: Route to NH-Free C2-Arylindoles.

J Org Chem 2019 01 17;84(1):228-238. Epub 2018 Dec 17.

LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie , Université Paris-Sud, CNRS, BioCIS-UMR 8076 , rue J.-B. Clément , Châtenay-Malabry F-92296 , France.

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http://dx.doi.org/10.1021/acs.joc.8b02623DOI Listing
January 2019

1,1-Diheterocyclic Ethylenes Derived from Quinaldine and Carbazole as New Tubulin-Polymerization Inhibitors: Synthesis, Metabolism, and Biological Evaluation.

J Med Chem 2019 02 21;62(4):1902-1916. Epub 2018 Dec 21.

BioCIS, Université Paris-Sud, CNRS, Équipe Labellisée Ligue Contre le Cancer , Université Paris-Saclay , F-92290 Châtenay-Malabry , France.

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http://dx.doi.org/10.1021/acs.jmedchem.8b01386DOI Listing
February 2019

Design, synthesis and anticancer properties of IsoCombretaQuinolines as potent tubulin assembly inhibitors.

Eur J Med Chem 2017 Feb 9;127:1025-1034. Epub 2016 Nov 9.

BioCIS, Univ. Paris-Sud, CNRS, Université Paris-Saclay, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2016.11.012DOI Listing
February 2017

A general synthesis of arylindoles and (1-arylvinyl)carbazoles via a one-pot reaction from N-tosylhydrazones and 2-nitro-haloarenes and their potential application to colon cancer.

Chem Commun (Camb) 2016 Oct;52(88):13027-13030

BioCIS, Equipe Labellisée Ligue Contre le Cancer, Univ. Paris-Sud, CNRS, University Paris-Saclay, 92290, Châtenay-Malabry, France.

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http://dx.doi.org/10.1039/c6cc07666aDOI Listing
October 2016

Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2-a]pyridines derivatives as protein kinase inhibitors.

Eur J Med Chem 2016 Nov 21;123:105-114. Epub 2016 Jul 21.

BioCIS, Univ. Paris-Sud, CNRS, équipe labellisée Ligue Contre le Cancer, Université Paris-Saclay, 92290, Châtenay-Malabry, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2016.07.040DOI Listing
November 2016

Selective Metal-Free Deoxygenation of Unsymmetrical 1,2-Dicarbonyl Compounds by Chlorotrimethylsilane and Sodium Iodide.

Org Lett 2016 07 23;18(13):3238-41. Epub 2016 Jun 23.

BioCIS, Université Paris-Sud, CNRS, équipe labellisée Ligue Contre le Cancer, Université Paris-Saclay , 92290 Châtenay-Malabry, France.

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http://pubs.acs.org/doi/abs/10.1021/acs.orglett.6b01491
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http://dx.doi.org/10.1021/acs.orglett.6b01491DOI Listing
July 2016

Anti-Tumoral Effects of Anti-Progestins in a Patient-Derived Breast Cancer Xenograft Model.

Horm Cancer 2016 Apr 3;7(2):137-47. Epub 2016 Mar 3.

Service de Gynécologie Obstétrique Médecine de la Reproduction, Hôpitaux Universitaires Est Parisien site Tenon, Assistance Publique-Hôpitaux de Paris, 4 Rue de la Chine, 75020, Paris, France.

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http://dx.doi.org/10.1007/s12672-016-0255-4DOI Listing
April 2016

Palladium-Catalyzed One-Pot Reaction of Hydrazones, Dihaloarenes, and Organoboron Reagents: Synthesis and Cytotoxic Activity of 1,1-Diarylethylene Derivatives.

J Org Chem 2015 Jul 12;80(13):6715-27. Epub 2015 Jun 12.

†Université Paris-Sud, CNRS, BioCIS-UMR 8076, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, rue J.-B. Clément, F-92296 Châtenay-Malabry, France.

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http://dx.doi.org/10.1021/acs.joc.5b00880DOI Listing
July 2015

Stereoretentive palladium-catalyzed arylation, alkenylation, and alkynylation of 1-thiosugars and thiols using aminobiphenyl palladacycle precatalyst at room temperature.

Chemistry 2015 Jun 15;21(23):8375-9. Epub 2015 Apr 15.

Univ. Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, 92296 (France).

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http://dx.doi.org/10.1002/chem.201501050DOI Listing
June 2015

Rapid synthesis of 4-arylchromenes from ortho-substituted alkynols: A versatile access to restricted isocombretastatin A-4 analogues as antitumor agents.

Eur J Med Chem 2015 Jan 15;90:834-44. Epub 2014 Dec 15.

University Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre Le Cancer, LabEx LERMIT, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry F-92296, France. Electronic address:

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http://dx.doi.org/10.1016/j.ejmech.2014.12.024DOI Listing
January 2015

Sulfinate derivatives: dual and versatile partners in organic synthesis.

Org Biomol Chem 2014 Dec;12(48):9743-59

Univ Paris Sud, CNRS, BioCIS UMR 8076, Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT, Faculté de Pharmacie, 5 rue J-B Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1039/c4ob01727gDOI Listing
December 2014

Synthesis of a 3-(α-styryl)benzo[b]-thiophene library via bromocyclization of alkynes and palladium-catalyzed to sylhydrazones cross-couplings: evaluation as antitubulin agents.

ACS Comb Sci 2014 Dec 25;16(12):702-10. Epub 2014 Sep 25.

Univ Paris Sud, CNRS, BioCIS-UMR 8076 , Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/co500115bDOI Listing
December 2014

Tandem one-pot palladium-catalyzed coupling of hydrazones, haloindoles, and amines: synthesis of amino-N-vinylindoles and their effect on human colon carcinoma cells.

J Org Chem 2014 Aug 29;79(16):7583-92. Epub 2014 Jul 29.

Laboratoire de Chimie Thérapeutique, Equipe Labellisée Ligue Contre le Cancer, LabEx LERMIT, Faculté de Pharmacie, Université Paris-Sud , CNRS, BioCIS-UMR 8076, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296 Paris, France.

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http://dx.doi.org/10.1021/jo501315qDOI Listing
August 2014

Therapeutic modalities of squalenoyl nanocomposites in colon cancer: an ongoing search for improved efficacy.

ACS Nano 2014 Mar 26;8(3):2018-32. Epub 2014 Feb 26.

Faculté de Pharmacie, Université Paris-Sud , Institut Galien Paris Sud, UMR CNRS 8612, 5 rue J.-B. Clément, Châtenay-Malabry, Paris, F-92296, France.

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http://dx.doi.org/10.1021/nn500517aDOI Listing
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4060170PMC
March 2014

Discovery and hit to lead optimization of novel combretastatin A-4 analogues: dependence of C-linker length and hybridization.

Anticancer Agents Med Chem 2013 Dec;13(10):1614-35

Univ. Paris-Sud 11, CNRS, BioCIS-UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.2174/187152061310131206162302DOI Listing
December 2013

Csp2-N bond formation via ligand-free Pd-catalyzed oxidative coupling reaction of N-tosylhydrazones and indole derivatives.

J Org Chem 2013 Sep 14;78(17):8485-95. Epub 2013 Aug 14.

Université Paris-Sud, CNRS, BioCIS-UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/jo401217xDOI Listing
September 2013

An efficient coupling of N-tosylhydrazones with 2-halopyridines: synthesis of 2-α-styrylpyridines endowed with antitumor activity.

Org Biomol Chem 2013 Jun;11(22):3664-73

Université Paris-Sud, CNRS, BioCIS UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J-B Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1039/c3ob40263kDOI Listing
June 2013

Design, synthesis and anticancer properties of 5-arylbenzoxepins as conformationally restricted isocombretastatin A-4 analogs.

Eur J Med Chem 2013 Apr 4;62:28-39. Epub 2013 Jan 4.

Univ. Paris-Sud, CNRS, BioCIS-UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry F-92296, France.

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http://dx.doi.org/10.1016/j.ejmech.2012.12.042DOI Listing
April 2013

Catalytic three-component one-pot reaction of hydrazones, dihaloarenes, and amines.

Org Lett 2013 Jan 18;15(1):148-51. Epub 2012 Dec 18.

Univ Paris-Sud , CNRS, BioCIS UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 Rue J. B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/ol303194sDOI Listing
January 2013

Synthesis of ortho/ortho'-substituted 1,1-diarylethylenes through cross-coupling reactions of sterically encumbered hydrazones and aryl halides.

J Org Chem 2013 Jan 3;78(2):445-54. Epub 2013 Jan 3.

Université Paris-Sud, CNRS, BioCIS-UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/jo3023268DOI Listing
January 2013

Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors.

Org Biomol Chem 2013 Jan 9;11(3):430-42. Epub 2012 Oct 9.

Université Paris-Sud, CNRS, BioCIS UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J-B Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1039/c2ob26253cDOI Listing
January 2013

Synthesis of 1,1-diarylethylenes via efficient iron/copper co-catalyzed coupling of 1-arylvinyl halides with Grignard reagents.

Org Lett 2012 Jun 22;14(11):2782-5. Epub 2012 May 22.

Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, Université Paris-Sud, CNRS, BioCIS UMR 8076, LabEx LERMIT, 5 Rue J. B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/ol3010112DOI Listing
June 2012

Conformationnally restricted naphthalene derivatives type isocombretastatin A-4 and isoerianin analogues: synthesis, cytotoxicity and antitubulin activity.

Eur J Med Chem 2012 Jun 9;52:22-32. Epub 2012 Mar 9.

Univ. Paris-Sud, CNRS, BioCIS-UMR 8076, LabEx LERMIT, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry F-92296, France.

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http://dx.doi.org/10.1016/j.ejmech.2012.03.001DOI Listing
June 2012

B-ring-modified isocombretastatin A-4 analogues endowed with interesting anticancer activities.

ChemMedChem 2011 Dec 11;6(12):2179-91. Epub 2011 Oct 11.

Université Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, 92296, France.

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http://dx.doi.org/10.1002/cmdc.201100325DOI Listing
December 2011

Copper-catalyzed reductive coupling of tosylhydrazones with amines: a convenient route to α-branched amines.

Org Biomol Chem 2011 Sep 28;9(18):6200-4. Epub 2011 Jul 28.

Université Paris-Sud 11, CNRS, BioCIS UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, Châtenay-Malabry, France.

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http://dx.doi.org/10.1039/c1ob05664fDOI Listing
September 2011

Discovery of isoerianin analogues as promising anticancer agents.

ChemMedChem 2011 Mar 14;6(3):488-97. Epub 2011 Jan 14.

Université Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 Rue J.-B. Clément, Châtenay-Malabry, 92296, France.

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http://dx.doi.org/10.1002/cmdc.201000456DOI Listing
March 2011

Cyclic peptides with a diversely substituted guanidine bridge: solid-phase synthesis and structural analysis.

Chemistry 2011 Feb 3;17(9):2566-70. Epub 2011 Feb 3.

Institut des Biomolécules Max Mousseron, CNRS UMR5247, Université Montpellier 1, Université Montpellier 2, Faculté de Pharmacie, Montpellier, France.

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http://dx.doi.org/10.1002/chem.201003299DOI Listing
February 2011

Pd-catalyzed reaction of sterically hindered hydrazones with aryl halides: synthesis of tetra-substituted olefins related to iso-combretastatin A4.

Org Lett 2010 Sep;12(18):4042-5

University Paris-Sud 11, CNRS, BioCIS UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry F-92296, France.

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http://dx.doi.org/10.1021/ol101639gDOI Listing
September 2010

Regioselective hydrostannation of diarylalkynes directed by a labile ortho bromine atom: an easy access to stereodefined triarylolefins, hybrids of combretastatin A-4 and isocombretastatin A-4.

Eur J Med Chem 2010 Sep 12;45(9):3617-26. Epub 2010 May 12.

University Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1016/j.ejmech.2010.05.007DOI Listing
September 2010

Solid-phase synthesis of dipeptidic and pseudo-dipeptidic potential NOS inhibitors through a side-chain anchoring approach.

Adv Exp Med Biol 2009 ;611:133-4

Institut des Biomolécules Max Mousseron, CNRS UMR5247, Université Montpellier 1, Faculté de Pharmacie, 15 avenue Charles Flahault, 34093 Montpellier cedex 5, France.

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http://dx.doi.org/10.1007/978-0-387-73657-0_59DOI Listing
June 2009

Palladium-catalyzed Markovnikov terminal arylalkynes hydrostannation: application to the synthesis of 1,1-diarylethylenes.

J Org Chem 2009 Feb;74(3):1337-40

Laboratoire de Chimie Therapeutique, Faculte de Pharmacie, Universite Paris-Sud, CNRS, BioCIS, UMR 8076, rue J. B. Clement, Chatenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/jo802460zDOI Listing
February 2009

Synthesis and antitumor activity of benzils related to combretastatin A-4.

Bioorg Med Chem Lett 2008 Jun 25;18(11):3266-71. Epub 2008 Apr 25.

Univ Paris-Sud, CNRS, BioCIS-UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, rue J.B. Clément, F-92296 Châtenay-Malabry, France.

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http://dx.doi.org/10.1016/j.bmcl.2008.04.053DOI Listing
June 2008

Regiocontrol of the palladium-catalyzed tin hydride addition to Z-enynols: remarkable Z-directing effects.

J Org Chem 2007 May 14;72(10):3868-74. Epub 2007 Apr 14.

Univ Paris-Sud, and CNRS, BioCIS UMR 8076, Laboratoire de Chimie Thérapeutique, Faculté de Pharmacie, 5 rue J.-B. Clément, Châtenay-Malabry, F-92296, France.

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http://dx.doi.org/10.1021/jo0701435DOI Listing
May 2007

Platinum oxide catalyzed silylation of aryl halides with triethylsilane: an efficient synthetic route to functionalized aryltriethylsilanes.

Org Lett 2006 Mar;8(5):931-4

Laboratoire de Chimie Thérapeutique, BioCIS - CNRS (UMR 8076), Université Paris-Sud XI, Faculté de Pharmacie, rue J.B. Clément, 92296 Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1021/ol052996uDOI Listing
March 2006

Platinum oxide catalyzed hydrosilylation of unsymmetrical internal aryl alkynes under ortho-substituent regiocontrol.

Org Lett 2005 Dec;7(25):5625-8

Laboratoire de Chimie Thérapeutique, BioCIS - CNRS (UMR 8076), Université Paris-Sud XI, Faculté de Pharmacie, rue J.B. Clément, 92296 Châtenay-Malabry Cedex, France.

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http://dx.doi.org/10.1021/ol052245sDOI Listing
December 2005

Mono- and bis-thiazolium salts have potent antimalarial activity.

J Med Chem 2005 May;48(10):3639-43

Laboratoire des Amino acides Peptides et Protéines (LAPP) CNRS-UMR 5810, CP 19, Université Montpellier I, Place E. Bataillon, 34095 Montpellier Cedex 5, France.

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http://dx.doi.org/10.1021/jm0492608DOI Listing
May 2005

Dual molecules as new antimalarials.

Comb Chem High Throughput Screen 2005 Feb;8(1):49-62

CNRS UMR 5810, Université de Montpellier II, CP 22, Place Eugène Bataillon, F- 34095 Montpellier Cedex 5, France.

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http://dx.doi.org/10.2174/1386207053328219DOI Listing
February 2005

Solid-phase synthesis of arginine-containing peptides and fluorogenic substrates using a side-chain anchoring approach.

J Org Chem 2004 Nov;69(24):8394-402

Laboratoire des Aminoacides Peptides et Protéines, CNRS UMR 5810, Universités Montpellier I et II, Faculté de Pharmacie, 15 avenue Charles Flahault, BP 14491, 34093 Montpellier cédex 5, France.

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http://dx.doi.org/10.1021/jo048792tDOI Listing
November 2004

Synthesis of various 3-substituted 1,2,4-oxadiazole-containing chiral beta 3- and alpha-amino acids from Fmoc-protected aspartic acid.

J Org Chem 2003 Sep;68(19):7316-21

Laboratoire des Aminoacides Peptides et Protéines, CNRS UMR 5810, Universités Montpellier I et II, Faculté de Pharmacie, 15 avenue Charles Flahault, BP 14491, 34093 Montpellier cédex 5, France.

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http://dx.doi.org/10.1021/jo0345953DOI Listing
September 2003